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N-(cyclopent-3-en-1-yl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
(1R,5R)-6-benzyl-3-(2,3-difluoro-4-methylbenzoyl)-3,6-diazabicyclo[3.2.2]nonane
N-(oxan-4-yl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-(5-chloro-2-methoxyphenyl)-3-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]propanamide
(1S,6R)-9-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
9-(2-methyl-5-propylpyrimidin-4-yl)-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(4-chlorophenyl)ethyl]-2-[4-(morpholin-4-yl)piperidin-1-yl]acetamide
1-propyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1H-pyrazole-5-sulfonamide
7-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-4-yl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(cyclohexylmethyl)-3-hydroxy-3-{[4-hydroxy-4-(pyridin-2-yl)piperidin-1-yl]methyl}piperidin-2-one
4-(pyrrolidin-1-ylmethyl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)benzamide
3-amino-1-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-3-(3,4-dimethoxyphenyl)propan-1-one
(2S,4S)-1-{[4-(diethylamino)phenyl]methyl}-4-{[(4-methoxynaphthalen-1-yl)methyl]amino}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
2-[(4aR,7aS)-4-(oxane-4-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
3-{[(3,4-dihydro-2H-1-benzopyran-3-yl)amino]methyl}phenol
4-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-3-(propan-2-yl)piperazin-2-one
1-methyl-4-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperazine-2-carboxylic acid
N-benzyl[(4,5,6,7-tetrahydro-1H-indazol-5-yl)amino]sulfonamide
1-[(2-cyclohexylpyrimidin-5-yl)methyl]-N-methylpiperidine-2-carboxamide
[1-(furan-3-ylmethyl)-3-(2-phenoxyethyl)piperidin-3-yl]methanol
1-cyclopentyl-4-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyrrolidin-2-one
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}acetamide
1-[(2R,3R)-3-(dimethylamino)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-(4-methylphenyl)ethan-1-one
N-(1-cycloheptylpiperidin-3-yl)-2-(4-methoxyphenyl)acetamide
1-(3-aminoazepan-1-yl)-3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propan-1-one
2-{[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]oxy}pyrimidine
(4aR,7aS)-1-benzyl-4-(4-methylpyrimidine-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-4-oxobutane-1-sulfonamide
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-3-phenylpyrrolidin-3-ol
2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
2-{4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-1-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
8-fluoro-3-(2-methoxyethyl)-3,4-dihydroquinazolin-4-one
1-(1,3-benzothiazol-2-ylmethyl)-4-(hydroxymethyl)azepan-4-ol
N-[(5-methylfuran-2-yl)methyl]-3-[1-(pyrazine-2-carbonyl)piperidin-3-yl]propanamide
9-[(4-methyl-6-phenylpyrimidin-2-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
6-methyl-2-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-1,3-benzothiazole
6-fluoro-N-methyl-2-(1-methyl-1H-pyrazol-4-yl)-N-(pyridin-3-ylmethyl)quinoline-4-carboxamide
1-[(2-methoxyphenyl)methyl]-4-(1-methyl-1H-imidazol-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4-(4-ethoxy-3-methylphenyl)-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]butanamide
5-ethyl-N4,6-dimethyl-N4-(thiophen-3-ylmethyl)pyrimidine-2,4-diamine
6-(1-cyclopentyl-6-oxopiperidine-3-carbonyl)-1-methyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
2-{1-[(2-chloro-6-fluorophenyl)methyl]-5-(pyrrolidin-3-yl)-1H-1,2,4-triazol-3-yl}acetamide
6-(hydroxymethyl)-N-[3-(4-methylphenyl)phenyl]-1,4-oxazepane-4-carboxamide
6-({cyclopropyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)naphthalen-2-ol
2-({1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperidin-3-yl}methyl)-1H-1,3-benzodiazole
(1R,6S)-9-methyl-3-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-3,9-diazabicyclo[4.2.1]nonane
4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]-1-[3-(1H-pyrazol-1-yl)benzoyl]piperidine
(3aS,6aS)-2-benzyl-5-(4-methoxybenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3aS,6aS)-2-cyclohexyl-5-[(trimethyl-1H-imidazol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{2-[1-(4-oxo-1,4-dihydroquinoline-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide