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4-(1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidin-4-yl)thiomorpholine
4-[2-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]piperazin-2-one
methyl (2S,4R)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(3,5-dimethoxyphenyl)methyl]pyrrolidine-2-carboxylate
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-acetamidopropanamide
1-{3-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
2-{4-[(5-cyclopentylthiophen-2-yl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-(2-hydroxybutyl)propanamide
5-[4-(2-hydroxyphenyl)piperazine-1-carbonyl]-N-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-amino-6-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]pyrimidine-4-carboxamide
(3aR,6aR)-2-(2,1,3-benzoxadiazol-4-ylmethyl)-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1H-pyrrole-2-carboxamide
N-(1H-1,2,3-benzotriazol-5-yl)-4-cyclohexylpiperazine-1-carboxamide
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-methyl-N-{3-[(5-methylpyridin-2-yl)amino]propyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
4-({1-[(6-methoxypyridin-3-yl)methyl]piperidin-3-yl}methyl)morpholine
2-(pyridin-3-yl)-5-(2,3,4-trimethoxyphenyl)-1,3-benzoxazole
3-({[(3R,5S)-1-benzyl-5-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}pyrrolidin-3-yl]amino}methyl)phenol
(4aR,7aS)-1-(2-methylpropyl)-4-[(1-phenyl-1H-pyrazol-4-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(2-chlorophenyl)methyl]-3-[3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]propanamide
dimethyl(2-{[(2-methyl-1,3-oxazol-4-yl)methyl](oxolan-2-ylmethyl)amino}ethyl)amine
1-(2-methoxyethyl)-N-[1-(4-methylbenzoyl)piperidin-4-yl]pyrrolidine-3-carboxamide
N-{1-[2-hydroxy-6-(trifluoromethyl)pyridine-3-carbonyl]piperidin-4-yl}methanesulfonamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxy-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]benzamide
(3R,4R)-4-hydroxy-3-methyl-N-[(2-methylphenyl)methyl]-4-(oxan-4-yl)piperidine-1-carboxamide
N-[(4-methoxyphenyl)methyl]-2-(trifluoromethyl)morpholine-4-carboxamide
7-[4-(3,5-dimethyl-1H-pyrazol-1-yl)butanoyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
(2R,4S)-1-[(2E)-3-(5-chloro-2-hydroxyphenyl)-2-methylprop-2-en-1-yl]-4-hydroxypiperidine-2-carboxylic acid
2-(2-methylphenoxy)-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
(1S,4S)-2-(4-chloro-2-methoxy-5-methylphenyl)-5-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-2,5-diazabicyclo[2.2.1]heptan-3-one
2-ethoxy-1-{2-[5-(4-methyl-1,4-diazepane-1-carbonyl)thiophen-2-yl]pyrrolidin-1-yl}ethan-1-one
3-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-1-[3-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]urea
2-methyl-1-{3-[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]propyl}-1H-1,3-benzodiazole
N-methyl-2-({4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}amino)ethane-1-sulfonamide
6-methyl-2-oxo-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}-1,2-dihydropyridine-3-carboxamide
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
(3-{2-[1-(2,6-dimethylpyridin-4-yl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
3-{3,9-diazaspiro[5.6]dodecan-9-ylmethyl}-5-methyl-1H-indole-2-carboxylic acid
2-(1-butyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)acetamide
1-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}-4-(furan-2-carbonyl)piperazine
2-[(5-{[methyl(2-phenylethyl)amino]methyl}-1,2-oxazol-3-yl)formamido]acetamide
2-(2-methoxyethyl)-9-[2-(oxolan-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2,6,8-trimethyl-4-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]quinoline
(2R,6R)-4-{3-[(dimethylamino)methyl]benzoyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-amino-4-[2-(morpholin-4-yl)-1,3-thiazol-5-yl]-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
N,1,3-trimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(1R,2S)-2-({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)cyclopentane-1-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(1-ethyl-1H-pyrazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
methyl 6-[1-(4-fluorophenyl)propan-2-yl]-2-(pyrrolidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(1R,6S)-N-[2-(2-fluorophenoxy)pyridin-3-yl]-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide