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(2S,4R)-4-cycloheptaneamido-N-ethyl-1-(1H-imidazol-4-ylmethyl)pyrrolidine-2-carboxamide
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-4-(propan-2-yl)-1,3-thiazole-2-carboxamide
N-methyl-2-[2-methyl-4-oxo-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
2-({3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}methyl)-6,8-dimethylquinolin-4-ol
2-[1-(propan-2-yl)piperidin-4-yl]-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)acetamide
3-[(3R,4S)-1-[(3-fluorophenyl)carbamoyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-benzyl-N-[2-(cyclohex-1-en-1-yl)ethyl]-4-hydroxy-2-methylpyrimidine-5-carboxamide
N-benzyl-1-methyl-5-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(4aS,7aR)-N-(4-methoxyphenyl)-6,6-dioxo-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-(1-cyclobutanecarbonylpiperidine-4-carbonyl)-4-(pyridin-3-yl)piperidin-4-ol
1-[3-(3-chlorophenyl)propyl]-4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
4-[3-(2-methoxyethyl)-1-methyl-1H-1,2,4-triazol-5-yl]-1-(2-methylpropyl)pyrrolidin-2-one
2-[4-({5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl}amino)piperidin-1-yl]acetamide
2-({4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}methyl)quinoline
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)butanamide
2-{[1-({3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)piperidin-4-yl]oxy}pyrimidine
(2R,6S)-4-[4-(4-chlorophenoxy)piperidine-4-carbonyl]-2,6-dimethylmorpholine
4-{[2-(pyridin-2-yl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
N-methyl-4-[3-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]-1,3-thiazol-2-amine
5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-pyrazole-4-carboxamide
ethyl 2-(1-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}piperidin-2-yl)acetate
2-(5-chlorothiophen-2-yl)-6-methylpyridine-3-carboxamide
4-hydroxy-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-2-(pyridin-2-yl)pyrimidine-5-carboxamide
2-[methyl(pyridin-3-ylmethyl)amino]-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}acetamide
4-[3-(3,4-dimethoxybenzoyl)piperidine-1-carbonyl]-7-fluoro-2-methylquinoline
1-(2,2-dimethylpropyl)-3-hydroxy-3-({[(3-methylphenyl)methyl]amino}methyl)piperidin-2-one
1-{1-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperidin-4-yl}piperidin-3-ol
1-{2-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}-3,3-dimethylurea
(3R,4R)-1-(2,3-dihydro-1H-inden-2-yl)-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
N-(1-carbamoylcyclopentyl)-2-fluoro-5-sulfamoylbenzamide
N-{[7-chloro-2-(3-methoxyphenyl)quinolin-3-yl]methyl}-N-(3-methoxypropyl)-3-methylthiophene-2-carboxamide
4-[4-methoxy-2-methyl-5-(propan-2-yl)phenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
6-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}-9H-purine
1-[5-methyl-4-(1-methyl-1H-1,2,4-triazol-5-yl)pyrimidin-2-yl]azonane
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
N-methyl-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
(2S,4S)-4-{2-[4-(dimethylamino)phenyl]acetamido}-N,N-diethyl-1-methylpyrrolidine-2-carboxamide
N-methyl-5-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(2S,4R,6S)-2-(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)-6-(2-methylpropyl)oxan-4-yl]acetamide
N-{1-[(5-fluoro-2-methylphenyl)carbamoyl]ethyl}-N'-(4-methylphenyl)propanediamide
2-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]pyrazine
2-{[4-(4-benzyl-5-{[(4-fluorophenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}phenol
N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
3-(1-methyl-1H-1,2,3-benzotriazol-5-yl)-1-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]urea
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
(1S,5R)-3-[(1-methyl-1H-indol-2-yl)methyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(4-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}piperazin-1-yl)-1,3-benzothiazole
2-(2,3-difluorophenoxymethyl)-N-(2-methoxyethyl)-N-methyl-1,3-oxazole-4-carboxamide
1-cyclopropanecarbonyl-4-(3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-5-yl)piperidine
2-[6-fluoro-2-(pyrimidin-5-yl)quinoline-4-carbonyl]-1,2,3,4-tetrahydroisoquinoline-7-carbonitrile