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2,4-dimethyl-5-{3-[1-(oxolan-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}-1,3-thiazole
N-[2-(3,5-difluorophenyl)ethyl]-1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
4-{4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carbonyl}pyridine
1-(2-chlorophenyl)-3-{1-[1-(2-methoxyacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-{2-[3-(trifluoromethyl)phenyl]ethyl}acetamide
2-amino-8-[5-chloro-2-(prop-2-en-1-yloxy)phenyl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
2-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,3-thiazole-4-carboxamide
N-(2-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)methanesulfonamide
4-(5-{1-[3-(1,3-oxazol-5-yl)phenyl]-1H-imidazol-2-yl}pyrimidin-2-yl)morpholine
(3S,4R)-4-methyl-1-(2-methyl-1,3-benzothiazole-5-carbonyl)piperidine-3,4-diol
1-({4-[2-hydroxy-3-(piperidin-1-yl)propoxy]phenyl}methyl)-N,4-dimethylpiperidine-4-carboxamide
1-[4-(2-{[3-(trifluoromethyl)phenyl]methyl}morpholin-4-yl)piperidin-1-yl]ethan-1-one
1-(4-fluorophenyl)-2,2-dimethyl-N-[(1r,4r)-4-hydroxycyclohexyl]cyclopropane-1-carboxamide
1-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-4-(pyridin-3-ylmethyl)piperazine
N-methyl-N-(2-{[3-(3-methylpiperidin-1-yl)-3-oxopropyl]amino}ethyl)methanesulfonamide
1-(2-{1-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
6-methyl-5-{[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]methyl}quinoline
1-(3-hydroxy-4-methylbenzoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-benzyl-2-cyclopropyl-4-hydroxy-N-(1,3-thiazol-2-ylmethyl)pyrimidine-5-carboxamide
2-[1-(2,2,2-trifluoroethyl)-1H-imidazol-2-yl]quinoline
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-4,6-dimethylpyrimidin-2-amine
2-(2,4-dichlorophenoxy)-N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
2-{[(3-ethoxyphenyl)methyl](1H-imidazol-2-ylmethyl)amino}ethan-1-ol
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}benzamide
3-[2-(1-cyclopentylpiperidin-2-yl)ethyl]-6-ethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-cyclopropyl-N-methyl-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}pyrimidine-5-carboxamide
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-4-(1H-pyrazol-3-yl)benzamide
(4aS,7aR)-1-[2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(2,6-dimethylpyridin-4-yl)-N-(6-fluoropyridin-3-yl)piperazine-1-carboxamide
1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-(2,2,3,3-tetrafluoropropoxy)ethan-1-one
methyl 5-{3-tert-butyl-1-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}-2-hydroxybenzoate
4-ethyl-3-{1-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(1R,6S)-9-methyl-3-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)-3,9-diazabicyclo[4.2.1]nonane
N-(2-phenylethyl)-6-[2-(phenylsulfanyl)acetyl]-6-azaspiro[2.5]octane-1-carboxamide
2-(7-hydroxy-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)benzoic acid
4-amino-2-(morpholin-4-yl)-5-[2-(morpholin-4-yl)propan-2-yl]-5H,6H,7H,8H-pyrido[2,3-d]pyrimidin-7-one
4-({4-[3-(cyclopropylmethyl)-1-ethyl-1H-1,2,4-triazol-5-yl]phenyl}methyl)-1λ6-thiomorpholine-1,1-dione
N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)propanamide
2-methyl-5-{[4-phenyl-5-(2-phenylethyl)-1H-imidazol-1-yl]methyl}-1,3,4-oxadiazole
1-ethyl-3-methyl-8-{[4-(pyrrolidin-1-yl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(2,4-dimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-1-(2-methoxyethyl)-1-(pyridin-3-ylmethyl)urea
N-[1-(2,5-difluorophenyl)cyclopropyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
8-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
4-hydroxy-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-(4-methylphenyl)pyrimidine-5-carboxamide
2-(3,4-dichlorophenyl)-4-(1-ethyl-1H-pyrazole-4-carbonyl)morpholine
(1R,7S)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-3-(3-methylbutyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
(2S,4S)-1-cyclohexyl-N-ethyl-4-(4-fluoro-3-methylbenzamido)pyrrolidine-2-carboxamide
3-[(2R,3R,6R)-5-(3-methyl-1H-pyrazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
3-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-[3-(sulfamoylmethyl)phenyl]urea
2-(adamantan-1-yl)-1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}ethan-1-one