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5-(8-methylquinolin-5-yl)pyridin-2-amine
[5-(1-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-1H-1,2,3-triazol-4-yl)furan-2-yl]methanol
{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}(methyl)[3-(1-methyl-1H-imidazol-2-yl)propyl]amine
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-fluoro-N-methyl-2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-4-amine
1-{[1-(2,5-dimethoxybenzoyl)piperidin-3-yl]methyl}-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
1-[3-(furan-2-yl)propanoyl]-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)(methyl)[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amine
1-{[3-(methylsulfanyl)phenyl]methyl}-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
N-[1-(2,5-dimethylphenyl)ethyl]-2-(pyridin-3-yl)acetamide
5-cyclopropanecarbonyl-1'-[(5-propylfuran-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
9-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2,6-dimethyl-4-[({[4-(methylcarbamoyl)phenyl]methyl}amino)methyl]phenyl acetate
2-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]-N-(1-methyl-1H-pyrazol-3-yl)acetamide
2-cyclopentyl-9-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
(2,1,3-benzoxadiazol-5-ylmethyl)({1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl})amine
3-[(2-fluorophenyl)methyl]-1-{thieno[2,3-d]pyrimidin-4-yl}piperidine-3-carboxylic acid
N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]-6-(piperidin-3-yl)pyrimidin-4-amine
1-[5-(methoxymethyl)thiophene-2-carbonyl]-4-(pyrrolidine-1-carbonyl)piperidine
{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(pyridin-3-yl)ethyl]amine
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
(2R,6S)-4-{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}-2,6-dimethylmorpholine
3-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-4-methylbenzene-1-sulfonamide
2-(3-methoxypropyl)-9-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
(3aR,6aR)-2-methanesulfonyl-5-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-({3-[(2-methoxyethyl)(thiophen-3-ylmethyl)carbamoyl]phenyl}amino)acetic acid
N-{2-[4-(hydroxymethyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-5-yl}cyclopentanecarboxamide
2-ethoxy-6-({3-[4-methyl-5-(prop-2-en-1-ylsulfanyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)phenol
N-(3-{3,9-diazaspiro[5.6]dodecane-9-sulfonyl}phenyl)acetamide
N-cyclopropyl-N-{[2-(2,5-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}oxolane-2-carboxamide
3-{2-[3-methyl-1-(3-methylphenyl)-1H-1,2,4-triazol-5-yl]ethyl}-3,4-dihydroquinazolin-4-one
(2R,3R,6R)-3-(4-methoxyphenyl)-5-{pyrazolo[1,5-a]pyridine-3-carbonyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
2-methyl-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-4-(piperidin-3-yl)benzamide
3-[(4-{furo[3,2-c]pyridin-4-yl}piperazin-1-yl)methyl]-1-methyl-1,2-dihydroquinolin-2-one
1-(2-methoxyethyl)-3-(2-methoxyphenyl)-3-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]pyrrolidine-2,5-dione
2-(1-{2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carbonyl}piperidin-2-yl)ethan-1-ol
(3R,5S)-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-N-[3-(dimethylamino)propyl]-1-[(4-hydroxyphenyl)methyl]piperidine-3-carboxamide
methyl 4-[(1-hydroxybutan-2-yl)(pyridin-2-ylmethyl)carbamoyl]benzoate
(1R,5S,8S)-3-[(4-butoxyphenyl)methyl]-3-azabicyclo[3.2.1]octan-8-ol
(1S,5R)-6-benzyl-3-[(6-methylpyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-[(3,5-dimethoxyphenyl)methyl]-4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
2-{2-[3-(5-chloro-2-hydroxyphenyl)-1H-pyrazol-1-yl]phenyl}acetic acid
2-(4-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carbonyl}piperidin-1-yl)acetamide
7-(3,6-dimethylpyrazin-2-yl)-4-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-{1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1H-pyrazole
2-[4-(6-amino-2-{[(4-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)-1-methylpiperazin-2-yl]ethan-1-ol
N-(2-hydroxyethyl)-8-methyl-N-(1,3-thiazol-2-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
2-{3,5-dimethyl-4-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]-1H-pyrazol-1-yl}ethan-1-ol
2-[({[4-(hydroxymethyl)oxan-4-yl]methyl}(methyl)amino)methyl]-6,8-dimethylquinolin-4-ol