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6-[(4aS,8aR)-1-[3-(methylsulfanyl)propyl]-2-oxo-decahydro-1,6-naphthyridin-6-yl]pyridine-2-carbonitrile
N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]-1,3-thiazole-4-carboxamide
3-(3-methyl-1H-pyrazol-1-yl)-1-[2-(piperidin-1-ylmethyl)-1,4-oxazepan-4-yl]propan-1-one
N-[1-(2,5-difluorophenyl)cyclopropyl]-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
2-methoxy-4-(2-phenoxyethyl)pyridine-3-carbonitrile
4-(4-{2-[2-(dimethylamino)ethyl]morpholine-4-carbonyl}phenyl)-2-methylbut-3-yn-2-ol
N-(2-methanesulfonamidoethyl)-3-methyl-2-[(quinazolin-4-yl)amino]butanamide
4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(1H-indol-3-yl)ethyl]acetamide
9-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-N-{[8-(3-phenylpropyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-1,3-thiazole-4-carboxamide
4-(4-{[4-(1H-imidazol-1-yl)phenyl]methyl}-2-oxopiperazin-1-yl)benzonitrile
4-{[1-(3-ethoxypropanoyl)pyrrolidin-3-yl]methyl}benzoic acid
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-5-methyl-1,2-oxazole-3-carboxamide
3-{[(2-methoxyethyl)(1,3-thiazol-2-ylmethyl)amino]methyl}-1,2-dihydroquinolin-2-one
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-2-ethyl-1-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
N-(3-fluorophenyl)-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
4-(2-methoxyphenoxy)-1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidine
1-(furan-3-ylmethyl)-N-[3-(1H-indol-2-yl)phenyl]piperidine-4-carboxamide
1-({5-[(3-hydroxy-4-methoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
2-{2-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}benzamide
3-({2-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}methyl)-1λ6-thiolane-1,1-dione
1-(2-methoxy-5-methylphenyl)-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
N-butyl-N-[(4-fluorophenyl)methyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
N-[1-(pyrazin-2-yl)piperidin-3-yl]pyridine-4-carboxamide
N-methyl-N-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
1-[2-(4-methoxyphenyl)ethyl]-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
methyl 5-oxo-5-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}pentanoate
3,5-dimethyl-1-{1-[(2,3,4-trifluorophenyl)methyl]pyrrolidin-3-yl}-1H-pyrazole
(4aS,7aR)-1-(2-oxo-1,2-dihydroquinoline-4-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-3-(1-methylpiperidin-2-yl)propanamide
N-[4-(5-methylfuran-3-amido)phenyl]piperidine-4-carboxamide
N-(prop-2-en-1-yl)-N-(pyridin-2-ylmethyl)-3-(4H-1,2,4-triazol-4-yl)benzamide
methyl (2S,4S)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(4-methoxy-2,3-dimethylphenyl)methyl]pyrrolidine-2-carboxylate
3-[2-(5-benzyl-4-phenyl-1H-imidazol-1-yl)ethyl]-1,3-oxazolidin-2-one
3-(azepane-1-carbonyl)-N-cyclopentyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-[2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]piperazin-2-one
(3S,4R)-1-(4-methyl-1,3-thiazole-5-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-2-methoxy-N-methylpyridine-4-carboxamide
2-[4-(2-hydroxyethoxy)phenyl]-1H-1,3-benzodiazole-6-carboxylic acid
N-[(1-{[4-(propan-2-yl)phenyl]methyl}pyrrolidin-3-yl)methyl]cyclopropanesulfonamide
3-methoxy-1-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}-1,2-dihydropyridin-2-one
2-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-3-(piperidine-1-carbonyl)pyrazine
3-methoxy-2-({3-[4-(naphthalen-1-yl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
4-[(5-ethyl-2-methylpyrimidin-4-yl)amino]-1λ6-thiane-1,1-dione
N-[2-(dimethylamino)ethyl]-3-fluoro-N-{[2-(4-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}benzamide
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-cyclopentanecarbonylpiperidine-4-carboxamide
3,4-dimethyl-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]-5-sulfamoylbenzamide
(3S,7S,8aS)-7-{[(3-chloro-1-benzothiophen-2-yl)methyl]amino}-3-methyl-octahydropyrrolo[1,2-a]piperazine-1,4-dione
N-methyl-2-({spiro[azepane-4,2'-chromene]-1-yl}carbonyl)aniline