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4-{[ethyl(pyridin-4-ylmethyl)amino]methyl}-N-(1,3,4-thiadiazol-2-yl)benzamide
2-{2-[1-(3-fluoropyridin-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
(9aR)-2-methyl-8-(3-methylbutyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-hydroxy-1-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}butan-1-one
4-(3-{1-[(1-methyl-1H-imidazol-5-yl)methyl]-1H-pyrazol-3-yl}phenyl)-6-(4-methyl-1H-pyrazol-1-yl)pyrimidine
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carboxamide
N-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(4-fluorophenyl)methyl]-N-[(2-methoxyphenyl)methyl]pyrrolidine-2-carboxamide
9-(2,3-dihydro-1H-indene-1-carbonyl)-2-[2-(dimethylamino)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[cyclohexyl(methyl)amino]-3-(2-{[(1-phenylcyclopropyl)amino]methyl}phenoxy)propan-2-ol
1-[(2,6-difluoro-3-methoxyphenyl)methyl]-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine
2-(2,4-dioxoimidazolidin-1-yl)-N-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}acetamide
6-[1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]pyrimidin-4-ol
1-methyl-4-({2-methyl-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-7-yl}methyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
(2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}quinolin-3-yl)methanol
3,4,7-trimethyl-2-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]-1H-indole
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-oxo-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-3,4-dihydrophthalazine-1-carboxamide
2-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}benzonitrile
ethyl 2-({5-[6-oxo-3-(propan-2-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl]pyrimidin-2-yl}amino)acetate
N-methyl-2-(2-oxopiperidin-1-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
6-{6-oxo-7-propyl-2,7-diazaspiro[4.5]decan-2-yl}pyridine-3-carboxylic acid
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(1H-imidazol-2-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
(1R,5R)-3-[1-(3,4-dimethoxyphenyl)cyclopentanecarbonyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonane
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-3-(1H-pyrazol-1-yl)butanamide
1-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
1-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
4-{[1-(5-ethyl-1,3-oxazole-4-carbonyl)pyrrolidin-3-yl]methyl}benzoic acid
2-[2-chloro-6-methoxy-4-({methyl[1-(1,3-thiazol-2-yl)ethyl]amino}methyl)phenoxy]acetic acid
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methylazepane-2-carboxamide
4-{[4-(morpholin-4-yl)piperidin-1-yl]methyl}-N-(1,2,3-thiadiazol-5-yl)benzamide
3-{3-[(dimethylsulfamoyl)amino]phenyl}-1-[(4-methyl-1,4-oxazepan-6-yl)methyl]urea
dimethyl(1-{1-[4-methyl-6-(methylsulfanyl)quinolin-2-yl]piperidin-4-yl}ethyl)amine
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]acetamide
(3S,4S)-1-[1-(oxan-4-yl)piperidine-4-carbonyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
(4aS,8aR)-1-(3-hydroxypropyl)-6-[2-(methylamino)pyridine-4-carbonyl]-decahydro-1,6-naphthyridin-2-one
1-{1-[(4-ethoxyphenyl)methyl]piperidin-4-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
N-[(1-propyl-1H-pyrazol-4-yl)methyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
(4S,4aS,8aS)-1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-4-phenyl-decahydroquinolin-4-ol
6-fluoro-2-[2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazole
4-[1-(2,6-dimethylphenoxy)propan-2-yl]-4H-1,2,4-triazole
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N,N-bis(prop-2-en-1-yl)acetamide
N-[(2-chlorophenyl)methyl]-2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(1-benzothiophen-2-ylmethyl)[(4-{2-[4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl]methylamine
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-[4-(propan-2-yl)benzoyl]pyrrolidin-3-yl]methanol
1-phenyl-4-{[1-(propan-2-yl)piperidin-4-yl]methyl}piperazin-2-one
2-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-6-methylpyridine-3-carbonitrile
2-ethoxy-N-[(2-methoxyphenyl)methyl]-N-(pyridin-3-ylmethyl)benzamide
2-[(2S)-2-(methylamino)propanoyl]-N-(pyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide