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ethyl 4-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperazine-1-carboxylate
N-[2-({[4-(morpholin-4-ylmethyl)phenyl]carbamoyl}amino)ethyl]pyridine-3-carboxamide
1-[5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-yl]-4-(pyridin-4-ylmethyl)piperazine
7-[3-(2-methoxyphenyl)propanamido]-N-propyl-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
5-[(2,3-dihydro-1H-inden-2-yl)amino]-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[(4-{5-[(cyclohexylmethyl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]-6-methylpyridine
1-{[4-(5-methylfuran-2-yl)phenyl]methyl}piperidine-4-carbonitrile
3-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
N-[2-(4-ethylpiperazin-1-yl)-2-methylpropyl]pyridine-4-carboxamide
3-[2-(2,4-difluorophenyl)ethyl]-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidine
2-(1-butyl-1H-pyrazol-4-yl)-8-methyl-4-(2-methylpyrrolidine-1-carbonyl)quinoline
2-{[4-(1H-1,2,3-benzotriazol-1-yl)piperidin-1-yl]methyl}pyridine-3-carboxylic acid
(1S,5R)-3-(5-chloropyridine-3-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{[(4-methoxyphenyl)methyl]amino}-N,5-dimethyl-N-(1,3-thiazol-4-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
N3-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}piperidine-1,3-dicarboxamide
5-cyclopropyl-N-[4-methyl-3-(4-methylbenzamido)phenyl]-1,2-oxazole-4-carboxamide
7-methoxy-3-(1,3-thiazol-4-ylmethyl)-2,3,4,5-tetrahydro-1H-3-benzazepine
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidine
4-[(1-ethyl-1H-imidazol-5-yl)methyl]-1-phenylpiperazin-2-one
[1-(2-{[4-(pyridin-2-yl)pyrimidin-2-yl]amino}ethyl)piperidin-2-yl]methanol
6-methyl-N-[(5-methylpyrazin-2-yl)methyl]-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
4-[(methylsulfanyl)methyl]-1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperidine
(4aS,8aR)-6-[5-(hydroxymethyl)furan-2-carbonyl]-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
5-ethyl-N4-methyl-N4-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}pyrimidine-2,4-diamine
3-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-2-yl}pyridine
4-[3-(2,4-dimethyl-1,4-diazepane-1-carbonyl)phenyl]-2-methylbutan-2-ol
1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-1H-pyrazole-4-carboxamide
2-[(4-chlorophenyl)methyl]-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1,3-benzoxazole-5-carboxamide
(3R)-3-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]-1,2,3,4-tetrahydroisoquinoline
N-{2-[(8-fluoro-4-oxo-1,4-dihydroquinolin-2-yl)formamido]ethyl}pyridine-3-carboxamide
1-(2-cyclohexylethyl)-3-({[(3-fluorophenyl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
(1S,5R)-3-(2-ethoxyethyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-butyl-3-{[2-(2-methoxyphenoxy)acetamido]methyl}piperidine-1-carboxamide
6-[methyl(2-methylprop-2-en-1-yl)amino]-N-[2-(1-methylpiperidin-2-yl)ethyl]pyridine-3-carboxamide
N-[2-(2-fluorophenoxy)ethyl]-1-methylpiperidin-4-amine
2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(4-hydroxyazepan-4-yl)methyl]acetamide
2-[1-(5-acetyl-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)pyrrolidin-3-yl]benzoic acid
N-[2-(5,7-difluoro-2-methyl-1H-indol-3-yl)ethyl]-2-(3-methyl-1,2-oxazol-5-yl)acetamide
2-[2-(1-{4-[(2-hydroxyethyl)(methyl)amino]benzoyl}piperidin-3-yl)-1H-imidazol-1-yl]acetamide
3-cyclopropyl-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazol-5-yl]-1H-1,2,4-triazole
5-[2-(4-fluorophenyl)piperidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
8-fluoro-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)quinoline-2-carboxamide
N-[(2-chloro-6-fluorophenyl)methyl]-N-ethyl-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
4-(2,4-dioxoimidazolidin-1-yl)-N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]benzamide
(4aS,8aR)-1-[3-(methylsulfanyl)propyl]-6-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-decahydro-1,6-naphthyridin-2-one
1-(1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazol-3-yl)ethan-1-one
2,3-dimethoxy-N-(2-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)benzamide
(1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methanol
(4aR,7aS)-1-(1H-imidazol-4-ylmethyl)-4-[(2E)-3-phenylprop-2-enoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(5-methoxyfuran-2-carbonyl)-3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine