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[1-(1H-imidazole-2-carbonyl)piperidin-4-yl](thiophen-2-yl)methanol
2-amino-4-(5-fluoro-2-methoxyphenyl)-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
N-[(3S,4R)-4-(4-methoxyphenyl)-1-{thieno[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl]acetamide
2-(3-hydroxypropyl)-8-(pyrazin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
1-benzyl-4-(2-tert-butyl-1H-imidazol-1-yl)piperidine
N-{4-[3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]phenyl}ethane-1-sulfonamide
4-({7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}methyl)phenol
4-{[3-(2-chlorophenoxy)azetidin-1-yl]methyl}pyridine
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl][2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amine
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-2-methyl-2-(thiophen-2-ylformamido)propanamide
N-[2-(4-chlorophenyl)-2-(pyrrolidin-1-yl)ethyl]-6-(methoxymethyl)pyridine-2-carboxamide
2-{1-[2-(1H-imidazol-1-yl)ethyl]-2,5-dioxo-3-phenylpyrrolidin-3-yl}-N-[(3-methoxyphenyl)methyl]-N-methylacetamide
N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}quinoxaline-6-carboxamide
2-(oxolan-2-ylmethyl)-9-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
3-[1-(cyclohex-1-ene-1-carbonyl)piperidin-3-yl]-N-(4-methoxy-2-methylphenyl)propanamide
4-{3-[5-(furan-2-yl)-4-phenyl-1H-imidazol-1-yl]propoxy}-1-methylpiperidine
1-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethan-1-one
N-methyl-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]propanamide
2-{1-[(3-methoxyphenyl)methyl]-4-(1-propylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
(4aS,7aR)-1-(3-hydroxy-2-methylbenzoyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{2-methylthieno[3,2-d]pyrimidin-4-yl}-1-(morpholine-4-carbonyl)piperidin-4-amine
1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-3-(3-methylphenoxymethyl)piperidine
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-ethyl-N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]acetamide
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-[3-(methylsulfanyl)propyl]benzamide
2,4-dimethyl-5-(2,3,4-trimethoxyphenyl)-1,3-thiazole
methyl 4-[({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)carbamoyl]butanoate
1-(1-ethylpiperidin-4-yl)-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
(2S,4S)-4-amino-1-(1,3-benzothiazole-5-carbonyl)-N-methylpyrrolidine-2-carboxamide
3-methyl-N-(1-{1-[2-(2-oxopyrrolidin-1-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)butanamide
4-{[1-methyl-10-oxo-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-4-yl]methyl}benzoic acid
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-(2-oxo-4-phenylpyrrolidin-1-yl)-N-(propan-2-yl)acetamide
2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(1-hydroxy-2-methylpropan-2-yl)acetamide
5-propyl-3-[2-(pyridin-2-yl)ethyl]-5-{1-[3-(thiophen-2-yl)propanoyl]piperidin-4-yl}imidazolidine-2,4-dione
(2R,3R,6R)-3-(3-methoxyphenyl)-5-(3-methyl-1H-pyrazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(1-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperidin-3-yl)-1,2,3,4-tetrahydroisoquinoline
7-(cyclobutylmethyl)-2-[3-(pyridin-2-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
(1S,5R)-3-[(2,3-dichloro-6-fluorophenyl)methyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{1-[(5-fluoro-2-methoxyphenyl)methyl]pyrrolidin-3-yl}benzoic acid
2-methyl-8-(quinolin-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-cyclopentyl-N-[(1R)-1-(3-methoxyphenyl)ethyl]-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
6-[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
methyl 4-{[4-(4-methoxyphenyl)-2-methyl-3-oxopiperazin-1-yl]methyl}benzoate
1-(2-{[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl](methyl)amino}ethyl)piperidin-2-one
2-amino-4-(1-ethyl-1H-pyrazol-4-yl)-6-(3-methylphenyl)pyridine-3-carbonitrile
N-[4-(4-{[3-(furan-2-yl)-3-phenylpropyl]amino}piperidin-1-yl)phenyl]pyrazine-2-carboxamide
6-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carboxylic acid
2-{5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}-2-azabicyclo[2.2.1]heptane
(1S,5R)-3-(oxan-4-yl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(2,3-dimethylphenyl)-N-(1-ethylpiperidin-4-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
3-(1H-1,3-benzodiazol-2-yl)-1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}propan-1-one