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(1R,5R)-3-(3-methoxybenzoyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
N-butyl-N-[(4-chlorophenyl)methyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
N-(2-{4-[(2-tert-butylpyrimidin-5-yl)methyl]morpholin-2-yl}ethyl)acetamide
2-[(3-methoxyphenyl)methyl]-8-(propane-1-sulfonyl)-2,8-diazaspiro[4.5]decan-3-one
4-({3-ethoxy-4-[(3-methylbut-2-en-1-yl)oxy]phenyl}methyl)piperazine-1-carboxamide
3-methyl-2-{4-phenyl-5-[4-(propan-2-yl)-1,3-thiazol-2-yl]-1H-imidazol-1-yl}butan-1-ol
1-[(3-methoxyphenyl)methyl]-N-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}piperidin-3-amine
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(3-methyl-1H-pyrazol-1-yl)propanamide
6-methyl-N4-[1-(2-methylphenyl)cyclopropyl]pyrimidine-2,4-diamine
3-(azocan-1-yl)-N-(3-hydroxypropyl)-N-(thiophen-2-ylmethyl)propanamide
N-[(7R,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
2-{[5-fluoro-2-(furan-3-yl)pyrimidin-4-yl]amino}ethan-1-ol
1-(5-methyl-1,3-oxazole-4-carbonyl)-4-phenoxypiperidine-4-carboxylic acid
ethyl 2-{1-[2-(3,5-difluorophenyl)acetyl]piperidin-2-yl}acetate
6-[(3-methyl-3-phenylpiperidin-1-yl)methyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]pyridine-4-carbonitrile
7-(1-benzothiophen-3-yl)-4-(furan-2-carbonyl)-9-[2-(pyridin-2-yl)ethoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2-(pyrazin-2-yl)acetamide
N-(1-{2-[(2-methylprop-2-en-1-yl)oxy]benzoyl}piperidin-4-yl)pyrimidin-2-amine
methyl({[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl})[3-(oxolan-2-yl)propyl]amine
2-(1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}piperidin-3-yl)-1,2,3,4-tetrahydroisoquinoline
3-methyl-1-(1-{6-[4-(propan-2-yl)piperazin-1-yl]pyridine-3-carbonyl}piperidin-3-yl)butan-1-one
1-[9-methoxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-phenylethan-1-one
N-({7-[2-(2,5-dimethoxyphenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-3-carboxamide
N-[(2-ethoxyphenyl)methyl]-N-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}cyclopropanamine
1-[(3-fluorophenyl)methyl]-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
2-{4-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}-5-fluoro-4-(pyrrolidin-1-yl)pyrimidine
(3S,4R)-4-(2-methylphenyl)-1-(5,6,7,8-tetrahydroquinoline-3-carbonyl)pyrrolidine-3-carboxylic acid
(3S,4S)-1-(1-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
2-(dimethyl-1,2-oxazol-4-yl)-N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]acetamide
6-ethyl-1,5-dimethyl-3-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-1,2-dihydropyridin-2-one
3-{[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}phenol
methyl 2-{[2-(cyclohex-1-en-1-yl)ethyl]sulfamoyl}-6-(3-hydroxybutyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-chloro-N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-1-methyl-1H-pyrazole-3-carboxamide
N-[(1-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-3-yl)methyl]furan-2-carboxamide
3-{[(4aR,8aR)-4a-hydroxy-7-methanesulfonyl-decahydro-2,7-naphthyridin-2-yl]methyl}-1,2-dihydroquinolin-2-one
N-[2-hydroxy-2-(3-phenoxyphenyl)ethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
2-methyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-2-ylmethyl)imidazo[1,2-a]pyridine-6-carboxamide
N-ethyl-N-methyl-6-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyrimidin-4-amine
N-butyl-3-({[3-(1H-indazol-1-yl)propyl]amino}methyl)-N-methylimidazo[1,2-a]pyridine-2-carboxamide
N-(6-phenoxypyridin-3-yl)-1-[(2-propylpyrimidin-5-yl)methyl]piperidine-2-carboxamide
5-(4-chloro-1H-indazol-1-yl)-N-methylfuran-2-carboxamide
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-4-phenoxybutan-1-one
4-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperazine-2-carboxylic acid
3-[(4aR,7aS)-4-[(4-methoxy-2-methylphenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
1-{4-chloro-3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}piperidine
1-{7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}pent-4-en-1-one
[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl](methyl){[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine