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methyl 3-[ethyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})carbamoyl]benzoate
N-cyclobutyl-2-[4-(2-methoxypyridine-4-carbonyl)morpholin-3-yl]acetamide
2-butyl-8-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
ethyl 1-[4-(1H-imidazol-1-yl)benzoyl]-3-(2-phenylethyl)piperidine-3-carboxylate
4-[2-(1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-2-yl)ethyl]morpholine
N-[(3-chloro-2-fluorophenyl)methyl]-2-(propan-2-yloxy)propanamide
N-methyl-N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-6-(piperidin-3-yl)pyrimidin-4-amine
2-(cyclopropylmethyl)-8-(2-hydroxyacetyl)-2,8-diazaspiro[5.5]undecan-3-one
4-ethyl-3-[1-(3-{imidazo[1,2-a]pyridin-2-yl}propanoyl)piperidin-4-yl]-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-2,1,3-benzoxadiazole
[(3S,4S)-1-{[5-(4-chlorophenyl)furan-2-yl]methyl}-4-(hydroxymethyl)pyrrolidin-3-yl]methanol
3-(2H-1,3-benzodioxol-5-yl)-5-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-cyclopropyl-5-oxo-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]pyrrolidine-3-carboxamide
2-{9-[(2R)-3-hydroxy-2-methylpropyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
2-{2-[({[1-(2-methoxyethyl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl)amino)methyl]phenoxy}ethan-1-ol
(1R,3S)-7-(2-amino-6-methoxypyrimidin-4-yl)-3-[2-(dimethylamino)ethoxy]-7-azaspiro[3.5]nonan-1-ol
(2S,4R)-4-hydroxy-N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)pyrrolidine-2-carboxamide
5-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-2-methyl-1H-1,3-benzodiazole
methyl 4-({3-[5-(benzylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)benzoate
5-phenyl-3-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]-1,2,4-oxadiazole
6-cyano-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]pyridine-3-carboxamide
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(3-fluorophenyl)methyl]-4-(1-methanesulfonylpyrrolidine-2-carbonyl)piperazine
3-({1-[(5-ethylpyridin-2-yl)methyl]pyrrolidin-3-yl}methyl)-1-phenylurea
1-(pyridin-2-yl)-N-(1,3-thiazol-2-ylmethyl)piperidine-3-carboxamide
1-[(2-fluorophenyl)methyl]-N-[2-methyl-2-(morpholin-4-ylmethyl)propyl]piperidin-3-amine
N-benzyl-4-{[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carboxamide
4-oxo-5-phenoxy-1-{3-[(pyridin-3-yl)amino]propyl}-1,4-dihydropyridine-3-carboxylic acid
4-({2-[1-(4-methoxyphenyl)-1H-imidazol-2-yl]-1H-imidazol-1-yl}methyl)-3,5-dimethyl-1,2-oxazole
1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-3-(4-methylphenoxymethyl)piperidine
4-[3-(1H-indol-4-yl)-1,2,4-oxadiazol-5-yl]-N,N-dimethylpiperidine-1-carboxamide
8-methyl-2-(1-methyl-1H-pyrazol-4-yl)-4-(thiomorpholine-4-carbonyl)quinoline
N-(1-benzylpyrrolidin-3-yl)-3-{1-[2-(2-fluorophenyl)acetyl]piperidin-4-yl}propanamide
2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]-N-butyl-N-methylacetamide
(3R,5S)-N-[2-(morpholin-4-yl)ethyl]-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-N-[2-(diethylamino)ethyl]-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-{3-[(5-methylpyridin-2-yl)amino]propyl}acetamide
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
[(2S)-1-[2-(2-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]pyrrolidin-2-yl]methanol
9-(1-methyl-1H-imidazole-2-carbonyl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-(furan-2-yl)-1-[2-(naphthalen-1-ylmethyl)morpholin-4-yl]propan-1-one
1-[(2-fluorophenyl)methyl]-N-methyl-N-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-3-amine
(1S,6R)-3-[2-(2,3-dihydro-1H-isoindol-2-yl)-2-oxoethyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
(4aS,7aR)-1-{2-[ethyl(methyl)amino]acetyl}-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[3-(furan-2-amido)-4-methoxyphenyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
(1S,6R)-9-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
2-[2-oxo-2-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)ethyl]-1,2-dihydrophthalazin-1-one
2-(2-methoxy-4-methylphenoxymethyl)-N-methyl-N-propyl-1,3-oxazole-4-carboxamide
4-[(4-cyclopentylpyrimidin-2-yl)amino]-1-ethylpyrrolidin-2-one
(3aS,6aR)-5-(1,4-dithiepan-6-yl)-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one