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(3S,4R)-3-ethyl-4-methyl-1-[1-(pyridine-4-carbonyl)piperidine-4-carbonyl]piperidin-4-ol
4-methyl-N-(oxolan-2-ylmethyl)-N-(2-phenoxyethyl)-1H-imidazole-5-carboxamide
1-cyclohexyl-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-1H-1,2,3-triazole-4-carboxamide
2-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-5-(4-methyl-1,4-diazepan-1-yl)-2,3-dihydropyridazin-3-one
1-[(3-methyl-1-benzofuran-2-yl)methyl]-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
2-chloro-5-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]pyridine
(2E)-1-(4-{4-[(methylamino)methyl]-1H-1,2,3-triazol-1-yl}piperidin-1-yl)-3-(3-methylphenyl)prop-2-en-1-one
6-chloro-2-[2-(trifluoromethyl)morpholin-4-yl]quinoline
4-{1-[(2-chloro-6-fluorophenyl)methyl]-3-ethyl-1H-1,2,4-triazol-5-yl}-1-oxaspiro[4.4]nonan-2-one
1-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(pyrrolidin-1-yl)ethan-1-one
N-[1-(3-phenylpropyl)piperidin-3-yl]pyrazine-2-carboxamide
3-{2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-oxoethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
2-benzyl-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-1,3-benzoxazole-5-carboxamide
4-(1H-pyrazol-3-yl)-N-{2-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]ethyl}benzamide
4-(1-cyclopentyl-5-oxopyrrolidine-3-carbonyl)-1-(3-methoxyphenyl)piperazin-2-one
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
1-[3-(dimethylamino)phenyl]-3-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}urea
2-(4-{[methyl(pyridin-2-ylmethyl)amino]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
N-[2-(4-chlorophenyl)ethyl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
N,4-dimethyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-thiazole-5-carboxamide
N-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-methylbenzamide
2-(5-acetylthiophen-3-yl)-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
N-[4-(pyridin-2-yl)butyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-3-azaspiro[5.5]undecan-9-amine
{2-[4-(5-methoxy-1-methyl-1H-indole-2-carbonyl)morpholin-2-yl]ethyl}dimethylamine
[(3R,4R)-1-(6-chloro-4-methylquinolin-2-yl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
N-[2-(3,5-dimethylphenoxy)ethyl]-N-methyl-2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetamide
4-[4-(3,3-dimethylbutanoyl)piperazin-1-yl]-2-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2,3-dihydro-1H-isoindole-1,3-dione
2-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-4-methyl-1H-1,3-benzodiazole
1-[(2,4-dimethylphenyl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(dimethylamino)ethyl]acetamide
(2R,6S)-2,6-dimethyl-4-[5-(morpholin-4-ylmethyl)imidazo[2,1-b][1,3]thiazole-6-carbonyl]morpholine
4-(2-hydroxy-4-methoxybenzoyl)-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
methyl[(4-methyl-1H-imidazol-2-yl)methyl][(5-propylfuran-2-yl)methyl]amine
2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}ethan-1-one
ethyl 4-benzyl-1-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}piperidine-4-carboxylate
5-methyl-4-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-1-(4-methylphenyl)piperazin-2-one
5-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)pyrazin-2-ol
4-(4-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-6-methylpyrimidin-2-amine
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-[(4-fluorophenyl)methyl]-N-methylpropanamide
1,3-dimethyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-ethyl-1'-[3-(5-methylfuran-2-yl)butyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-[1-(ethylsulfanyl)ethyl]-1-(2-phenylethyl)-1H-1,2,4-triazole
1-(2-methoxybenzoyl)-4-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}piperazine
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-(1,2,5-thiadiazole-3-carbonyl)piperidine
3-(2-methylpropyl)-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-1,2-oxazole-5-carboxamide
6-cyclopentyl-1-methyl-N-[3-(methylamino)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
methyl 2-[(2-methylpropyl)sulfamoyl]-6-[(3,4,5-trifluorophenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N2-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-5-methylpyrimidine-2,4-diamine