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1-phenyl-2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethan-1-ol
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-2-ethyl-N-methylpyrimidine-5-carboxamide
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-3-(3-hydroxy-3-methylbutyl)benzamide
N-[(5-ethylpyridin-2-yl)methyl]-N,5,7-trimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
2-(hydroxymethyl)-N-[(2S)-1-methoxy-3-phenylpropan-2-yl]-1H-1,3-benzodiazole-5-carboxamide
3-(1H-1,3-benzodiazol-1-yl)-1-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}propan-1-one
7-(2,2-dimethylpropyl)-2-[(6-methylpyridin-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
3-[(2,3-dihydro-1-benzofuran-2-ylmethyl)(methyl)amino]-N-(2-methylphenyl)propanamide
(2-{2,8-dimethyl-[1,2,4]triazolo[1,5-a]pyridin-6-yl}phenyl)methanol
dimethyl(2-{2-[1-(1-methyl-1H-indole-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
N3-(1-benzylpyrrolidin-3-yl)-N5-butyl-1-cyclohexyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-4-(1-phenyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-(2-chlorophenyl)-3-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}propanamide
1,2-dimethyl-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)-1H-imidazole-4-sulfonamide
N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[3-(1H-imidazol-1-yl)propyl]-9-(oxane-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
4-(2-methylphenoxy)-1-[1-(piperidin-4-yl)pyrrolidine-2-carbonyl]piperidine
(1S,5R)-3-(2-methyl-1,3-benzothiazole-5-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
5-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-amine
2-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carboxamide
9-[1-(4-chlorophenyl)cyclopropanecarbonyl]-1,4,9-triazaspiro[5.5]undecan-5-one
N-(2-methyl-1,3-benzothiazol-5-yl)-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
6-(4-fluorophenyl)-N-(2-hydroxypropyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
(2S,4R)-4-amino-1-{[2,5-dimethyl-1-(pyridin-3-yl)-1H-pyrrol-3-yl]methyl}-N-methylpyrrolidine-2-carboxamide
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
7-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1,3-diazepane-2,4-dione
5-[(4-hydroxypiperidin-1-yl)methyl]-N,N-bis(2-methylpropyl)-1,2-oxazole-3-carboxamide
1-[4-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl]-3-[1-(pyrazin-2-yl)piperidin-3-yl]urea
(3S,4R)-4-methyl-1-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]piperidine-3,4-diol
N-methyl-4-[3-(4-methylphenoxymethyl)piperidine-1-carbonyl]-1,3-thiazol-2-amine
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1-benzofuran-5-carboxamide
2-methyl-5-{4-[1-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}-1,4-dihydropyridin-4-one
3-{imidazo[1,2-a]pyridin-2-yl}-1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
N-[2-(2-chlorophenyl)-2-(dimethylamino)ethyl]-1-cyclohexyl-1H-1,2,3-triazole-4-carboxamide
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[(1R,5S,6R)-6-[(dimethylamino)methyl]-3-azabicyclo[3.1.0]hexan-3-yl]ethan-1-one
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-3-methyl-1H-pyrazole-4-carboxamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]acetamide
1-methyl-N-{[1-(4-methylpiperazin-1-yl)cyclopentyl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[3-(1H-imidazol-1-yl)propyl]-3-{[(3-methoxyphenyl)methyl]amino}-5-(pyrrolidine-1-sulfonyl)benzamide
N-ethyl-5,7-dimethyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
[2-(diethylamino)ethyl]({[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl})methylamine
N-cyclopropyl-N-{[3-(2-methylpropoxy)phenyl]methyl}-4-(trifluoromethyl)benzamide
(3S,4S)-4-methoxy-N-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-(propan-2-yl)pyrrolidin-3-amine
2-amino-4-[5-(hydroxymethyl)furan-2-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-[2-(1H-1,2,4-triazol-3-yl)benzoyl]-1,4-diazepane
2-{4-[1-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}-N,N-dimethylacetamide
2-[(2-methylprop-2-en-1-yl)oxy]-N-[2-(pyridin-3-yloxy)propyl]benzamide