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3-hydroxy-3-{[(oxan-4-yl)amino]methyl}-1-(3-phenylpropyl)piperidin-2-one
1-cyclopentyl-5-oxo-N-[2-(pyridin-2-ylsulfanyl)ethyl]pyrrolidine-3-carboxamide
2-(4-{[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]amino}piperidin-1-yl)pyridine-4-carbonitrile
1-(2-methoxyethyl)-3-[3-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]-1-(pyridin-3-ylmethyl)urea
1-(1-benzofuran-5-ylmethyl)-4-[(3-fluorophenyl)methyl]piperazine
2,8-dimethyl-N-[2-(pyridin-2-ylsulfanyl)ethyl]quinoline-4-carboxamide
1-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-methoxyethan-1-one
N-[2-(diethylamino)ethyl]-4-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridine-2-carboxamide
3-{1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]piperidin-4-yl}-N-[2-(dimethylamino)ethyl]propanamide
2-(3-cyanopiperidin-1-yl)-6-methylpyridine-3-carboxylic acid
3-({1-[2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetyl]pyrrolidin-3-yl}methyl)benzoic acid
2-{4-[6-(azepan-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazin-1-yl}ethan-1-ol
2-[1-(2-methoxyphenyl)-5-(4-propylpyrimidin-5-yl)-1H-1,2,4-triazol-3-yl]acetamide
(2R,3R,6R)-5-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{[5-(2-chlorophenyl)-1,2-oxazol-3-yl]methyl}-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
(1R,7S)-N-methyl-3-(3-methylbutyl)-4-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-butyl-4-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(3S,4R)-1-[(5-ethylfuran-2-yl)methyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
(1S,5R)-6-(cyclopropylmethyl)-3-{[2-(methylsulfanyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-(1-methylpiperidin-2-yl)ethyl]-6-[(2-methylpropyl)amino]pyridine-3-carboxamide
4-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]benzamide
N-[2-(tert-butylsulfanyl)ethyl]-5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
4-(cyclopropylsulfamoyl)-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]benzamide
4-methyl-1-[(3-methylquinoxalin-2-yl)methyl]pyrrolidin-2-one
N-[3-(4-{[2-(1,3-thiazol-4-yl)ethyl]amino}piperidin-1-yl)phenyl]-3-(trifluoromethyl)benzamide
4-(3-hydroxybenzoyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(2-hydroxy-3-methoxybenzoyl)-1-(4-methylphenyl)piperazin-2-one
N-(4-{[3-(2-hydroxyethyl)-4-(propan-2-yl)piperazin-1-yl]methyl}phenyl)acetamide
N-[2-(adamantan-1-yl)-2-hydroxyethyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
2-[4-(6-methoxypyrimidin-4-yl)-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-propyl-1H-1,2,4-triazole
N,2-dimethyl-7-oxo-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
methyl (2S,4S)-1-methyl-4-{1-[(4-methylphenyl)amino]cyclopentaneamido}pyrrolidine-2-carboxylate
7-(methylsulfanyl)-3-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
8-(2-methoxypyridine-4-carbonyl)-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-amino-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}cyclopropane-1-carboxamide
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-6-methylpyridine-3-carboxamide
1-{1-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-1-oxopropan-2-yl}pyrrolidin-2-one
2-{[(1-hydroxycyclohexyl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
3-(1,4-diazepane-1-carbonyl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)benzene-1-sulfonamide
N-[5-({[2-(4,6-dimethylpyrimidin-2-yl)ethyl]carbamoyl}amino)-2-methoxyphenyl]acetamide
1-(5-{[(2S)-4-methyl-2-phenylpiperazin-1-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carbonyl)azocane
7-fluoro-3-methyl-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)-1-benzofuran-2-carboxamide
5-(4-methylpiperidine-1-carbonyl)-4-oxo-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]pyrrolidine-1-sulfonamide
3-[5-({methyl[(5-methyl-1H-pyrazol-3-yl)methyl]amino}methyl)thiophen-2-yl]prop-2-yn-1-ol
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]pyrrolidine-1-sulfonamide
methyl 5-cyano-6-{[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]amino}-2-methylpyridine-3-carboxylate
5-[4-oxo-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1,2-dihydropyridin-2-one
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-4H-thieno[3,2-b]pyrrole-5-carboxamide