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5-ethyl-N,2-dimethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]pyrimidin-4-amine
2-methoxy-2-phenyl-N-{1-[1-(1H-pyrazol-3-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}acetamide
2,3-dimethyl-6-(2,3,6-trimethylquinoline-4-carbonyl)-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-3-[4-(3-methylphenyl)piperazin-1-yl]propan-1-one
8-(butan-2-yl)-1-[2-(4-methoxyphenyl)ethyl]-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1S,4S)-5-[1-(4-chlorophenyl)cyclobutanecarbonyl]-2-[2-(methylsulfanyl)phenyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
methyl 2-[(2,3-dimethylphenyl)sulfamoyl]-6-(1-methylcyclopropanecarbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(3S,4R)-1-{3-[4-(dimethylamino)phenyl]propanoyl}-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
3-{4-methyl-6H,7H,8H-cyclopenta[g]quinolin-2-yl}propanamide
1-{[5-(1-benzofuran-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-3,3-dimethylurea
3-(1-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-1H-1,2,3-triazol-4-yl)phenol
(4aR,7aS)-1-cyclobutanecarbonyl-4-(thiophen-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1-[(2-methoxyphenyl)methyl]-N-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
N-benzyl-5-(2,2-diphenylethyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-(cyclopropylsulfamoyl)-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}benzamide
5-ethyl-4-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}pyrimidin-2-amine
2-{8-chloro-5-methyl-[1,2,4]triazolo[4,3-a]quinolin-1-yl}-1,3-thiazole
2-(3-{[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}phenyl)ethan-1-amine
8-benzoyl-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-{1-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-4-phenyl-1H-imidazol-5-yl}phenol
(3R,4R)-4-(4-methylpiperazin-1-yl)-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-3-ol
3-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(5-fluoro-2-methylphenyl)urea
1-{2-[4-(2-chlorobenzoyl)piperazin-1-yl]ethyl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
3-(pentan-2-yl)-8-(pyridine-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
8-(4-hydroxybenzoyl)-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
4-methyl-2-{1-methyl-3-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenol
2-(dimethylamino)-2-(3-fluorophenyl)-N-[(1-propyl-1H-imidazol-2-yl)methyl]acetamide
N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-2-(1H-pyrazol-1-yl)butanamide
1-methyl-9-(1-propyl-1H-pyrazole-5-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
4-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-2-[(4-methoxyphenyl)methyl]morpholine
5-{[benzyl(methyl)amino]methyl}-N-[1-(pyrazin-2-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
N-{3-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]-3-oxopropyl}methanesulfonamide
N-{2-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]ethyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
(1S,5R)-3-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-methyl-8-(2-methyl-1-benzofuran-7-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
6-[4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
7-chloro-3-{[(3-ethoxypropyl)amino]methyl}-1-(2-phenoxyethyl)-1,2-dihydroquinolin-2-one
1'-(3,5-dimethylphenyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
[2-(4-methoxyphenyl)ethyl][(3-methyl-1H-indol-2-yl)methyl][(1-methylpiperidin-4-yl)methyl]amine
4-benzyl-1-(2-phenylpropanoyl)-1,4-diazepan-5-one
(3S,4R)-1-{2-[(2R,6S)-2,6-dimethylpiperidin-1-yl]acetyl}-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)benzamide
6-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]quinoxaline
1-(3,5-dimethyl-1-benzofuran-2-carbonyl)-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
4-(4-fluorophenyl)-1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-ol
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)pyridine-4-carboxamide
(4aS,8aR)-6-[2-(methylsulfanyl)acetyl]-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
1-(2-hydroxyethyl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-1,3-benzodiazole-5-carboxamide
1-[2-(1H-imidazol-5-yl)ethyl]-3-(phenoxymethyl)-5-[5-(propan-2-yl)-1,2-oxazol-3-yl]-1H-1,2,4-triazole
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-methyl-2-(2-methylphenoxy)butan-1-one