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3-(1H-indol-3-yl)-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]propanamide
3-{1-[(1R,2S,3R,4S)-3-amino-7-oxabicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-N-(3-methylphenyl)propanamide
(1S,4S)-2-(2-chlorophenyl)-5-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-5-methyl-N-[3-(methylsulfanyl)propyl]thieno[2,3-d]pyrimidine-6-carboxamide
1-(4-fluorophenyl)-4-(1-propylpiperidin-3-yl)piperazine
methyl 4-[2-(1-cyclopentyl-3-oxopiperazin-2-yl)acetamido]butanoate
4,5,6,7-tetramethyl-2-{5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}-1H-1,3-benzodiazole
N-(5-methyl-1,3,4-thiadiazol-2-yl)-2-[(2R)-oxolane-2-carbonyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
2-({4-[6-(propan-2-yl)pyridin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethan-1-ol
1-[2-(pyridin-3-yl)piperidin-1-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
2-{[2-(1-{thieno[2,3-d]pyrimidin-4-yl}piperidin-3-yl)-1H-imidazol-1-yl]methyl}pyridine
(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1-{pyrazolo[1,5-a]pyridine-7-carbonyl}-1,2,3,6-tetrahydropyridine
6-(1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}piperidin-4-yl)-2-methyl-3,4-dihydropyrimidin-4-one
1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-methyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
2-[4-(5-fluoropentyl)phenyl]-2-methylpropanamide
4-[(3R,4R)-4-amino-3-hydroxypiperidin-1-yl]-1-(4-methylphenyl)butan-1-one
4-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]piperazine-2-carboxylic acid
3-{5-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
3-({[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(prop-2-en-1-yl)amino)-1λ6-thiolane-1,1-dione
2-methyl-2-(2-{[(1-methylpiperidin-4-yl)methyl]amino}-4-(morpholin-4-yl)pyrimidin-5-yl)propanoic acid
5-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)-3-(2-phenylethyl)-1H-1,2,4-triazole
(furan-2-ylmethyl)({[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl})(prop-2-yn-1-yl)amine
3-(8-chloro-2-ethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-[4-(3-methoxyphenyl)piperazin-1-yl]propan-1-one
methyl 3-(cyclobutylmethoxy)-5-[(2S)-2-(hydroxymethyl)pyrrolidine-1-carbonyl]benzoate
N,N-dimethyl-2-[(1S,5R)-3-{[2-(methylsulfanyl)phenyl]methyl}-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
3-{1-[4-(dimethylamino)benzoyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
(2E)-N-{[3-methyl-7-(1,3-thiazole-5-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
5-{[(5-fluoro-2-methylphenyl)methyl]amino}-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-(quinolin-2-ylmethyl)piperazin-2-yl}ethan-1-ol
5-{[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]methyl}-1-phenyl-1H-1,2,3,4-tetrazole
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)pyrrolidin-3-yl]methanol
2-(3-fluorophenyl)-1-(3-propyl-1H-pyrazole-5-carbonyl)azepane
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}acetamide
1-(2-methoxyacetyl)-N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]piperidine-3-carboxamide
4-(2-methoxyphenyl)-2-methyl-1-(3-phenyl-1,2,4-oxadiazol-5-yl)piperazine
N-[2-(2,4-dimethylphenoxy)ethyl]-4-(hydroxymethyl)-N-methylbenzamide
1-{2-[(4aR,8aR)-octahydro-2H-1,4-benzoxazin-4-yl]-2-oxoethyl}-3-methoxy-1,2-dihydropyridin-2-one
7-{[4-(propan-2-yl)phenyl]methyl}-2-(thiophene-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
6-(4-chlorophenyl)-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-1-[2-(trifluoromethoxy)phenyl]urea
5-cyclopropyl-N-[1-(2-propoxyphenyl)ethyl]-1,3,4-oxadiazol-2-amine
2-{4-[2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carbonyl]morpholin-2-yl}ethan-1-amine
7-(5-methoxy-1H-indole-2-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
N-[(3S,4R)-4-propyl-1-[4-(1H-pyrazol-3-yl)benzoyl]pyrrolidin-3-yl]acetamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(1-methyl-1H-imidazole-5-carbonyl)pyrrolidin-3-yl]methanol
N-{3-[4-phenyl-5-(1,3-thiazol-2-yl)-1H-imidazol-1-yl]propyl}pyridin-3-amine
N-[2-(dimethylamino)ethyl]-1-methyl-N-[(5-methylthiophen-2-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-2-(thiophen-3-yl)ethan-1-one