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2-(dimethylamino)-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}acetamide
N-[5-(morpholin-4-yl)pentyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
4-(4-butyl-1H-1,2,3-triazol-1-yl)-1-(oxolan-3-ylmethyl)piperidine
N-{2-[4-(dimethylamino)phenyl]ethyl}-2-(1-methylpiperidin-2-yl)acetamide
2,3,5-trimethyl-N-[3-(pyrrolidin-1-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-(4-methoxyphenoxymethyl)-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1,3-oxazole-4-carboxamide
4-(1-ethyl-1H-imidazol-2-yl)-1-[4-(1H-imidazol-1-yl)benzoyl]piperidine
1-(2,3-dihydro-1H-inden-2-yl)-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-3-carboxamide
2-(2H-indazol-2-yl)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]ethan-1-one
N-methyl-N-({1-[2-(pyridin-2-yl)ethyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)furan-2-carboxamide
2-[(2,6-dichlorophenyl)methyl]-5-(piperazine-1-carbonyl)pyrimidin-4-ol
4-{4-[2-(1H-imidazol-1-yl)ethyl]piperazin-1-yl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
8-[(4,5-dimethylfuran-2-yl)methyl]-3-{3-[methyl(2-methylpropyl)amino]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(3-{3-[2-(dimethylamino)ethyl]-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}-3-oxopropyl)-N-methylmethanesulfonamide
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-3-(3-methoxypropyl)piperidine
N-[(3S,4R)-1-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}-4-propylpyrrolidin-3-yl]acetamide
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}pyrimidin-4-amine
(4aS,8aR)-1-(3-hydroxypropyl)-6-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]propanamide
1-cycloheptyl-N-[2-(1H-indol-1-yl)ethyl]-6-oxopiperidine-3-carboxamide
11-{[(3,4-difluorophenyl)methyl]amino}-4-[2-(dimethylamino)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-benzyl-8-(1H-indol-2-ylmethyl)-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,9aR)-8-(4-phenylbenzoyl)-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(2,5-dimethylphenyl)(pyridin-3-yl)methyl]-2-(ethylamino)pyrimidine-5-carboxamide
N-(butan-2-yl)-N-[(4-chlorophenyl)methyl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
(2R,3R,6R)-N-benzyl-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
7-hydroxy-4-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-6-methyl-1,2,3,4-tetrahydroquinolin-2-one
5-(1,3-benzothiazol-2-ylmethyl)-N-cyclopropyl-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-methyl-8-(9H-purin-6-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
methyl 1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}-1H-imidazole-4-carboxylate
2-[5-(1,3-benzothiazol-2-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
N-(3-methoxypropyl)-1-methyl-N-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}piperidin-4-amine
3-[(6-amino-2-methylpyrimidin-4-yl)amino]-1-(pyrrolidin-1-yl)propan-1-one
2-{1-[(2-ethoxyphenyl)methyl]-4-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2-(1H-indazol-3-yl)acetamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl]propanoic acid
1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-4-[4-(2-phenylethyl)-1H-pyrazol-5-yl]piperidine
N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}imidazo[1,2-a]pyridine-2-carboxamide
1-(4-methyl-2-{methyl[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]amino}pyrimidin-5-yl)ethan-1-one
4-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-4-oxobutanamide
1-[5-(2,6-dimethoxyphenyl)-1,2,4-triazin-3-yl]-4-(pyridin-2-ylmethyl)-1,4-diazepane
1-(2-methoxyphenyl)-4-[4-(trimethyl-1H-pyrazol-4-yl)-1H-imidazol-2-yl]pyrrolidin-2-one
N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
{3-[1-(2-fluorophenyl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]propyl}dimethylamine
3-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-1-(2-methoxyphenyl)urea
(1R,5R)-6-benzyl-3-(3-propyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-{1-[5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]piperidin-3-yl}propan-2-ol
9-{[2,4-bis(prop-2-en-1-yloxy)phenyl]methyl}-1,4,9-triazaspiro[5.5]undecan-5-one
1-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-3-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]urea