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N-(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)-2-(1,3-thiazol-2-yl)pyrrolidine-1-carboxamide
3-methyl-8-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-methoxy-N-[3-(4-{[1-(1,3-thiazol-2-yl)ethyl]amino}piperidin-1-yl)phenyl]benzamide
5-butyl-4-(2-fluoro-5-methylphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-(3-{1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}phenyl)imidazolidin-2-one
N-cyclohexyl-3-{[3-(4-hydroxyphenyl)phenyl]formamido}propanamide
1-[6-(morpholine-4-carbonyl)pyrazin-2-yl]azepan-4-amine
4-(benzyloxy)-1-[4-(3-hydroxypiperidin-1-yl)piperidin-1-yl]butan-1-one
3-fluoro-N-methyl-N-[1-(1,3-thiazol-5-yl)ethyl]imidazo[1,2-a]pyridine-2-carboxamide
2-{4-[2-(methylamino)pyridine-4-carbonyl]piperazin-1-yl}-1-(morpholin-4-yl)ethan-1-one
N-ethyl-5-{[4-(4-methylphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyrimidin-2-amine
2-{1-cyclopentyl-4-[(2,4-difluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
2-(1,1-dioxo-1λ6-thiolan-3-yl)-N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]acetamide
8-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(2-ethoxyethyl)-N-[(4-hydroxy-1-methylpiperidin-4-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-4-(1H-imidazol-2-yl)piperidine
N-cyclopropyl-N-{2-phenyl-1-[1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperidin-4-yl]ethyl}pyridine-2-carboxamide
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-4-(3-hydroxy-3-methylbutyl)benzamide
4-(4-methoxy-2-methylbenzoyl)-1-(2-methoxyphenyl)piperazin-2-one
3-(2-methoxyethyl)-1-(4-methoxyphenyl)-5-[(methylsulfanyl)methyl]-1H-1,2,4-triazole
5-(3-cyclobutyl-1H-1,2,4-triazol-5-yl)-8-methoxyquinoline
3-(2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}phenyl)-1H-1,2,4-triazole
N-[(2-ethoxypyridin-3-yl)methyl]-4-hydroxy-2-phenylpyrimidine-5-carboxamide
1-(cyclopropylmethyl)-5-(1H-indole-3-carbonyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)-2-(thiophen-3-yl)acetamide
(3S,4S)-4-cyclopropyl-1-[(6-methylpyridin-2-yl)methyl]pyrrolidine-3-carboxylic acid
1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-3-(3-methylthiophene-2-carbonyl)piperidine
5-{[3-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-3-propyl-1,2,4-oxadiazole
5-{3-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-1-methyl-3-(propan-2-yl)-1H-pyrazole
N-cyclopentyl-1-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)-1H-1,2,3-triazole-4-carboxamide
2-amino-6-(5-methylpyridin-2-yl)-4-(thiophen-2-yl)pyridine-3-carbonitrile
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
(3S,5R)-5-[(pyridin-3-ylmethyl)carbamoyl]-1-(1H-pyrrole-2-carbonyl)piperidine-3-carboxylic acid
2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-5-(piperidin-1-ylmethyl)pyridine
4-(2,4-dioxoimidazolidin-1-yl)-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)benzamide
1'-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-(piperidine-1-carbonyl)-2-[4-(1H-pyrazol-1-yl)phenyl]pyridine
1-{5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
(3R,4R)-1-[4-(4-fluorophenyl)oxane-4-carbonyl]-4-methyl-3-(propan-2-yl)pyrrolidin-3-ol
2-{1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-2-yl}acetic acid
methyl 8-(1,3-benzothiazol-2-ylmethyl)-1-(benzyloxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
1-{7-methylthieno[3,2-d]pyrimidin-4-yl}-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
{3-[(4-fluorophenyl)methyl]-1-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl}methanol
N-(4-fluorophenyl)-1-(2,3,4-trimethoxybenzoyl)piperidin-3-amine
3-[2-(carbamoylmethoxy)-5-methylphenyl]-N-cyclopropylbenzamide
methyl 4-methoxy-3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)benzoate
1-(5-methyl-1,2-oxazole-3-carbonyl)-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidine-3-carboxamide
N-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-1-propyl-1H-pyrazole-5-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1-[4-(1H-imidazol-1-yl)phenyl]piperidin-4-amine