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2-methoxy-N-{3-[4-(morpholin-4-ylmethyl)phenoxy]propyl}acetamide
5-{4-[1-(2-methoxyethyl)-5-oxopyrrolidine-3-carbonyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(2-methylpropyl)acetamide
9-(2,1-benzoxazole-3-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
N-[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-(3-ethoxypropyl)acetamide
N-{2-[2-(quinolin-2-yl)-1H-imidazol-1-yl]ethyl}pyridin-3-amine
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-5-(methoxymethyl)furan-2-carboxamide
1-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
6-(methoxymethyl)-2-[2-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
1-(4-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}phenyl)-1H-pyrazole
[3-(2-phenylethyl)-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl]methanol
2-methyl-4-(2-methylphenyl)-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperazine
1-(2,3-dihydro-1H-isoindol-2-yl)-3-[4-(3-methylphenyl)piperazin-1-yl]propan-1-one
7-{2-[(5-ethyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
4-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}thiomorpholine
1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-4-(2-methylpyridin-4-yl)-1,4-diazepane
N-ethyl-2-(4-methanesulfonyl-1,4-diazepan-1-yl)pyrimidin-4-amine
6-[2-(2,5-dioxopyrrolidin-1-yl)ethyl]-2-methoxy-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
1-{4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}propan-1-one
N5-cyclooctyl-N3-ethyl-N3-(2-methylprop-2-en-1-yl)-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-(dimethylamino)-4-methyl-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)pyrimidine-5-carboxamide
2-[(1-{5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-yl}piperidin-4-yl)amino]acetamide
N-[2-(dimethylamino)ethyl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
2-{[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]methyl}-1H-1,3-benzodiazole
1-methyl-3-{[3-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
6-(4-fluorophenyl)-N-[2-methyl-1-(morpholin-4-yl)propan-2-yl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-methyl-4-[(1-methyl-1H-imidazol-5-yl)methyl]-1-phenylpiperazin-2-one
4-[3-({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)propyl]piperazin-2-one
4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]benzamide
(1S,4S)-2-{5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-yl}-2-azabicyclo[2.2.1]heptane
[(2-chloro-6-fluorophenyl)methyl]({[2-(2-methoxyphenoxy)pyridin-3-yl]methyl})amine
5-{[4-(1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}-2-(pyridin-2-yl)pyrimidine
3-(1-ethyl-1H-imidazol-2-yl)-N-(4-methoxyphenyl)piperidine-1-carboxamide
1-(cyclohexylmethyl)-3-({[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-3-hydroxypiperidin-2-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1,5-dimethyl-4-{[methyl(1,2,3,4-tetrahydronaphthalen-1-yl)amino]methyl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
7-(4-phenoxybutanoyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
N-({1-[(5-ethylpyridin-2-yl)methyl]piperidin-4-yl}methyl)-3-methylfuran-2-carboxamide
3-chloro-4-fluoro-N-[1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]-1-benzothiophene-2-carboxamide
1-butyl-3-cyclopropyl-5-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-1,2,4-triazole
3-{2-[2-(pyridin-2-yl)pyrrolidin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
2-({[5-(pyrimidin-2-ylsulfanyl)furan-2-yl]methyl}amino)-N-(1,3-thiazol-2-yl)acetamide
2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}-1,3-thiazole-4-carboxamide
ethyl 1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-4-(2-phenylethyl)piperidine-4-carboxylate
3-({4-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)pyridine
N-cyclopropyl-3-({1-[(4-fluorophenyl)methyl]piperidin-4-yl}oxy)-4-methoxybenzamide
N-methyl-1-[2-(morpholin-4-yl)ethyl]-6-oxo-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)piperidine-3-carboxamide
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}quinoxalin-2-amine
(3S,4R)-1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid