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N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
5-benzyl-3-(pyridin-3-ylmethyl)-5-{1-[(2,4,5-trimethylphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
1-[(2-methoxyphenyl)methyl]-N-(3-methylbutyl)-4-oxo-5-[4-(propan-2-yl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
1-(4-amino-5-methylpyrimidin-2-yl)-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylic acid
1-[(3-{1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)methyl]pyrrolidine
4-{2-[3-(trifluoromethyl)phenyl]acetyl}piperazine-1-sulfonamide
methyl 3-(2-methylbutanamido)-1-(oxolan-2-ylmethyl)-5-[(propan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
ethyl 2-{2-benzyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-1,3-oxazole-4-carboxylate
3-{1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]pyrrolidin-2-yl}pyridine
3-acetyl-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-1H-pyrazole-5-carboxamide
5-(methoxymethyl)-N-methyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]thiophene-2-carboxamide
[(2S,6S)-4-{[2-(propylamino)pyrimidin-5-yl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
3-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-5,6,7,8-tetrahydroquinoline
1-ethyl-5-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-3-(oxan-4-yl)-1H-1,2,4-triazole
4-[(2-fluorophenyl)methyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine
N-(3-hydroxypropyl)-1-(1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
methyl 3-acetamido-5-[(3-hydroxy-3-methylbutan-2-yl)amino]-1-[2-(1H-indol-3-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(2-methoxyethyl)-9-(5-propylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-(2-{1-[3-(4-methylphenyl)propanoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
1-[7-(3-chlorophenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methoxyethan-1-one
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-7-(2-methoxyacetamido)-N,1-dimethyl-2-phenyl-1H-1,3-benzodiazole-5-carboxamide
7-{[ethyl(pyridin-4-ylmethyl)amino]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
3-(1-benzothiophen-7-yl)-1-(cyclopropylmethyl)-6-[1-(pyridin-2-yl)propan-2-yl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-3-(pyridin-3-yl)propan-1-one
1-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]-2-(2-methylphenoxy)ethan-1-one
2-(3-methoxypropyl)-8-[2-(2-methylphenyl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
2-{4-[(5-ethylpyridin-2-yl)methyl]piperazin-1-yl}-N-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
3-{1-[2-(5-oxopyrrolidin-2-yl)acetyl]piperidin-4-yl}-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
[(1,3-dimethyl-1H-pyrazol-5-yl)methyl](methyl)[1-(4-methylpyridin-2-yl)propan-2-yl]amine
[4-({2-[2-(dimethylamino)ethoxy]-3-methoxyphenyl}methyl)-1-methylpiperazin-2-yl]methanol
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
[(2E)-3-(furan-2-yl)prop-2-en-1-yl]({2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl})amine
N-[(4-fluorophenyl)methyl]-5-[(2-hydroxyethyl)amino]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(2-{[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]amino}-4-methylpyrimidin-5-yl)ethan-1-one
N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}-3-(pyridin-2-yl)propanamide
3-(1-butyl-1H-imidazol-2-yl)-1-(2,3-dimethoxybenzoyl)piperidine
4-(1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)pyrimidine
N-[(4-methyl-1,3-benzoxazol-2-yl)methyl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
4-[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]benzene-1-sulfonamide
2-(4-{[cyclopropyl(thiophen-3-ylmethyl)amino]methyl}phenyl)-6-ethyl-3,4-dihydropyrimidin-4-one
2,3,5-trimethyl-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-N,4,6-trimethyl-2-oxo-2H-pyran-5-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}acetamide
1-[1'-(1-ethylpiperidine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
1-(1-cyclohexylpiperidin-4-yl)-N-cyclopropylpiperidine-3-carboxamide
4-(2-chlorophenoxy)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine
2-amino-4-[3-(4-fluorophenyl)-1H-pyrazol-4-yl]-6-(pyridin-3-yl)pyridine-3-carbonitrile
(3R,4S)-1-[1-methyl-5-(thiophen-2-yl)-1H-pyrazole-3-carbonyl]-4-propylpyrrolidin-3-amine