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N-[3-(oxolan-3-yl)propyl]-4-sulfamoylbenzamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
3-{[3-cyclopropyl-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
2-methyl-4-{5-[(oxan-2-ylmethoxy)methyl]-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl}pyridine
4-ethyl-3-(1-{2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]acetyl}piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
8-[(2,2-difluoro-2H-1,3-benzodioxol-5-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-(2H-1,3-benzodioxol-5-yl)-1-[9-methoxy-7-(quinolin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
1-[9-(2,3-dihydro-1H-inden-1-yloxy)-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(dimethyl-1,2-oxazol-4-yl)ethan-1-one
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
5-(4-cyclopentyl-1,4-diazepane-1-carbonyl)-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
3-(2-{2-[2-(1H-imidazol-1-yl)ethyl]piperidin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
N-tert-butyl-6-[(oxolan-2-ylmethyl)sulfamoyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
(1S,5R)-N-(2-phenylethyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
1-{2-[3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]ethyl}azepan-2-one
3-[(4aR,7aS)-4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
(4aR,7aS)-1-(2-methoxyethyl)-4-(3-phenylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[4-methyl-5-({1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidin-4-yl}methyl)-4H-1,2,4-triazol-3-yl]methanol
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(2-methyl-1H-pyrrole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
4-[(2S)-2-hydroxypropanoyl]-1-(2-phenylphenyl)piperazin-2-one
N-[(5-chlorothiophen-2-yl)methyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2,5-dimethyl-3-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]pyrazine
(3S,4S)-1-[(4-fluoro-3-methylphenyl)methyl]-4-(piperidin-1-yl)pyrrolidin-3-ol
N-(2,3-dihydro-1H-inden-2-yl)-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
3-[(3R,4S)-4-(dimethylamino)-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidin-3-yl]propanoic acid
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-(2,2,2-trifluoroethyl)piperidine-3-carboxamide
4-(2,3-dihydro-1-benzofuran-7-yl)-5-phenyl-1H-pyrazol-3-amine
8-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-ylmethyl]-5-(hydroxymethyl)-2-methylpyridin-3-ol
{1-[(2-ethoxyphenyl)methyl]-4-(2-phenoxyethyl)piperidin-4-yl}methanol
4-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholine
N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
(4aR,7aS)-1-cyclobutanecarbonyl-4-(1H-pyrazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{1-[4-(pyridin-2-yl)pyrimidin-2-yl]piperidin-4-yl}-1,3-oxazolidin-2-one
1-(2-methoxyethyl)-3-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-1-[(2-methylphenyl)methyl]urea
2-methyl-4-[4-({3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenyl]but-3-yn-2-ol
N-[3-(4-fluorophenyl)-3-(furan-2-yl)propyl]-3-(pyridin-4-yl)propanamide
1-cyclohexyl-4-[6-(pyrrolidin-1-yl)pyridine-3-carbonyl]-1,4-diazepane
1-[4-({3-[3-(methoxymethyl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)phenyl]ethan-1-one
(3S,4R)-4-(3-methoxyphenyl)-1-(2-methyl-1,3-thiazole-4-carbonyl)pyrrolidine-3-carboxylic acid
1-[(3-fluorophenyl)methyl]-4-(1H-indol-4-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4-benzyl-1-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(4-methyl-1,3-thiazol-5-yl)-N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]propanamide
N-[(3S,4R)-4-(4-methylphenyl)-1-[(trimethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl]cyclopropanecarboxamide
1-(2-hydroxyethyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]azepane-2-carboxamide
3-({2-[2-(furan-2-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}methyl)-1,5-dimethyl-1H-indazole
N-[1-(2-chlorophenyl)ethyl]-1-(4-methylquinazolin-2-yl)piperidine-4-carboxamide
1-methyl-N-[1-methyl-4-(pyridin-3-yloxy)-1H-indazol-3-yl]-2-oxoimidazolidine-4-carboxamide
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N,4,6-trimethylpyrimidin-2-amine