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N-cyclopropyl-2-methoxy-N-[(2-methoxyphenyl)methyl]-5-methylbenzamide
N-(2,3-dihydro-1H-inden-2-yl)-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
N-(dimethyl-1H-1,2,4-triazol-3-yl)-4-({[1-(furan-2-yl)ethyl](methyl)amino}methyl)benzamide
(3R,4R)-1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-(4-methylpiperazin-1-yl)piperidin-3-ol
ethyl 4-(2-phenylethyl)-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperidine-4-carboxylate
1-{[1-(3,5-dimethoxybenzoyl)piperidin-3-yl]methyl}-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
4-{4-[(2-fluoro-3-methoxyphenyl)methyl]piperazin-1-yl}-2-methyl-6-propylpyrimidine
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-3-(1H-pyrazol-1-yl)benzamide
1-[(4-methoxyphenyl)methyl]-4-{[4-(methylsulfanyl)phenyl]methyl}piperazin-2-one
3-(2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
1-[2-({[(5-fluoro-2-methylphenyl)methyl]amino}methyl)-6-methoxyphenoxy]-3-(morpholin-4-yl)propan-2-ol
1-(2-ethoxyphenyl)-4-[1-(2-methoxyethyl)piperidine-3-carbonyl]piperazine
3-(4-methyl-1,3-thiazol-5-yl)-1-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}propan-1-one
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N,6-dimethylpyridine-3-carboxamide
9-methoxy-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-(1-methylcyclohexanecarbonyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-hydroxy-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(3-methylphenyl)pyrimidine-5-carboxamide
2-(1-benzothiophen-7-yl)-2-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]acetic acid
N-[2-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)ethyl]-2-fluorobenzamide
7-(2-methoxyethyl)-2-{6-methylthieno[2,3-d]pyrimidin-4-yl}-2,7-diazaspiro[4.5]decan-6-one
1-[2-(1H-imidazol-1-yl)ethyl]-5-methyl-5-phenylpiperidin-2-one
5-[3-(4-methylphenoxymethyl)piperidine-1-carbonyl]-2-(propan-2-yl)pyrimidine
2-(pyrrolidin-1-yl)-N-[3-(1H-1,2,4-triazol-1-yl)propyl]benzamide
4-{1-[3-(piperidin-1-ylmethyl)phenyl]-1H-imidazol-2-yl}benzoic acid
N-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
4,4-difluoro-N-[4-(oxan-2-ylmethoxy)phenyl]piperidine-1-carboxamide
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
methyl 3-(2-chlorobenzenesulfonamido)-5-({[3-(propan-2-yl)-1H-pyrazol-5-yl]formamido}methyl)benzoate
1-(4-methoxyphenyl)-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]cyclopentane-1-carboxamide
N-{[2-(4-acetylpiperazin-1-yl)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)-2-(thiophen-3-yl)acetamide
1-[(4-fluorophenyl)methyl]-5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-{[(2,5-difluorophenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
2-{[4-(2-methoxyphenyl)-5-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
3-{1-[2-amino-6-(propan-2-yl)pyrimidine-4-carbonyl]piperidin-4-yl}-N-cyclopropylpropanamide
2-amino-4-(3-hydroxyphenyl)-6-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
1,6-dimethyl-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-{1-[(2-ethoxyphenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(2-methylpropyl)-1-benzofuran-2-carboxamide
4-[(2-oxopyrrolidin-3-yl)sulfamoyl]-N-phenylbenzamide
{4-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methanol
4-methyl-2-(2-{4-[2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}propyl)pyridine
2-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-amine
2-[(E)-2-(furan-2-yl)ethenyl]-7-methyl-1H-1,3-benzodiazole
(4aR,8aR)-1-(adamantane-1-carbonyl)-6-phenylmethanesulfonyl-decahydro-1,6-naphthyridine
1-[1-(2,5-dimethylbenzoyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
1-{2-[3-(3-methylphenoxymethyl)piperidin-1-yl]-2-oxoethyl}piperidin-2-one
1-[2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)acetyl]-4-phenylpiperidine-4-carbonitrile
N-(1-carbamoylcyclopentyl)-6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-{4-[2-(oxolan-2-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-(thiophen-3-yl)ethan-1-one
(2R)-2-[4-phenyl-5-(1-propyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]propanamide