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6-methoxy-3-{[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]methyl}quinolin-2-ol
5-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonane-7-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl][(2-ethylpyrimidin-4-yl)methyl]methylamine
4-[(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)amino]-1-[2-(4-methoxyphenyl)ethyl]pyrrolidin-2-one
2-(dimethylamino)-2-(3-fluorophenyl)-1-[3-(pyridin-3-yl)azetidin-1-yl]ethan-1-one
4,4-difluoro-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidine
1-[1-(1-methylpiperidine-2-carbonyl)piperidin-4-yl]-2-(phenoxymethyl)-1H-1,3-benzodiazole
3,5-dimethyl-2-[3-(pyridin-3-yl)azetidine-1-carbonyl]-1H-indole
3-methyl-N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]pyridine-2-carboxamide
N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-2-(pyridin-2-yl)acetamide
4-[3-(3-methyl-1H-pyrazol-1-yl)phenyl]-4H-1,2,4-triazole
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-[3-(naphthalen-2-yl)-1H-pyrazol-1-yl]acetamide
2-ethyl-N-{[3-(2-methoxyphenyl)-1,2-oxazol-5-yl]methyl}pyrimidine-5-carboxamide
4-[3-(1H-pyrazol-1-yl)benzoyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
3,5-dimethyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]benzamide
3-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1-[3-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]urea
5-methyl-N-{4-[2-(oxolan-3-yl)-1H-imidazol-1-yl]phenyl}furan-2-carboxamide
3-(2-hydroxyphenyl)-N-[(1R,2S)-2-phenylcyclohexyl]-1H-pyrazole-5-carboxamide
N-[(2,6-difluoro-3-methylphenyl)methyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(4-{9-oxa-2-azaspiro[5.5]undecan-2-ylmethyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol
1-[2-(4-chlorophenyl)ethyl]-N-(1H-indol-4-ylmethyl)-6-oxopiperidine-3-carboxamide
N-methyl-2-propyl-N-[1-(pyridin-3-yl)pentyl]-1,3-thiazole-4-carboxamide
1-(3-fluorophenyl)-4-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-3-(5-methylfuran-2-yl)-1H-pyrazole
methyl 5-(2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
(3R,4S)-N,N-dimethyl-1-[2-(morpholin-4-yl)benzoyl]-4-propylpyrrolidin-3-amine
2-hydroxy-4-methyl-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}benzamide
4-(4-methyl-5-{[2-(piperidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)-1-[3-(5-methylfuran-2-yl)butyl]piperidine
1-methyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(4-methoxyphenyl)methyl]acetamide
N-[(4-methoxyphenyl)methyl]-3-{2-methyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}propanamide
N-(1-methoxybutan-2-yl)-2-(1H-1,2,4-triazol-3-yl)benzamide
N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-3-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]thiophene-2-carboxamide
2-{5-[(2R)-2-(hydroxymethyl)pyrrolidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
N-ethyl-N-methyl-2-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)acetamide
N-[(2-chlorophenyl)methyl]-3-acetamido-N-(prop-2-en-1-yl)propanamide
1-[4-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)piperidin-1-yl]ethan-1-one
3-(2-methyl-1H-imidazol-1-yl)-1-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
2-{1-[(3,4-difluorophenyl)methyl]-4-(quinoxalin-5-ylmethyl)piperazin-2-yl}ethan-1-ol
2-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidine-1-carbonyl]-4H-chromen-4-one
1-(3-hydroxyphenyl)-N-methyl-5-oxo-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}pyrrolidine-3-carboxamide
2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
1-[2-(benzyloxy)ethyl]-4-(1H-pyrazole-4-carbonyl)-1,4-diazepan-6-ol
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-4-amine
2-[1-(difluoromethyl)-3-methyl-1H-pyrazol-4-yl]-6-methoxy-N,N-bis(propan-2-yl)benzamide
11-(5-chloro-2,4-dimethoxyphenyl)-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
N-methyl-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]-N-[(5-propyl-1H-pyrazol-3-yl)methyl]acetamide
(3R,4R)-3-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]-1-methylpiperidin-4-ol
5,6-dimethyl-2-[4-({methyl[(3-methylthiophen-2-yl)methyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
5-ethyl-N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]thiophene-3-carboxamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanamide