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3-(5-methyl-1,3,4-thiadiazol-2-yl)-1-(piperidin-4-ylmethyl)urea
3-(5-{[(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)amino]methyl}thiophen-2-yl)prop-2-yn-1-ol
2-{4-[hydroxy(pyridin-2-yl)methyl]piperidine-1-carbonyl}-6-methyl-4H-pyran-4-one
(2R,6R)-11-methoxy-4-(pent-2-yn-1-yl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-(4-{[ethyl({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)amino]methyl}thiophen-2-yl)ethan-1-one
3-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)-1-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}urea
2-(methoxymethyl)-5-{[4-(2-methoxyphenoxy)piperidin-1-yl]methyl}pyrimidine
5-{[3-(3-chlorobenzoyl)piperidin-1-yl]methyl}-2-(2-methylphenyl)pyrimidine
N,N,2-trimethyl-7-[(3-methylthiophen-2-yl)sulfonyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]oxolane-3-carboxamide
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-4-[(2-methylprop-2-en-1-yl)oxy]benzamide
1-{4-[(4-cyclopentyl-1,4-diazepan-1-yl)methyl]-2-methoxyphenoxy}-3-(diethylamino)propan-2-ol
4-(5-{[3-(2-hydroxyethyl)-4-[(6-methylpyridin-2-yl)methyl]piperazin-1-yl]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
methyl 9-(cyclopentyloxy)-3-[4-(4-methoxyphenyl)butan-2-yl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-[1-(5-chloro-4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)-N-(2-phenylethyl)formamido]propanamide
3-chloro-N-cyclopentyl-4-[(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-4-yl)oxy]benzamide
N-({1-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]piperidin-3-yl}methyl)acetamide
4-({[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}methyl)-N-(1,3,4-thiadiazol-2-yl)benzamide
1-[cyclohexyl(methyl)amino]-3-[2-methoxy-4-({[(5-methylfuran-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
5-methyl-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]pyrazine-2-carboxamide
1-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-2-(3,4-difluorophenyl)ethan-1-one
9-[(2-methoxy-4-methylphenyl)methyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(3-fluorophenyl)-4-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-1H-pyrazole
1-[(2-methylphenyl)methyl]-3-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
1-(2-methoxyethyl)-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(naphthalen-2-yl)-1-[2-(pyrrolidine-1-carbonyl)piperazin-1-yl]ethan-1-one
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-[4-(ethylamino)pyrimidin-2-yl]-1-methylpiperazine-2-carboxylic acid
1-{1'-[(2-fluoro-5-methylphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-(1,2-oxazol-3-ylmethyl)pyridin-2-amine
5-chloro-N-[1-(4-methyl-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]thiophene-2-sulfonamide
2-[3-benzyl-1-(4-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-methyl-N-(prop-2-en-1-yl)acetamide
1-[(3-methoxyphenyl)methyl]-N-{[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl}piperidin-3-amine
6-(2-aminoethyl)-N,2-dimethyl-N-(oxan-2-ylmethyl)pyrimidin-4-amine
6-ethyl-2-methyl-N-(1-methyl-6-oxopiperidin-3-yl)quinoline-4-carboxamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[4-(morpholine-4-sulfonyl)piperazin-1-yl]propan-1-one
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}thiophene-3-carboxamide
(4aS,7aR)-N-(4-chlorophenyl)-6,6-dioxo-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-(2,4-dichlorophenoxy)-N-(5-oxo-1-propylpyrrolidin-3-yl)acetamide
1-ethyl-4-{[(1S,5R)-6-(2-methoxyethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-1H-pyrrole-2-carbonitrile
1-cyclopropanecarbonyl-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}piperidine-4-carboxamide
N-[2-(6-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-4-(3-hydroxy-3-methylbutyl)benzamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
3-[(4aR,7aS)-4-(1-benzofuran-5-ylmethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
[(3aS,6aS)-2-[2-(1H-indol-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
4-benzyl-3-{1-[(2S)-2-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenylurea
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyloxane-2-carboxamide
3-(pyrrolidin-1-yl)-1-{[2-(trifluoromethyl)phenyl]methyl}piperidine
2-(2-fluorophenyl)-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}acetamide