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2-{[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]methyl}-5-methoxypyridin-4-ol
(3S,4R)-3-methoxy-1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidin-4-amine
5-(4-butylpiperazine-1-carbonyl)-2-(phenoxymethyl)pyrimidin-4-ol
2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-{4-[(2-fluorophenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
(3S,5S)-1-(3-cyclopropylpropanoyl)-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
3-[2-(5-chloro-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]-4-[(5-methylfuran-2-yl)methyl]piperazin-2-one
1-{2,7-dimethylimidazo[1,2-a]pyridine-3-carbonyl}-4-methanesulfonyl-1,4-diazepane
3-chloro-N-cyclopentyl-4-{[1-(thian-4-yl)piperidin-4-yl]oxy}benzamide
4-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-1-methyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
4-(1-butyl-1H-imidazol-2-yl)-1-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]piperidine
N4-[(1-cyclopentylpyrrolidin-3-yl)methyl]-5-ethyl-6-methylpyrimidine-2,4-diamine
1-{3-[(benzylamino)methyl]phenoxy}-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
4-[1-(cyclopent-1-ene-1-carbonyl)piperidin-3-yl]-5-methyl-2-[(pyridin-3-ylmethyl)sulfanyl]pyrimidine
1-(4,4-difluoropiperidin-1-yl)-3-(pyridin-4-yl)propan-1-one
N-{1-[1-(oxolane-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
2-(2-chlorophenyl)-1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
N-benzyl-N-(1,1-dioxo-1λ6-thiolan-3-yl)-3-(pyridin-4-yl)propanamide
N-[4-(1H-imidazol-1-yl)phenyl]-6-oxopiperazine-2-carboxamide
2-[2-(4-chlorophenyl)morpholine-4-carbonyl]-1,8-naphthyridine
7-(cyclopropylmethyl)-2-(2-methyl-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
3-(5-{[3-(4-methylphenoxymethyl)piperidin-1-yl]methyl}thiophen-2-yl)prop-2-yn-1-ol
4-(5-ethylpyrimidin-2-yl)-1-methylpiperazine-2-carboxylic acid
1-(4-chloro-2-ethylphenyl)-3-[2-(pyrrolidine-1-sulfonyl)ethyl]urea
N-{2-[4-(hydroxymethyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-5-yl}-3-phenylpropanamide
2-[(1-ethyl-1H-imidazol-2-yl)methyl]-7-(2-methylbenzoyl)-2,7-diazaspiro[4.5]decane
N-[3-(cyclohexyloxy)propyl]-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
2-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazine
N-{1-[3-(methylsulfanyl)propanoyl]azepan-3-yl}oxane-4-carboxamide
1-(8-fluoro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-(2-methoxyethyl)-3-(1,3-thiazol-2-ylmethyl)urea
1-methyl-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(4-methoxy-2-methylphenyl)-3-(1-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}piperidin-3-yl)propanamide
3-({2-[4-(1H-imidazol-1-yl)phenyl]-1H-imidazol-1-yl}methyl)-1-(propan-2-yl)piperidine
4-cyclohexyl-3-(1-methylpiperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-4-(pyrimidin-2-yl)-1,4-diazepane
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(1H-pyrazol-3-ylmethyl)acetamide
4-[(4-methoxyphenyl)methyl]-3-(1-methyl-1H-pyrazol-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
6-(methoxymethyl)-1-methyl-N-(3-phenylpropyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-{2-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-2-oxoethyl}-5,5-dimethylimidazolidine-2,4-dione
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(1r,4r)-4-(3-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}pyrrolidine-1-carbonyl)cyclohexan-1-ol
3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}propanamide
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-[3-(hydroxymethyl)piperidin-1-yl]pyridine-3-carboxamide
(4aS,7aR)-4-butanoyl-6,6-dioxo-N-(thiophen-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-[3-(5-ethyl-4H-1,2,4-triazol-3-yl)phenyl]-4-(furan-2-ylmethyl)piperazine-1-carboxamide
N-{3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-3-oxopropyl}-2-fluorobenzamide
[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]({2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl})amine
1-[1-(3-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]-3,3-dimethylurea
2-(1-methylpyrrolidin-3-yl)-9-(1H-pyrrole-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(3-chloro-4-hydroxyphenyl)-1-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]ethan-1-one
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-decahydro-1,6-naphthyridin-2-one