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(3S,4S)-1-[(2-fluoro-5-methoxyphenyl)methyl]-4-(piperidin-1-yl)pyrrolidin-3-ol
N-cyclohexyl-2-[methyl(piperidin-4-yl)amino]-N-(pyridin-2-ylmethyl)acetamide
1-methyl-2-{1-[(5-methylfuran-2-yl)methyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
6-[(2-fluorophenyl)methoxy]-1-[(4-methoxyphenyl)methyl]-4-(pyridin-2-ylmethyl)-1,4-diazepan-2-one
N-(2-methoxyethyl)-3-(5-methylfuran-2-yl)-N-(1,3-thiazol-2-ylmethyl)-1H-pyrazole-5-carboxamide
1-(4-{5-fluoro-2-[(2-methoxyphenyl)methyl]-1H-1,3-benzodiazol-1-yl}piperidin-1-yl)butan-1-one
4-methyl-3-{2-[2-(4-phenyl-1,3-thiazol-2-yl)-1H-imidazol-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(azepan-1-yl)-2-phenylethyl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
2-{2-[(3-oxopiperazin-1-yl)methyl]-4-(pyridin-3-yl)phenoxy}acetic acid
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1H-1,2,3-benzotriazole-5-carboxamide
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-1-[6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]ethan-1-one
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[2-(5-methoxy-1H-indol-3-yl)ethyl]propanamide
4-(4-methyl-1H-imidazole-5-carbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
3-(1-{[1-(furan-3-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)pyridine
{4-[(2-chlorophenyl)methyl]-1-(2-phenylethyl)piperidin-4-yl}methanol
4-benzyl-3-{1-[2-(pyridin-3-yl)acetyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[4-(furan-2-carbonyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
3-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]propanamide
N,2-dimethyl-1-phenyl-N-(1H-pyrazol-3-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
1-{2-[4-(trifluoromethyl)phenyl]ethyl}-1H-imidazole
{5-[2-(3-phenyl-1,2-oxazol-5-yl)-1H-imidazol-1-yl]-1H-1,3-benzodiazol-2-yl}methanol
2-methoxy-5-{[methyl(quinolin-2-ylmethyl)amino]methyl}phenol
(3R,4R)-1-[8-chloro-2-(furan-2-yl)quinoline-4-carbonyl]-3,4-dimethylpyrrolidin-3-ol
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}thiophene-3-carboxamide
N-{[1-(cyclohex-2-en-1-yl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}-3-cyclopentylpropanamide
N-cyclopropyl-2-methyl-4-phenyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]pyrimidine-5-carboxamide
6-{4-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]piperazin-1-yl}pyrimidine-2,4-diamine
N-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-N-methyloxan-4-amine
2,6-dimethyl-4-(4-methyl-2-phenylpiperazine-1-carbonyl)quinoline
(2R,3R)-3-(1H-imidazol-1-yl)-1'-(pyrimidine-5-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidine-3-carbonyl)pyridine
2-methyl-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]-3-(1H-1,2,3,4-tetrazol-5-yl)urea
N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
1-benzyl-3-(2-methoxyethyl)-8-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-1,4,6-trimethyl-1,2-dihydropyridin-2-one
3-methoxy-N-methyl-4-[(1-methylpiperidin-4-yl)oxy]-N-[1-(pyridin-3-yl)ethyl]benzamide
[(2-cyclohexylpyrimidin-5-yl)methyl](methyl)[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]amine
1'-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-{2-[(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-3-hydroxypiperidin-1-yl]-2-oxoethyl}acetamide
[(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl](methyl)(pyridin-2-ylmethyl)amine
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-[5-(3-fluoro-4-methoxyphenyl)-1H-indazol-1-yl]acetamide
2-(4-fluorophenyl)-N-(2-{7-[(2,4,5-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
1-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}-2-(methylamino)ethan-1-one
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-ethyl-N-methyl-5-{1-[2-(1H-1,2,4-triazol-1-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
2-cyclopropanecarbonyl-1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
1-ethyl-N-[2-(2-methyl-1H-indol-3-yl)ethyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
3-{1-[3-(2-fluorophenyl)-1H-pyrazol-5-yl]-N-(pyridin-3-ylmethyl)formamido}propanoic acid