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4-{6-cyclopropyl-3-methyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-2-(4-methylpentyl)morpholine
6-(4-tert-butylbenzoyl)-1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octane
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-5-methoxy-1-methyl-1H-indole-2-carboxamide
2-cyclopropyl-4-hydroxy-N-[4-(4-methoxyphenyl)butan-2-yl]pyrimidine-5-carboxamide
(4aS,7aR)-1-[(1-phenyl-1H-pyrazol-4-yl)methyl]-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(propan-2-yl)-4-[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]-1,3-thiazole
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(4-{2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridine-5-carbonyl}piperidin-1-yl)acetamide
6-{[1-(2-fluorophenyl)propan-2-yl]amino}-2-methylheptan-2-ol
3-methoxy-1-[(2,4,5-trifluorophenyl)methyl]-1,2-dihydropyridin-2-one
3-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-4-yl}-N-(2,4-dimethoxyphenyl)propanamide
5-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}pyrazin-2-ol
3-phenyl-5-(thiomorpholine-4-sulfonyl)benzoic acid
N5-cycloheptyl-N1,3-dicyclopropyl-4-oxo-N3-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
1-(2H-1,3-benzodioxol-5-yl)-N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}piperidin-4-amine
N-[3-(1H-pyrazol-5-yl)phenyl]azocane-1-carboxamide
2-(4-propanoylphenoxy)-N-[2-(1H-1,2,4-triazol-1-yl)propyl]acetamide
N-(4-hydroxybutyl)-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
N-(adamantan-1-yl)-5-ethyl-1,3,4-oxadiazol-2-amine
5-methyl-1'-{thieno[3,2-d]pyrimidin-4-yl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[1-(4-methyl-1,3-thiazole-5-carbonyl)-1,2,3,6-tetrahydropyridin-4-yl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1H-pyrazole-3-carboxamide
2-(dimethylamino)-1-[4-(3-hydroxypropyl)piperazin-1-yl]-2-(3-methylphenyl)ethan-1-one
N4-methyl-N4-[(4-methyl-1H-imidazol-2-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-3-phenyl-1H-pyrazole-4-carboxamide
methyl({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
3-[2-(cyclohexylmethyl)morpholine-4-carbonyl]-N-methylpyridin-2-amine
2-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}-6-methoxyphenol
1-(2-{[(3-ethoxy-4-methoxyphenyl)methyl]amino}ethyl)-N-(pyridin-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
(1R,2R,6S,7S)-4-(2-benzyl-1,3-thiazole-4-carbonyl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
3-({1-[4-(furan-2-yl)phenyl]piperidin-4-yl}amino)-2,3-dihydro-1λ6-thiophene-1,1-dione
(3S,4S)-4-(naphthalen-2-yl)-1-(pyrrolidine-1-sulfonyl)piperidin-3-ol
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(pyridin-3-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(2S)-1-(7-fluoro-3-methyl-1-benzofuran-2-carbonyl)pyrrolidine-2-carboxamide
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-3,5-dimethylfuran-2-carboxamide
2-[4-(piperidin-1-ylmethyl)phenyl]-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
[3-(1H-imidazol-1-yl)propyl](3-methylbut-2-en-1-yl)(pyridin-4-ylmethyl)amine
2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)acetamide
1-cyclopentyl-4-[2-methoxy-4-(4-methoxypiperidine-1-carbonyl)phenoxy]piperidine
N-(butan-2-yl)-N-ethyl-1H-1,2,3-benzotriazole-5-carboxamide
dimethyl({[4-methyl-5-(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl})amine
(benzylsulfamoyl)[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]amine
{5-[(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)methyl]furan-2-yl}methanol
2-(2,4-dioxoimidazolidin-1-yl)-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}acetamide
2-{[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-4H-pyrido[1,2-a]pyrimidin-4-one
6-(1-phenoxyethyl)-2-[4-(pyrrolidin-1-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
3-[(3S,7S,8aS)-3-[(2S)-butan-2-yl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(5-fluoro-2-methylphenyl)urea
4-(3-fluoropyridine-4-carbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(3-methyl-3-phenylpiperidin-1-yl)-3-(pyrrolidine-1-carbonyl)pyridine
1-{3-[4-(2-methoxybenzoyl)piperazin-1-yl]-3-oxopropyl}pyrrolidin-2-one