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1-propanoyl-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
1-(propan-2-yl)-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]-1H-pyrazole-4-carboxamide
6-[(3-methoxyphenyl)methoxy]-1-(2-methylpropyl)-4-(pyrazine-2-carbonyl)-1,4-diazepan-2-one
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-({[5-(4-methylphenyl)-1,2-oxazol-3-yl]methyl}amino)acetamide
1-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-4-(3-methylpyridin-2-yl)piperazine
5-(4,4-difluoropiperidine-1-carbonyl)-2-(pyridin-4-yl)pyrimidine
(1S,5R)-3-(pyrimidin-2-yl)-6-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
2-(3-{[methyl(propan-2-yl)amino]methyl}phenyl)-6-(1-phenoxyethyl)-3,4-dihydropyrimidin-4-one
2-(7-fluoro-2-methyl-1H-indol-3-yl)-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
N-cyclopentyl-2-(dimethylamino)-2-(4-fluorophenyl)-N-propylacetamide
1-[2-(4-fluorophenyl)morpholin-4-yl]-2-(4-phenylpiperidin-1-yl)ethan-1-one
(4aS,7aR)-1-(2-methoxypyridine-4-carbonyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-({methyl[1-(pyridin-3-yl)ethyl]amino}methyl)quinolin-7-ol
3-{5-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1,2,4-oxadiazol-3-yl}-6-methylpyridazine
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-[3-(pyridin-2-yl)propyl]acetamide
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-{3-[methyl(phenyl)amino]propyl}acetamide
1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}-4-(6-methylpyridin-2-yl)piperazine
2-methyl-6-{2-[3-(1H-pyrazol-1-yl)propyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}pyridine
[1-(2-methanesulfonylethyl)-3-(3-methoxypropyl)piperidin-3-yl]methanol
N-methyl-2-(1H-pyrazol-1-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}butanamide
2-[2-(ethoxymethyl)pyrimidin-4-yl]pyridine-4-carboxylic acid
5-[(4-fluorophenyl)methyl]-5-{1-[(2-hydroxyphenyl)methyl]piperidin-4-yl}-3-(2-methoxyethyl)imidazolidine-2,4-dione
4-hydroxy-1-(2-phenoxybenzoyl)piperidine-4-carboxylic acid
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(cyclopent-1-ene-1-carbonyl)piperidine-4-carboxamide
4-[2-({5-methyl-4-[1-(oxolane-3-carbonyl)piperidin-3-yl]pyrimidin-2-yl}sulfanyl)ethyl]morpholine
1-{4-[(cyclopropylamino)methyl]-2-methoxyphenoxy}-3-(morpholin-4-yl)propan-2-ol
3-[({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)amino]-N-(thiophen-2-ylmethyl)propanamide
3-[2-(3,4-difluorophenyl)ethyl]-1-(1,3-thiazole-4-carbonyl)piperidine
(2R,6R)-4-(3-fluorobenzoyl)-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-[(5-ethylpyridin-2-yl)methyl]-4-(piperidine-1-sulfonyl)-1,4-diazepane
4,4,4-trifluoro-1-[3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]butan-1-one
N-{[2-(3-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]-2-(thiophen-3-yl)acetamide
methyl 1-(2-methoxyethyl)-2-oxo-3-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylate
N-(3-hydroxybutyl)-5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,2-oxazole-3-carboxamide
3-chloro-N-{[2-(diethylamino)pyridin-3-yl]methyl}benzamide
N-methyl-3-({4-[methyl(2-phenylethyl)amino]-6-oxo-1,6-dihydropyridazin-1-yl}methyl)-1,2,4-oxadiazole-5-carboxamide
N-(isoquinolin-5-ylmethyl)-N-methyl-2-(1-methyl-3-oxopiperazin-2-yl)acetamide
1-(4-fluorophenyl)-N-[(2-methoxyphenyl)methyl]-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-amine
{[2-({6-[(dimethylamino)methyl]pyrazin-2-yl}oxy)phenyl]methyl}dimethylamine
2-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}benzonitrile
N-[1-(7-fluoro-3-methyl-1-benzofuran-2-carbonyl)pyrrolidin-3-yl]-N-methylacetamide
(3S,4S)-1-[3-(azetidine-1-carbonyl)benzenesulfonyl]-4-(dimethylamino)pyrrolidin-3-ol
(dicyclopropylmethyl)({[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl})methylamine
2-cyclopentyl-9-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(5-ethyl-1,3,4-thiadiazol-2-yl)-N'-[2-(4-ethylphenoxy)ethyl]-N'-methylethanediamide
methyl 6-({4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}amino)-1,2,3,4-tetrahydroquinoline-1-carboxylate
1-[(2E)-but-2-en-1-yl]-4-[1-(methoxymethyl)cyclobutanecarbonyl]-1,4-diazepane-6-carboxylic acid
1-(4-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methoxy}phenyl)ethan-1-one
N,N-dimethyl-3-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propanamide
1-[2-(1-methyl-1H-imidazol-2-yl)benzoyl]-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine