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3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[1-(4-fluorophenyl)ethyl]benzamide
1-cyclopropyl-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
2-(diethylamino)-1-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
N-methyl-3-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-N-[2-(pyridin-2-yl)ethyl]propanamide
N-{[1-(3-methoxypropanoyl)piperidin-3-yl]methyl}naphthalene-1-carboxamide
N-(3-chloro-4-methoxyphenyl)-3-(morpholin-4-yl)piperidine-1-carboxamide
3-{[3-(3,4-difluorophenyl)-1,2,4-oxadiazol-5-yl]methyl}pyridine
methyl 2-[4-(3-fluorophenoxy)piperidin-1-yl]pyridine-3-carboxylate
5-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1H-1,2,4-triazol-3-amine
8-methoxy-2-(2-methoxyphenyl)-3-(1H-pyrazol-1-ylmethyl)quinoline
[3-({[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]amino}methyl)-2,4,6-trimethylphenyl]methyl acetate
2-ethyl-9-[2-(4-fluorophenoxy)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-3-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]urea
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methylfuran-2-carboxamide
N-benzyl-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide
3-(methylsulfanyl)-1-[3-(4-phenylbenzoyl)piperidin-1-yl]propan-1-one
2-(pyridin-3-yl)-1-{3-[2-(pyridin-4-yl)pyridin-4-yl]pyrrolidin-1-yl}ethan-1-one
2-[2-(4-phenylpiperidin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
1-(2-{4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethyl)piperazine
2-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoacetamide
3-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-2-methylphenol
2-(4-fluorophenyl)-1-(5-phenyl-1,2-oxazole-3-carbonyl)piperidine
1-{[5-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-3,3-dimethylurea
6-methyl-N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)imidazo[1,2-a]pyridine-2-carboxamide
2-methyl-7-[2-phenyl-2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-[(2-chlorophenyl)methyl]-4-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
(1S,5R)-3-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{[3-cyclopropyl-1-(2-hydroxybutyl)-1H-1,2,4-triazol-5-yl]methyl}-1,2-dihydrophthalazin-1-one
6-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-[(4-fluorophenyl)methyl]-3-{1-[4-(1H-imidazol-1-yl)benzoyl]piperidin-4-yl}propanamide
N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-3-(4H-1,2,4-triazol-4-yl)benzamide
6-(2-chlorophenyl)-2-(3-ethylpiperazine-1-carbonyl)-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-1-methyl-1H-indole-6-carboxamide
(3S,5R)-5-(3,3-diphenylpiperidine-1-carbonyl)pyrrolidin-3-ol
N-cyclopropyl-2-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}acetamide
3-methyl-1-(1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)butan-1-ol
4-(2-oxo-1,2-dihydropyridin-4-yl)-2,2-diphenylbutanenitrile
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidine
1-ethyl-6,7,8-trifluoro-3-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-1,4-dihydroquinolin-4-one
5-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
3-[2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]-4-[(4-phenylphenyl)methyl]piperazin-2-one
8-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]-1-(benzyloxy)-1,8-diazaspiro[4.5]decan-2-one
4-hydroxy-N-(2-methylpropyl)-2-(pyridin-3-yl)-N-(pyridin-4-ylmethyl)pyrimidine-5-carboxamide
2-(1-cyclohexyl-4-{[5-(methoxymethyl)furan-2-yl]methyl}piperazin-2-yl)ethan-1-ol
3-hydroxy-1-[7-(1,2,3,4-tetrahydroquinoline-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]propan-1-one
N'-(3,5-dimethylphenyl)-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]propanediamide
1-(5-methylpyridin-3-yl)-5-oxopyrrolidine-3-carboxylic acid
2-methyl-8-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(2S,4S)-N-ethyl-1-(3-methylbut-2-en-1-yl)-4-[3-(4-methylphenyl)propanamido]pyrrolidine-2-carboxamide