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1-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]-3-(3-methyl-1-propyl-1H-pyrazol-5-yl)urea
5-{4-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}pentan-1-ol
6-methyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-4-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
1-methyl-8-(6-methyl-2-propylpyrimidin-4-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-methyl-N-[(5-{[3-(2-methylpiperidin-1-yl)azetidin-1-yl]methyl}furan-2-yl)methyl]methanesulfonamide
N-[1-ethyl-2-(2-fluorophenyl)-7-(thiomorpholine-4-carbonyl)-1H-1,3-benzodiazol-5-yl]acetamide
N3-(2-methoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-N5-[(5-methylfuran-2-yl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-ethyl-8-[5-(ethylsulfanyl)thiophene-2-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[4-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)phenyl]imidazolidine-2,4-dione
N-{1-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methylbenzamide
6-fluoro-2-{[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
3-ethyl-5-hydroxy-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]adamantane-1-carboxamide
3-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}urea
1-[(3-chlorophenyl)methyl]-4-[1-(methoxymethyl)cyclobutanecarbonyl]piperazine
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-3,4,7-trimethyl-1H-indole-2-carboxamide
methyl 3-[(4-chlorophenyl)methyl]-9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
1-[2-(2-aminoethyl)quinazolin-4-yl]-4-(piperidin-1-yl)piperidine-4-carboxamide
2-(4-ethylpiperazin-1-yl)-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]acetamide
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-[(propan-2-yloxy)carbonyl]piperidine-4-carboxylic acid
N-(5-chloro-2-methoxyphenyl)-3-[1-(1H-indole-2-carbonyl)piperidin-3-yl]propanamide
2-{3-[(4-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}pyridine-3-carboxamide
methyl N-[1-({[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}carbamoyl)ethyl]carbamate
2-[bis(pyridin-3-ylmethyl)amino]-2-(4-methoxy-3,5-dimethylphenyl)acetic acid
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-2-(methylamino)-1,3-thiazole-4-carboxamide
6-(methoxymethyl)-2-(4-{[methyl(1H-pyrazol-5-ylmethyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
3-(2,3-dihydro-1H-inden-2-yl)-8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{1-[5-(methoxymethyl)thiophene-2-carbonyl]piperidin-3-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
3-methyl-1-{3-methyl-5H,6H-imidazo[2,1-b][1,3]thiazole-2-carbonyl}-3-phenylpiperidine
2-methyl-5-(4-{[(9H-purin-6-yl)amino]methyl}piperidin-1-yl)-2,3-dihydropyridazin-3-one
N-butyl-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
(2S,4S)-4-amino-N-methyl-1-{2-[2-oxo-5-(trifluoromethyl)-1,2-dihydropyridin-1-yl]acetyl}pyrrolidine-2-carboxamide
1-[(5-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}thiophen-3-yl)methyl]piperidine
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(furan-3-carbonyl)pyrrolidin-3-yl]-2-methyl-1,3-thiazole-4-carboxamide
2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}acetamide
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-methylbutan-1-one
(4aR,7aS)-1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[(1S,5R)-6-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
[1-(pyridin-2-ylmethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
7-{2-amino-6-[(4-fluorophenyl)sulfanyl]pyrimidin-4-yl}-2,7-diazaspiro[4.4]nonane-1,3-dione
4-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-2-(2-phenylethyl)morpholine
4-(4-methylpiperazin-1-yl)-6-[2-(2-methylpropoxy)phenyl]pyrimidin-2-amine
4-(4-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane-9-carbonyl}phenyl)-2-methylbutan-2-ol
7-(cyclopropylmethyl)-2-[(3,5-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
3-(2-methoxyethyl)-1-[(4-methoxypyridin-2-yl)methyl]piperidine-3-carboxylic acid
(2R,6R)-11-methoxy-4-[2-(piperidin-1-yl)acetyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-amino-1-{[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]methyl}pyrrolidine-3-carboxylic acid
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-[(5-fluoro-2-methoxyphenyl)methyl]pyrrolidin-3-yl]methanol
N-[(1R,3R)-3-aminocyclopentyl]-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzamide
3-[2-(2,6-difluorophenyl)ethyl]-1-(1-methyl-1H-pyrazole-3-carbonyl)piperidine