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1-[(4aR,8aS)-6-[2-(4-methoxyphenyl)acetyl]-decahydro-1,6-naphthyridin-1-yl]-2-(cyclohex-1-en-1-yl)ethan-1-one
N-(3,4-dimethoxyphenyl)-1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperidin-3-amine
1-(isoquinoline-3-carbonyl)-N,N-dimethylazepan-4-amine
N-[2-(dimethylamino)ethyl]-N-[(3-methylthiophen-2-yl)methyl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
[(5-methylthiophen-2-yl)methyl]({[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl})(pyridin-4-ylmethyl)amine
2-[3-(5-chlorothiophen-2-yl)-4-methyl-1H-pyrazol-1-yl]-N-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)acetamide
N-butyl-1-ethyl-N-(furan-2-ylmethyl)-3,5-dimethyl-1H-pyrazole-4-carboxamide
1-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-3-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}urea
2-(4-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
3-[3-({[3-(2,3-dihydro-1H-indol-1-yl)propyl]amino}methyl)-1H-indol-1-yl]propanamide
6-methyl-5-{5-[1-(pyrrolidin-1-yl)propyl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
[7-(1H-indazol-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
1-methyl-5-[4-(pyridin-4-yl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
2-({[(3R,4R)-1-(5-fluoro-1,3-dimethyl-1H-indole-2-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
(3S,4S)-1-(4-methoxybenzoyl)-4-(thiomorpholin-4-yl)pyrrolidin-3-ol
(1R,4S)-N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1,7,7-trimethyl-3-oxo-2-oxabicyclo[2.2.1]heptane-4-carboxamide
N-[3-(1H-imidazol-5-yl)phenyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
2-(3,4-dimethoxyphenyl)-1-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}ethan-1-one
4-{1-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]piperidin-3-yl}benzoic acid
2-(5-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline
2-(naphthalen-1-yl)-1-[2-(pyrrolidin-1-yl)ethyl]-1H-imidazole
3-{1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-4-yl}-N-phenylpropanamide
(3R,4R)-4-(azepan-1-yl)-1-[(5-ethylfuran-2-yl)methyl]piperidin-3-ol
3-(azepan-1-ylmethyl)-1-[(2,3-difluorophenyl)methyl]-3-hydroxypiperidin-2-one
N-[2-(6-hydroxypyrimidin-4-yl)ethyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
1-[(2-fluorophenyl)methyl]-6-oxo-N-[2-(2-oxoimidazolidin-1-yl)ethyl]piperidine-3-carboxamide
2-(2-{[(3S,4R)-4-amino-3-methoxypiperidin-1-yl]methyl}-4-(pyrimidin-2-yl)phenoxy)acetic acid
(2S)-2-amino-N-ethyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]-3-(1,3-thiazol-4-yl)propanamide
4-methyl-N-(2-phenylethyl)-N-(pyridin-3-ylmethyl)pyrimidine-5-carboxamide
N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
1-(3-cyano-4-methylphenyl)-3-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(2-methoxyethyl)urea
2-methanesulfonamido-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]acetamide
8-(3-phenyl-1,2,4-oxadiazol-5-yl)-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
2-{4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
3-(5-{[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
3-(1-butyl-1H-imidazol-2-yl)-1-[2-(trifluoromethyl)benzoyl]piperidine
5-[3-(4-fluorophenyl)propyl]-1-(propan-2-yl)-1H-1,2,4-triazole
3-(1H-imidazol-1-ylmethyl)-4-(2-methoxy-5-methylphenyl)-4H-1,2,4-triazole
8-[2-methyl-2-(morpholin-4-yl)propanoyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
(3R,4S)-3-[(2,5-dimethylpyrimidin-4-yl)amino]-N,N-dimethyl-4-propylpyrrolidine-1-sulfonamide
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-[(5-methylfuran-2-yl)methyl]piperidine
(2S,4R)-N,N-diethyl-1-methyl-4-(7-methyl-2,3-dihydro-1,4-benzodioxine-6-amido)pyrrolidine-2-carboxamide
8-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
N-(1H-1,2,3,4-tetrazol-5-ylmethyl)-5,6,7,8-tetrahydroquinoline-3-carboxamide
N-[(3S,4R)-1-[3-(3,4-dimethoxyphenyl)propanoyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
N-[2-(azepan-1-yl)ethyl]-N-ethyl-2-(5-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetamide
ethyl 3-[(2,4-difluorophenyl)methyl]-1-[3-(2-oxopyrrolidin-1-yl)propanoyl]piperidine-3-carboxylate
4-[(4-fluorophenyl)methyl]-1-(2-hydroxyacetyl)-3-(propan-2-yl)-1,4-diazepan-5-one
4-(3-fluorophenoxy)-1-(3-methoxypyrazin-2-yl)piperidine-4-carboxylic acid