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4,5-dimethyl-6-{4-[3-(methylsulfanyl)propyl]piperazin-1-yl}pyrimidine
5-methyl-1-[4-(4-{[(2S)-3-methylbutan-2-yl]amino}piperidin-1-yl)phenyl]pyrrolidin-2-one
N-[(2-ethoxy-3-methoxyphenyl)methyl]-2-(1H-imidazol-2-yl)-N-methylbenzamide
N-[1-(6-methylpyridin-2-yl)propan-2-yl]-2-[4-(morpholin-4-yl)-6-oxo-1,6-dihydropyridazin-1-yl]acetamide
N-[1-(naphthalen-1-yl)ethyl]-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
N-(3-hydroxypropyl)-4-(1H-imidazol-1-yl)-N-(pyridin-4-ylmethyl)benzamide
[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl][1-(2-fluorophenyl)propan-2-yl]amine
4-(1,3-dimethyl-1H-pyrazol-5-yl)-3-(diphenylmethyl)-4H-1,2,4-triazole
2-{1-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]-1,4-diazepan-6-yl}acetic acid
(3S,4S)-4-cyclopropyl-1-(dimethyl-1,3-thiazole-5-carbonyl)pyrrolidine-3-carboxylic acid
1-[2-({[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}amino)ethyl]imidazolidin-2-one
3-ethyl-5-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-4-methyl-1H-pyrazole
N-phenyl-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-amine
(3S,5R)-N5-(4-fluorophenyl)-N3,N3-dimethyl-1-(naphthalen-2-ylmethyl)piperidine-3,5-dicarboxamide
(3aS,6aR)-5-(piperidine-1-sulfonyl)-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-[5-({2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)-1,2-oxazol-3-yl]pyridine
7-(1-benzothiophen-3-yl)-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(4-methylphenyl)-5-[4-(pyrrolidin-1-yl)piperidine-1-carbonyl]pyrimidin-4-ol
N-[(3,4-difluorophenyl)methyl]-3-[1-(1,3-thiazole-5-carbonyl)piperidin-3-yl]propanamide
N-(3-hydroxypropyl)-2,8-dimethyl-N-(thiophen-2-ylmethyl)quinoline-4-carboxamide
6,8-difluoro-2-methyl-4-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]quinoline
2-phenyl-1-[1-(thiophen-2-ylmethyl)piperidin-4-yl]ethan-1-ol
1-(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}ethan-1-one
1-{2-[1-(2,6-difluorobenzenesulfonyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
4-benzyl-1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(1,2,2,6,6-pentamethylpiperidin-4-yl)-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
6-{3-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]-3-oxopropyl}-2,3-dihydropyridazin-3-one
4-[(dimethylamino)methyl]-1-[3-(furan-2-yl)benzoyl]azepan-4-ol
2-(dimethylamino)-N-methyl-6-(4-methylthiophen-2-yl)-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]pyridine-3-carboxamide
1-(2-{methyl[(2E)-3-phenylprop-2-en-1-yl]amino}pyrimidin-4-yl)piperidin-4-ol
2-[3-(2-phenylethyl)piperidine-1-carbonyl]benzonitrile
2-amino-4-(1-methyl-1H-pyrazol-4-yl)-6-[4-(morpholin-4-yl)phenyl]pyridine-3-carbonitrile
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-2H-1,3-benzodioxole-5-carboxamide
3-benzyl-4-[3-(1H-pyrrol-1-yl)benzoyl]piperazin-2-one
N,N-dimethyl-2-[(1S,5R)-3-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}ethan-1-one
N-{[7-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3-dihydro-1,4-benzodioxine-6-carboxamide
1-[(1-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methyl]pyrrolidin-2-one
7-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-1H-indole
1-methyl-6-oxo-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-1,6-dihydropyridazine-3-carboxamide
2,3-dimethyl-6-(2-{1-oxo-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-2-yl}acetyl)-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
4-ethyl-3-(1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[4-hydroxy-4-(2-methylquinolin-6-yl)piperidin-1-yl]-2-(2-methoxyethoxy)ethan-1-one
3-{2-[2-(4-methanesulfonylphenyl)-1H-imidazol-1-yl]ethyl}-1,3-oxazinan-2-one
3-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]-1-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}urea
3-(1,1-dioxo-1λ6-thiolan-3-yl)-3-ethyl-1-[3-(1,3-thiazol-4-yl)phenyl]urea
N-(4-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-4-oxobutan-2-yl)acetamide