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(2S,3S)-2-{[(5-methoxy-2-methylphenyl)carbamoyl]amino}-3-methylpentanamide
N-({1-[(dimethyl-1,2-oxazol-4-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)-N-ethyl-2-methoxyacetamide
N-(2-methanesulfonylethyl)-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
N-({1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-3-yl}methyl)naphthalene-1-carboxamide
1-[2-(morpholin-4-yl)ethyl]-6-oxo-N-[3-(pyridin-4-yl)propyl]piperidine-3-carboxamide
4-methyl-2-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]phenol
1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)pyrrolidin-3-amine
6-[3-(dimethylamino)propyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-[(3R,4S)-4-cyclopropyl-1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)pyrrolidin-3-yl]-3-hydroxypropanamide
1-{4-[3-hydroxy-3-(2-methylphenyl)pyrrolidine-1-carbonyl]-3,5-dimethyl-1H-pyrrol-2-yl}ethan-1-one
N-cyclopropyl-1-{1-[(2-fluoro-4-methylphenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
3-{1-[(3,7-dimethyl-1H-indol-2-yl)methyl]piperidin-3-yl}-N-[(3-methoxyphenyl)methyl]propanamide
{[1-butyl-2-(cyclohexanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[(1-methylpyrrolidin-2-yl)methyl]amine
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-(prop-2-en-1-yl)propanamide
3,5-dimethyl-4-{1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1-phenyl-1H-pyrazole
N-cyclopropyl-2-[(3,5,7-trimethyl-1H-indol-2-yl)formamido]acetamide
1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(pyrrolidine-1-carbonyl)piperidine
2-(4-fluoro-2-methoxyphenyl)-2-{methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}acetic acid
1-(4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl)-4-methylpentane-1,2-dione
2-(4-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-1-(3-methylbut-2-en-1-yl)piperazin-2-yl)ethan-1-ol
1-{2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
N-(cyclopropylmethyl)-2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-propylacetamide
(4aS,7aR)-1-(2-hydroxybenzoyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
propan-2-yl 4-chloro-3-{[(oxolan-2-ylmethyl)carbamoyl]amino}benzoate
{[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}[3-(1H-imidazol-1-yl)propyl]amine
1-cyclopropyl-3-{2-[3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-2-oxoethyl}-3-(4-phenylphenyl)pyrrolidine-2,5-dione
N5-benzyl-N6,N6-dimethyl-N5-[(4-methyl-1,3-thiazol-5-yl)methyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-3-(pyridin-2-yl)propan-1-one
3-(1H-pyrazol-4-yl)-N,N-bis(pyridin-3-ylmethyl)benzamide
3-(5-methoxy-1H-indol-2-yl)-N,N-dimethyl-1H-1,2,4-triazol-5-amine
4-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)morpholine
N-(2-methoxyethyl)-N-[(3-methoxyphenyl)methyl]-2-methyl-1,3-thiazole-4-carboxamide
N-cyclopentyl-1-{1-[(2,4-dimethylphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-3,5-dimethyl-N-(pyridin-4-ylmethyl)-1,2-oxazole-4-carboxamide
8-(2-methyl-5-propylpyrimidin-4-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
1-[2-(4-ethoxyphenyl)ethyl]-3-(1,2,3-thiadiazol-5-yl)urea
1-({2,4-dimethyl-5H,6H-furo[2,3-d]pyrimidin-6-yl}methyl)-1,2,3,4-tetrahydroquinolin-2-one
5-methanesulfonyl-2-methyl-4-[4-(thiophene-2-carbonyl)piperazin-1-yl]pyrimidine
2-(3-fluoro-4-hydroxyphenyl)-1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-[5-(methoxymethyl)furan-2-carbonyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
5-ethyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]pyrimidin-2-amine
1-(2,1,3-benzothiadiazol-5-ylmethyl)-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
2-cyclopropyl-5-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}pyrimidine
2-(2-phenylethyl)-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine
2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
3-(4-fluorophenoxymethyl)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine
2-methyl-8-[6-methyl-2-oxo-4-(thiophen-2-yl)-1,2,3,4-tetrahydropyrimidine-5-carbonyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-(1-methyl-1H-pyrrol-2-yl)-2-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethane-1,2-dione
1-[5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-yl]piperidin-4-ol