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5-(2,4-difluorophenoxymethyl)-N-(5-methylhexan-2-yl)-1,2-oxazole-3-carboxamide
7,7-dimethyl-N-(4-methylquinolin-2-yl)-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
(2R,3R,6R)-3-(4-fluorophenyl)-5-(trimethyl-1H-pyrazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
{[5-(oxan-2-yl)furan-2-yl]methyl}bis(1,3-oxazol-4-ylmethyl)amine
N-methyl-N-[(5-methylfuran-2-yl)methyl]-5-phenyl-1H-pyrrole-2-carboxamide
2-{4-[2-(methylamino)pyridine-3-carbonyl]piperazin-1-yl}-1-(pyrrolidin-1-yl)ethan-1-one
4-[(3-ethylmorpholin-4-yl)methyl]-N-(2-methoxy-6-methylphenyl)benzamide
2-(1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-5-fluoro-1H-1,3-benzodiazole
N-(3-methylphenyl)-3-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}propanamide
2-amino-N,4-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1,3-benzothiazole-6-carboxamide
2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(6-methylpyridin-2-yl)methyl]acetamide
3-{4-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]phenyl}prop-2-yn-1-ol
(1R,3R)-N1-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]cyclopentane-1,3-diamine
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
3-[2-(pyridin-3-yl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-methyl-N-(3-{4-[(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]phenoxy}propyl)piperidine-2-carboxamide
1-(5-chloropyridin-2-yl)-4-[(2,3,4-trimethoxyphenyl)methyl]piperazine
8-[(2-aminopyridin-3-yl)methyl]-3-{3-[3-(dimethylamino)pyrrolidin-1-yl]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(3-chloro-1,2-oxazol-5-yl)-1-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]propan-1-one
1-(cyclopropylmethyl)-5-[3-(2-methoxyphenyl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(2S,4S)-4-({[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}amino)-N-methyl-1-(propan-2-yl)pyrrolidine-2-carboxamide
N-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
4-ethyl-1-({8-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]acetyl}-3-methyl-1-(2-methylpropyl)piperazin-2-one
2-[ethyl({[(3R,4R)-1-(2-fluoro-4-methylbenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl})amino]ethan-1-ol
2,6-dimethyl-N-[3-(2H-1,2,3,4-tetrazol-2-yl)adamantan-1-yl]pyrimidine-4-carboxamide
1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(thiophen-3-yl)ethan-1-one
1-[(3,4-difluorophenyl)methyl]-4-[1-(methoxymethyl)cyclobutanecarbonyl]piperazine
N-({1-[(1-ethenyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)-1H-pyrrole-2-carboxamide
N-[2-(dimethylamino)ethyl]-5-(6-methylpyridazin-3-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-{3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}acetamide
5-methyl-N-[(1-phenylcyclopentyl)methyl]-1-propyl-1H-pyrazole-4-carboxamide
N-methyl-4-{[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]methyl}benzamide
6-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-5,6-dihydro-1,6-naphthyridin-5-one
N-[2-(dimethylamino)ethyl]-5-(3-methyl-1H-pyrazole-5-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-1-(2-methoxyacetyl)piperidine-3-carboxamide
2-{1-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]-1-oxobutan-2-yl}-2,3-dihydro-1H-isoindol-1-one
N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)imidazo[1,2-a]pyrimidine-2-carboxamide
N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3,4,9-tetrahydro-1H-carbazole-1-carboxamide
(4aS,8aS)-2-[(4-chloro-3-fluorophenyl)methyl]-decahydroisoquinolin-4a-ol
2-ethyl-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-2,5-dihydro-1H-pyrrole
4-ethyl-1-[(2E)-3-phenylprop-2-en-1-yl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[2-(dimethylamino)ethyl]-9-[(3-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-5-methylphenol
5-(2-butylpyrimidin-4-yl)-2-ethoxybenzoic acid
8-chloro-2-{[4-(thiomorpholin-4-yl)piperidin-1-yl]methyl}quinoline
2-{[2-(dimethylamino)ethyl][(5-methylthiophen-2-yl)methyl]amino}acetic acid
1-(4-methyl-1,3-thiazole-5-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
4-cyano-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1-methyl-1H-pyrrole-2-carboxamide