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3-(2H-1,3-benzodioxol-5-yl)-1-{1-methyl-octahydropyrrolo[1,2-a]piperazin-2-yl}propan-1-one
3-[(3R,4S)-4-(morpholin-4-yl)-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl]propanoic acid
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(4-hydroxyphenyl)ethan-1-one
1-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-3-(6-methoxynaphthalene-2-carbonyl)piperidine
N-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-(1H-1,3-benzodiazol-2-yl)-2-{methyl[2-(oxan-2-yl)ethyl]amino}acetamide
ethyl 1-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
(1R,3S)-7-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-7-azaspiro[3.5]nonane-1,3-diol
4-benzyl-1-(cyclobutylmethyl)-3-ethyl-1,4-diazepan-5-one
6-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2,3,4-tetrahydroquinoline
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-[4-(hydroxymethyl)phenyl]ethan-1-one
(2S,4S)-1-[(4-chlorophenyl)methyl]-4-[(naphthalen-2-ylmethyl)amino]-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
7-(2-methoxyethyl)-N-[(4-methoxyphenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
N-[(3R,4S)-1-(oxane-4-carbonyl)-4-phenylpyrrolidin-3-yl]methanesulfonamide
benzyl 3-({[(1,3-dimethyl-1H-pyrazol-5-yl)carbamoyl]amino}methyl)piperidine-1-carboxylate
4-(methoxymethyl)-6-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyrimidine
5-(3-fluorophenoxymethyl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1H-pyrazole-3-carboxamide
5-[3-({2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)propyl]-1,3,4-thiadiazol-2-amine
N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]naphthalene-1-carboxamide
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-2-(2-oxoazepan-1-yl)acetamide
2-amino-4-ethyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-1,3-thiazole-5-carboxamide
3-cyclopentyl-1-[(4-methylphenyl)methyl]-5-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-1,2,4-triazole
1-[(2-chlorophenyl)methyl]-N-{[3-(trifluoromethoxy)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-hydroxy-2,2-dimethylpropyl)acetamide
4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-[1-(1,3-thiazol-2-yl)ethyl]butanamide
[1-(cyclohexylmethyl)-5-[2-(pyrazin-2-yl)ethyl]-1H-1,2,4-triazol-3-yl](phenyl)methanol
2-amino-6-{4-[(5-chloro-2,3-dimethoxyphenyl)methyl]piperazin-1-yl}pyrimidin-4-ol
3-{[(2-cyclopropylphenyl)carbamoyl](2-phenylethyl)amino}propanamide
2-(propan-2-yloxy)-1-[4-(pyridin-4-yl)piperazin-1-yl]propan-1-one
1-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}-2-(1H-pyrazol-1-yl)butan-1-one
1-methyl-3-(2-{3-methyl-1-[(4-methylphenyl)methyl]-1H-1,2,4-triazol-5-yl}ethyl)piperidine
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
N-[1-(methoxymethyl)cyclopentyl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
2-{4-[3-cyclopropyl-1-(3,4-dimethylphenyl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}acetamide
5-[2-(furan-2-yl)pyrrolidine-1-carbonyl]-1H-imidazole-4-carboxylic acid
3-ethyl-1-[3-fluoro-5-(trifluoromethyl)phenyl]-3-(4-hydroxybutyl)urea
(3aR,6aR)-2-[(3-chloropyridin-4-yl)methyl]-5-cyclopentyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(2H-1,3-benzodioxol-5-yl)-1-{2-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-3-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
[(1-ethyl-1H-pyrazol-4-yl)methyl]({[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})methylamine
4-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-N-methylpyridin-2-amine
benzyl({[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})ethylamine
1-[(4-fluorophenyl)methyl]-4-[1-(methoxymethyl)cyclobutanecarbonyl]-2-(propan-2-yl)-1,4-diazepane
[2H-1,3-benzodioxol-5-yl(3-cyclopropyl-1H-1,2,4-triazol-5-yl)methyl]dimethylamine
2-[1-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-2-methylbutyl]-2,3-dihydro-1H-isoindol-1-one
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-({[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]amino}methyl)piperidin-2-one
(4aR,7aS)-1-ethyl-4-(2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}acetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-sulfonyl}-N-(pyrrolidin-3-yl)benzamide
2,5-difluoro-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)benzamide
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-2-(cyclohex-1-en-1-yl)acetamide
5-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-2-(pyridin-3-yl)pyrimidine