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methyl 5-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-ethyl-2-({2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}sulfanyl)-1H-1,3-benzodiazole
1-(3-{[4-(4-fluorophenyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)propan-1-one
4-(1-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}piperidin-3-yl)pyrimidine
N-(2,3-dihydro-1H-inden-2-yl)-4-methyl-N-propylpyrimidine-5-carboxamide
6-ethyl-N-[2-hydroxy-3-(piperazin-1-yl)propyl]-2-methylquinoline-4-carboxamide
2-methoxy-2-methyl-N-{1-phenyl-3,6-diazatricyclo[4.3.1.13,8]undecan-9-yl}propanamide
3-[(4aR,7aS)-4-[(4-fluoro-3-methylphenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
5-(2-chloroprop-2-en-1-yl)-7-[(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
1-(1-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}piperidin-4-yl)-3-(pyrrolidine-1-carbonyl)piperidine
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-3-azaspiro[5.5]undecan-9-amine
1-methyl-5-{[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]sulfanyl}-1H-1,2,3,4-tetrazole
4-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methylpyrimidine
N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
3-(5-{2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
N-{[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(pyridin-2-yl)pyrimidin-2-amine
N-(2,3-dihydro-1H-inden-2-yl)-2-(2,2-dimethylpropanamido)-N,5-dimethylthiophene-3-carboxamide
[5-(1-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}-1H-1,2,3-triazol-4-yl)furan-2-yl]methanol
2-[(3,4-difluorophenyl)methyl]-8-(oxolane-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
3-fluoro-N-{1-[1-(thiophene-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
N2,N4,N4,5-tetramethyl-N2-(pyrimidin-4-ylmethyl)pyrimidine-2,4-diamine
2-(4-benzylmorpholin-2-yl)-1-[3-(pyridin-2-yl)azetidin-1-yl]ethan-1-one
2-amino-N-[2-(4-hydroxypiperidin-1-yl)-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl]-2-methylpropanamide
N-(2,1,3-benzothiadiazol-4-yl)-4-methanesulfonylpiperazine-1-carboxamide
N,1-dimethyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-5-phenyl-1H-pyrrole-2-carboxamide
3-{[1-(6-methylpyrimidin-4-yl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
1-(2,4-difluorophenyl)-4-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-3-(2-methylphenyl)-1H-pyrazole
(2S,4S)-4-amino-N-methyl-1-{[4-(methylsulfamoyl)phenyl]methyl}pyrrolidine-2-carboxamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-6-(2-methoxyphenyl)pyridazin-3-amine
N4-[(4-methylphenyl)methyl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
[(4aS,8aR)-1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-6-(pyrazin-2-yl)-decahydro-1,6-naphthyridin-4a-yl]methanol
4-[(3-fluorophenyl)methyl]-1-(2-methyl-1,3-thiazole-4-carbonyl)-1,4-diazepan-5-one
N-[(5-phenyl-1H-pyrazol-3-yl)methyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
4-(2-methyl-1H-imidazol-1-yl)-1-[2-(thiophen-3-yl)acetyl]piperidine-4-carboxylic acid
6-chloro-N,N-dimethyl-3-[(4-methyl-3-phenylpiperazin-1-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
1-{7-[cyclohexyl(methoxy)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethan-1-one
4-(3-carbamoylpyridin-2-yl)-N-[3-methyl-1-(propan-2-yl)-1H-pyrazol-5-yl]piperazine-1-carboxamide
2-(5-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)-N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)acetamide
(1R,5R)-6-(3-methylbut-2-en-1-yl)-3-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-1-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
4-(4,6-dimethylpyrimidin-2-yl)-N-(5-methyl-4H-1,2,4-triazol-3-yl)piperazine-1-carboxamide
N-[2-(dimethylamino)ethyl]-N-[(5-methylthiophen-2-yl)methyl]-2-(pyridin-4-yl)acetamide
3-(3-methoxypyrazin-2-yl)quinoline
6-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]-9H-purin-2-amine
3-(4-methanesulfonyl-1,4-diazepan-1-yl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraene
4-methyl-N-[4-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]-1,2,3,6-tetrahydropyridine-1-carboxamide
N-[(5-chloro-2-methoxyphenyl)methyl]-1-(2-methoxyethyl)-N-methyl-6-oxopiperidine-3-carboxamide
[(4-{1-[1-(methoxymethyl)cyclobutanecarbonyl]piperidin-2-yl}phenyl)methyl]dimethylamine
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-1-[2-(1H-pyrazol-1-ylmethyl)pyrrolidin-1-yl]propan-1-one
4-(piperidin-4-yl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol