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ethyl 1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)-3-(2-phenoxyethyl)piperidine-3-carboxylate
8-(3-acetylbenzoyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-methyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-4-(pyridin-4-yl)pyrimidin-2-amine
(1S,5R)-6-propyl-3-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-{1-[(2-chlorophenyl)methyl]-3-methyl-1H-pyrazol-5-yl}-1-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]urea
N-cyclopropyl-5-[2-(2-methoxyphenoxy)acetyl]-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(3,4-difluorophenyl)methyl]-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(2-{1-[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]piperidin-2-yl}ethyl)pyrrolidin-2-one
N-(1-benzylpyrrolidin-3-yl)-3-(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)propanamide
3-{2-[2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
3-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-1-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}urea
(1R,5R)-6-propyl-3-(3-propyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-(2-methyl-1,3-thiazol-4-yl)-5-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]pyrimidin-4-ol
3,4-dimethoxy-N-(2-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}ethyl)benzamide
N-(2-phenylethyl)-1-[1-(1,3-thiazol-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(pyrazine-2-carbonyl)piperidin-3-ol
1-{4-[(1-benzothiophen-5-ylmethyl)amino]-2-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
2-(3-hydroxyphenyl)-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]acetic acid
1-[(3-fluorophenyl)methyl]-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
2-(2-{[2-(phenylsulfanyl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
3-({3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)pyridine
1-[(3,3-dimethylbutan-2-yl)amino]-3-(3-methoxyphenoxy)propan-2-ol
3-(hydroxymethyl)-1-[1-(6-methyl-2-phenylpyrimidin-4-yl)piperidin-4-yl]pyrrolidin-3-ol
3-({3-[3-(2-fluorophenyl)phenyl]-1H-pyrazol-1-yl}methyl)-5-methyl-1,2,4-oxadiazole
N-cyclopropyl-5-(phenoxymethyl)-N-(thiophen-3-ylmethyl)-1H-pyrazole-3-carboxamide
N-({7-[2-(4-chlorophenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
(1S,5R)-6-propyl-3-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
5-{[(5-fluoro-2-methylphenyl)methyl]amino}-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-1λ6-thiomorpholine-1,1-dione
1-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-3-methoxy-1,2-dihydropyridin-2-one
7-ethyl-2-[3-(3-methoxyphenyl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(2-oxo-1,2-dihydroquinolin-1-yl)acetamide
1-methyl-2-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-1H-1,3-benzodiazole
N-(2,5-difluorophenyl)-3-{4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}propanamide
methyl 2-{[2-(2-cyclohexylacetamido)-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazol-5-yl]formamido}-4-(methylsulfanyl)butanoate
N-[(3S,4R)-4-(4-methylphenyl)-1-[2-(piperidin-1-yl)acetyl]pyrrolidin-3-yl]acetamide
N-[(2-chloro-6-fluorophenyl)methyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
6-(2,5-dimethylfuran-3-yl)-8-oxo-7-(prop-2-en-1-yl)-N-[(1r,4r)-4-hydroxycyclohexyl]-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-(2,5-dimethoxyphenyl)-2-{5-methyl-4-[4-(piperidin-1-yl)piperidine-1-carbonyl]-1H-pyrazol-1-yl}pyrimidine
4-[3-(3-methoxypropyl)piperidin-1-yl]-2-methylpyridine
5-[7,8-dimethyl-4-(2-methylpyrrolidine-1-carbonyl)quinolin-2-yl]-N,N-dimethylpyrimidin-2-amine
N-methyl-1-[2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamido]cyclohexane-1-carboxamide
1-(3,5-dimethylphenyl)-4-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazin-2-one
{4-[5-(2-methyl-1,3-thiazol-4-yl)-1,2,4-oxadiazol-3-yl]phenyl}methanol
2-(dimethylamino)-N-methyl-2-(3-methylphenyl)-N-[2-(phenylsulfanyl)ethyl]acetamide
3-methoxy-1-(2-{3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydropyridin-2-one
4-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,3λ6,4-oxathiazinane-3,3-dione
methyl({[5-(4-methylpyrimidin-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl})[(3-methylthiophen-2-yl)methyl]amine
5-(oxolan-2-yl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)thiophene-2-carboxamide
N-(3-cyanothiophen-2-yl)-3-[(1,1-dioxo-1λ6-thiomorpholin-4-yl)methyl]benzamide