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5-cyclobutyl-1-(2-phenylethyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
1-ethyl-3-(propan-2-yl)-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-5-carboxamide
[3-(3-methoxypropyl)-1-(thiophen-3-ylmethyl)piperidin-3-yl]methanol
(3S,9aR)-3-(cyclohexylmethyl)-8-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-{1-[(2-chlorophenyl)methyl]pyrrolidin-3-yl}benzoic acid
N-(3-methoxypropyl)-N-{[6-(2-methylphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-4-(1H-pyrazol-1-yl)benzamide
6-(3-chlorophenyl)-7-(cyclopropylmethyl)-N-(2,2-difluoroethyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-5,6-dimethylpyrimidin-4-amine
3-chloro-N-cyclopentyl-4-{[1-(thiophene-3-carbonyl)piperidin-4-yl]oxy}benzamide
4-cyano-1-methyl-N-[2-(3-phenylpiperidin-1-yl)ethyl]-1H-pyrrole-2-carboxamide
7-fluoro-3-{[methyl({[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl})amino]methyl}-1,2-dihydroquinolin-2-one
4-fluoro-N-[2-(4-{[methyl(naphthalen-1-ylmethyl)amino]methyl}phenoxy)ethyl]benzamide
4-[3-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]quinoline
4-(4-benzyl-1H-pyrazol-5-yl)-1-(1H-pyrrole-2-carbonyl)piperidine
5-[2-(cyclopropylamino)pyrimidin-4-yl]-2-ethoxybenzoic acid
4-(piperidin-1-yl)-1-[2-(pyrrolidin-1-yl)-6-(thiophen-2-yl)pyridine-3-carbonyl]piperidine-4-carboxamide
1-(2-aminoethyl)-N-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
1-[4-(methylsulfanyl)phenyl]-3-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-3-(pyridin-2-ylmethyl)urea
(3aR,6aR)-2-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(2-{7,7-dimethyl-4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl}ethyl)piperidine-4-carboxamide
4-[4-(cycloheptylcarbamoyl)piperidin-1-yl]pyrimidine-5-carboxylic acid
1-amino-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}cyclobutane-1-carboxamide
4-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl}-1-(2-methoxyphenyl)piperazin-2-one
2-(4-{[3-(furan-2-yl)phenyl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
methyl 4-[(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-4-yl)formamido]butanoate
2-cyclopropyl-1-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}ethan-1-one
(4-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}morpholin-2-yl)methanamine
7-{[4-(propan-2-yl)phenyl]methyl}-2-(thian-4-yl)-2,7-diazaspiro[4.5]decan-6-one
2-[3-(cyclopropylmethyl)-5-(methoxymethyl)-1H-1,2,4-triazol-1-yl]benzoic acid
N-benzyl-N-methyl-3-{3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.5]decan-7-yl}propanamide
1-{3-[4-(3-methylphenyl)piperazin-1-yl]propanoyl}piperidine-3-carbonitrile
(3aS,6aR)-N-benzyl-3-[2-(4-methoxyphenyl)ethyl]-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-carboxamide
ethyl 1-[(4-methoxyphenyl)methyl]-5-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(oxolan-2-ylmethyl)({[2-(pyridin-2-yl)pyrimidin-5-yl]methyl})(pyridin-2-ylmethyl)amine
N-(1-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-4-yl)acetamide
5-methyl-5-(1-{[2-(propylamino)pyrimidin-5-yl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
(4aR,7aS)-1-acetyl-4-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(pentan-3-yl)-3-{[2-(1,3-thiazol-4-yl)ethyl]sulfamoyl}benzamide
1-(4-benzylpiperazin-1-yl)-3-[1-(2-methoxypyridine-3-carbonyl)piperidin-3-yl]propan-1-one
3-methyl-7-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N'-(2-fluoro-5-methylphenyl)-N-{2-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}butanediamide
4-methyl-N-(2-methylpropyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-1H-imidazole-2-carboxamide
9-[3-(methylsulfanyl)propyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(2-methoxyethyl)-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-5-oxopyrrolidine-3-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-5-hydroxypyrazine-2-carboxamide
2-(oxolan-2-ylmethyl)-4-{4-[2-(thiophen-3-yl)acetyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[1-(methoxymethyl)cyclopropanecarbonyl]piperidin-3-ol
4-ethyl-1-methyl-3-(1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(3,5-dimethylphenyl)-4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperazin-2-one
1-({1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid