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(3aS,6aR)-5-(3-phenylpropyl)-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(3R,4R)-1-[(5-chloro-2-hydroxyphenyl)methyl]-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
(2S,4R)-4-{[(3,4-difluorophenyl)methyl]amino}-1-(2,3-dihydro-1H-inden-2-yl)-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
1-{2-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-oxoethyl}piperidin-2-one
4-(benzyloxy)-1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidine
(3S,9aR)-8-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
ethyl 4-[(4-chlorophenyl)methyl]-1-(5-methylpyrazine-2-carbonyl)piperidine-4-carboxylate
methyl 9-(2,3-dihydro-1H-inden-2-yloxy)-3-(oxan-4-yl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-cyclobutanecarbonyl-4-(5,6-dimethylpyrimidin-4-yl)-1,4-diazepane
(3aR,6aS)-N-[5-(cyclopropylcarbamoyl)-2-methoxyphenyl]-octahydropyrrolo[3,4-c]pyrrole-2-carboxamide
(3S,4R)-1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-[2-hydroxy-1-(thian-4-yl)ethyl]-5-phenyl-1,2-oxazole-3-carboxamide
ethyl 1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-(2-phenoxyethyl)piperidine-3-carboxylate
3-(1-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}-1H-imidazol-2-yl)benzonitrile
2-chloro-N-methyl-5-(5-methylfuran-2-yl)benzamide
2-{methyl[4-(morpholin-4-yl)butyl]amino}-2-[4-(propan-2-yloxy)phenyl]acetic acid
1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
1-[3-(1,3-oxazol-5-yl)phenyl]-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}piperidin-4-amine
3-hydroxy-3-{[methyl(thiophen-3-ylmethyl)amino]methyl}-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-3-(3-methylphenoxy)azetidine
1'-(4-methyl-1,3-oxazole-5-carbonyl)-5-(3-methylbut-2-en-1-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
propan-2-yl 3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carboxylate
2-{2-[(dimethylamino)methyl]-4-phenylphenoxy}-N-{[2-(trifluoromethyl)phenyl]methyl}acetamide
1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
5-[1-(5-phenyl-1H-pyrazole-3-carbonyl)pyrrolidin-2-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
2-(pyrazin-2-yl)-1-[(1R,5R)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
2-(5-acetylthiophen-3-yl)-N-[(2,5-difluorophenyl)methyl]acetamide
4-methyl-6-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-1,3-benzothiazol-2-amine
methyl 6-(2-acetylbenzoyl)-2-(pyrrolidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(1R,5R)-6-methyl-3-[1-(3-methylphenyl)piperidin-4-yl]-3,6-diazabicyclo[3.2.2]nonane
4-(2,5-dimethoxyphenyl)-1H-pyrrolo[2,3-b]pyridine
4-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]-2,3,6-trimethylquinoline
1-[(2,3-difluorophenyl)methyl]-4-[1-(4-methyl-1H-imidazole-2-carbonyl)pyrrolidin-3-yl]piperidine
1-cyclobutanecarbonyl-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)piperidine-4-carboxamide
3-(cyclopropylmethyl)-1-(5-methylthiophene-3-carbonyl)piperidine-3-carboxylic acid
N-[2-(dimethylsulfamoyl)ethyl]-1H-imidazole-2-carboxamide
3-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
4-benzyl-3-{1-[2-(ethylsulfanyl)propanoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(1-benzofuran-2-ylmethyl)-octahydropyrrolo[1,2-a]piperazine
methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]{[5-(pyridin-4-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}amine
4-({[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)phenol
3-cyclopropyl-3-[(2-ethoxyphenyl)methyl]-1-(5-fluoropyridin-3-yl)urea
1,7-dimethyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-1H-indole-2-carboxamide
3-{[(1,3-benzoxazol-2-ylmethyl)amino]methyl}-3-hydroxy-1-(2-phenylethyl)piperidin-2-one
2-[(1S,5R)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-3-carbonitrile
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
ethyl 3-benzyl-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidine-3-carboxylate
5-[1-(2-ethylbutyl)-4-hydroxypiperidin-4-yl]-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
N-{4-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]phenyl}-2-(morpholin-4-yl)acetamide
4,6-dimethyl-3-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]-1,2-dihydropyridin-2-one