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5-chloro-6-[3-(1-methyl-1H-pyrazol-5-yl)phenyl]pyridine-3-carboxylic acid
4-(propan-2-yloxy)-6-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]pyrimidin-2-amine
1-[2-(1H-imidazol-1-yl)ethyl]-2-(3-methyl-1-benzofuran-2-yl)-1H-imidazole
5-{[4-(2-methoxyethyl)piperazin-1-yl]methyl}-2-(naphthalen-1-yl)pyrimidine
6-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)pyridine-2-carbonitrile
5-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-2-methylpyridine
3-({cyclopropyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-6-methoxy-1,2-dihydroquinolin-2-one
N-[(3S,4R)-1-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-4-(1H-pyrazol-3-yl)benzamide
1-(morpholin-4-yl)-3-(1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}piperidin-4-yl)propan-1-one
2-[(1S,4S)-5-benzyl-2,5-diazabicyclo[2.2.1]heptane-2-carbonyl]-3,5-dimethyl-1H-indole
N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)-1H-pyrrole-2-carboxamide
2-[5-cyclopropyl-4-(4-propylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]-4-(thiophen-2-yl)pyrimidine
1-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
3-acetamido-N-methyl-N-[3-(1H-pyrazol-1-yl)propyl]benzamide
N-(2,2-dimethyloxan-4-yl)-5-methyl-4-[(pyridin-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
N-(1,3-dihydro-2-benzofuran-5-yl)-2-(furan-2-yl)pyrrolidine-1-carboxamide
(2S)-N-[3-(1H-pyrazol-1-yl)phenyl]-1-[2-(4H-1,2,4-triazol-4-yl)ethyl]pyrrolidine-2-carboxamide
2-[methyl(2-phenylethyl)amino]-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
6-methoxy-N,3-dimethyl-N-(1,3-thiazol-2-ylmethyl)-1-benzofuran-2-carboxamide
2-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrazine
6-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]pyridine-2-carboxylic acid
2-(2-chlorophenyl)-N-(2-methoxyethyl)-N,3-dimethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-3,5-dimethyl-1,2-oxazole-4-carboxamide
methyl 3-methyl-4-({methyl[(1-methyl-1H-imidazol-2-yl)methyl]carbamoyl}amino)benzoate
1'-{2,8-diazaspiro[4.5]decane-3-carbonyl}spiro[indene-1,4'-piperidine]
1-[3-(1H-1,3-benzodiazol-2-yl)azetidin-1-yl]-4-(4-fluorophenyl)butane-1,4-dione
3-{[4-(3-chlorophenyl)-5-({methyl[(3-methylquinoxalin-2-yl)methyl]amino}methyl)-4H-1,2,4-triazol-3-yl]sulfanyl}propan-1-ol
5-[(4-methoxyphenyl)methyl]-5-{3-oxo-3-[3-(2-phenylacetyl)piperidin-1-yl]propyl}pyrrolidin-2-one
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}[(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
N,N-dimethyl-5-(trimethylpyrimidin-4-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(thiophen-3-ylmethyl)pyrrolidin-3-yl]-2,4-dimethyl-1,3-oxazole-5-carboxamide
3-methyl-7-(1H-pyrrole-2-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-[2-(2-chlorophenyl)-2-hydroxyethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
(4aS,8aR)-6-(1H-imidazol-2-ylmethyl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
2-cyclopentyl-1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]ethan-1-one
4-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)butan-1-ol
3-(3,3-diphenylpiperidin-1-yl)propan-1-ol
2-[2-(2-fluorophenyl)ethyl]-4-[4-(furan-2-ylmethyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
6-(piperidin-4-yl)-N-(prop-2-en-1-yl)-N-(pyridin-3-ylmethyl)pyrimidin-4-amine
{4-methyl-5-[(1-{[5-(oxan-2-yl)furan-2-yl]methyl}piperidin-4-yl)methyl]-4H-1,2,4-triazol-3-yl}methanol
(1R,2R)-N-[(4-chlorophenyl)methyl]-N-ethyl-2-phenylcyclopropane-1-carboxamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-(piperidin-1-yl)pyridine-3-carboxamide
N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]acetamide
4-(azocane-1-carbonyl)-1,2-dihydroisoquinolin-1-one
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-(propan-2-yl)pyrimidin-4-amine
N-{1-[(4-chlorophenyl)methyl]piperidin-4-yl}-2,5,6-trimethylpyrimidin-4-amine
2-{4-[(4-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}thiophen-3-amine
4-ethyl-1-methyl-3-(1-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]acetyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(1-ethylpiperidine-2-carbonyl)-1-(2-methoxyphenyl)-2,2-dimethylpiperazine