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2,5-dimethoxy-N-{1-oxa-8-azaspiro[4.5]decan-3-yl}benzamide
4-hydroxy-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-[(phenylsulfanyl)methyl]pyrimidine-5-carboxamide
N-(1H-imidazol-2-ylmethyl)-N-methyl-3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
2-{5-[3-cyclopropyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]-1H-pyrazol-3-yl}phenol
7-(4-methoxypyrimidin-2-yl)-N-[(2S)-oxolan-2-ylmethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-[3-(1H-imidazol-2-yl)piperidin-1-yl]-4-oxobutane-1-sulfonamide
[(4-cyclopropyl-5-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
5-[2-(3-ethoxy-4-methoxyphenyl)-1H-imidazol-1-yl]pyridine-3-carboxylic acid
3-methyl-3-[(5-methyl-1H-pyrazol-3-yl)methyl]-1-(2,2,4,4-tetrafluoro-2,4-dihydro-1,3-benzodioxin-6-yl)urea
N-(cyclobutylmethyl)-1-methyl-2-oxo-N-(oxolan-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
2-amino-8-(1-ethyl-1H-1,2,4-triazol-5-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
1'-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
2-(dimethylamino)-8-[4-(1H-1,2,4-triazol-1-yl)phenyl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
1-(4-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-[(2-methylpiperidin-1-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
(2S,4R)-4-amino-1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-N-ethylpyrrolidine-2-carboxamide
6-ethyl-3-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
4-(3-chloro-4-methoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-6-amine
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-1-methyl-4-phenylpiperidine-4-carboxamide
(4aS,8aR)-6-(3-methanesulfonylpropanoyl)-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
4-(3,3-diethylpyrrolidine-1-carbonyl)-2-(3-methoxyphenoxymethyl)-1,3-oxazole
N-ethyl-1-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-5-phenyl-1H-pyrrole-2-carboxamide
7-hydroxy-6-methoxy-4-(quinolin-4-yl)-1,2,3,4-tetrahydroquinolin-2-one
9-[3-(methylsulfanyl)propyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-3-[5-(2-methylbutan-2-yl)-1,3,4-thiadiazol-2-yl]-1-[1-(pyridin-2-yl)ethyl]urea
3-[1-(quinoline-6-carbonyl)piperidin-3-yl]benzoic acid
(3R,4S)-N,N-dimethyl-1-(5-methylthiophene-3-carbonyl)-4-(propan-2-yl)pyrrolidin-3-amine
2-methyl-6-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-2,3-dihydropyridazin-3-one
N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-(6-amino-2-{[(4-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)-4-(hydroxymethyl)piperidin-4-ol
3-[2-(cyclopropylmethyl)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
4,6-dimethyl-N-[2-(3-methylpyridin-2-yl)ethyl]pyrimidin-2-amine
5-{4-[1-(dimethylamino)ethyl]phenyl}-2-methoxybenzamide
4-(4-methoxyphenoxy)-1-(2-methyl-1,3-thiazole-5-carbonyl)piperidine
2-(3-chlorophenyl)-N-[4-(4-{[1-(thiophen-2-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
7-[(2S)-4,4-difluoropyrrolidine-2-carbonyl]-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-(4-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}piperazin-1-yl)-1-azabicyclo[2.2.2]octane
(3aS,6aS)-2-cyclobutanecarbonyl-5-[4-(trifluoromethyl)pyridin-2-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-(dimethylamino)-2-{2-[3-(2-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-2,3-dihydropyridazin-3-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]propanamide
2,6-dimethyl-4-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
2-(2-{[(1S)-1-cyclohexylethyl]amino}-4-(morpholin-4-yl)pyrimidin-5-yl)-2-methylpropanoic acid
3-(1-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)pyridine
3-hexyl-8-[2-(4-methylpiperazin-1-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]benzonitrile
1-(1,3-thiazol-2-yl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylic acid
4-(2-chloro-4-fluorophenyl)-2-methyl-1H-imidazole
2-[4-(5-cyclopropyl-1,3-oxazole-4-carbonyl)piperazin-1-yl]-4-methyl-6-(trifluoromethyl)pyrimidine
2-[methyl(pyridin-3-ylmethyl)amino]-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]acetamide
1-methyl-5-[4-(trifluoromethyl)phenyl]-1H,4H-pyrazolo[3,4-d]imidazole