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N,N-dimethyl-1-[3-(1H-1,2,4-triazol-1-yl)adamantane-1-carbonyl]azepan-4-amine
6-[(diethylamino)methyl]-N-[(5-methylpyrazin-2-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1,4-diazepane
(1R,3S)-3-amino-N-[(3-phenylphenyl)methyl]cyclohexane-1-carboxamide
2-(2-{1-[2-(oxolan-2-ylmethoxy)acetyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-3-(pyridin-2-yl)propanamide
methyl({[4-phenyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl})[1-(pyridin-2-yl)ethyl]amine
3,5,7-trimethyl-2-(3-phenoxyazetidine-1-carbonyl)-1H-indole
4-(2-phenoxyethyl)-1-(thiophen-2-ylmethyl)-1,4-diazepan-5-one
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-1,3-thiazole-4-carboxamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-(3-methylbutyl)benzamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(5-methylfuran-2-yl)methyl]pyrrolidin-3-yl]-6-oxo-1,6-dihydropyridine-3-carboxamide
[(2S,6S)-11-methoxy-4-[3-(trifluoromethyl)pyridin-2-yl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
2-{6-[(pyridin-4-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,3-thiazole-4-carboxamide
7-methyl-3-({[1-(2-methyl-1,3-thiazol-4-yl)ethyl]amino}methyl)-1-[(3-methylphenyl)methyl]-1,2-dihydroquinolin-2-one
1-(2,5-dimethoxyphenyl)-3-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}urea
4-pentanamido-N-[2-(pyridin-3-yloxy)propyl]benzamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-5-(2-methoxy-4-methylphenoxymethyl)-1,2-oxazole-3-carboxamide
5-{1-[(2-methylphenyl)methyl]pyrrolidin-2-yl}-N-(pyridin-4-yl)thiophene-2-carboxamide
8-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-[1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1H-pyrazol-3-yl]-4-methyl-N-(thiophen-2-ylmethyl)-1,3-thiazol-2-amine
(1S,5R)-6-(cyclobutylmethyl)-3-(4-ethylbenzenesulfonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-{5-[5-(methoxymethyl)furan-2-yl]-3-(pyridin-2-yl)-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
2-[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]-1H-imidazole
5-(2,1,3-benzoxadiazol-5-ylmethyl)-N-(2-hydroxyethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-(3-methanesulfonamidophenyl)-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
1-{4-[(3S)-3-hydroxypyrrolidin-1-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl}cyclopropane-1-carbonitrile
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-3-(3-methoxyphenyl)propan-1-one
1-(3-cyclopropyl-1,2-oxazole-5-carbonyl)-3-[2-(4-fluorophenyl)ethyl]piperidine
N-cyclohexyl-3-(3-hydroxy-3-methylbutyl)-N-(2-hydroxyethyl)benzamide
1-(2-chlorophenyl)-3-(1-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
(1S,6R)-9-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
(3S)-3-benzyl-4-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperazin-2-one
3-[2-(4-fluorophenoxy)ethyl]-5,5-dimethyl-1,3-oxazolidine-2,4-dione
2-butyl-8-(1,3-thiazol-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
5-{[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]amino}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
2-chloro-5-acetamido-N-(2-hydroxy-2-phenylethyl)benzamide
3-[1-(3-phenyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]benzoic acid
4-{[(trimethylpyrimidin-4-yl)amino]methyl}hexane-1,4-diol
4-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-2-[(3-methoxyphenyl)methyl]morpholine
3-{methyl[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]amino}propane-1,2-diol
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]pyrrolidin-3-yl]methanol
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-(3-butyl-4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)acetamide
1-{2-[2-(3-methoxyphenyl)azetidin-1-yl]-2-oxoethyl}piperidine-4-carboxamide
1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
ethyl 4-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperazine-1-carboxylate
3-(3-hydroxyquinoxalin-2-yl)-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)propanamide
N-(1-oxo-1,3-dihydro-2-benzofuran-5-yl)-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carboxamide
2-(3-methoxyphenoxy)-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}propan-1-one