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2-[(2-{[(1S)-1-carbamoyl-3-methylbutyl]carbamoyl}phenyl)amino]acetic acid
3-(2-methoxyphenyl)-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
N-(3-{[(2-fluorophenyl)methyl]sulfanyl}propyl)-5-methoxy-4-oxo-1,4-dihydropyridine-2-carboxamide
N-(butan-2-yl)-3,5-difluoro-N-(pyridin-4-ylmethyl)pyridine-2-carboxamide
N-[(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-3-yl)methyl]cyclobutanecarboxamide
2-{1'-[(6-methylpyridin-2-yl)methyl]-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl}acetamide
[(2-chloropyridin-3-yl)methyl][(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]methylamine
7-(cyclopropylmethyl)-2-[(5-ethylfuran-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
[(3R,4R)-1-(4,6-dimethylquinolin-2-yl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
3-(1-{[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]methyl}piperidin-4-yl)-N-(2-methoxyethyl)propanamide
1-methyl-8-(2-methylbenzoyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
N-[1-(azepan-1-yl)-2-methylpropan-2-yl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
3-(3-fluorophenyl)-N-(2-hydroxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
1-{2-[4-(pyridin-3-yloxy)piperidin-1-yl]ethyl}-1H-indazole
4-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-{4-[benzyl(methyl)amino]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl}benzamide
1-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)but-3-en-1-one
1-(2,3-dihydro-1H-inden-2-yl)-4-(dimethyl-1,3-oxazole-4-carbonyl)-1,4-diazepane
5-[(4-hydroxypiperidin-1-yl)methyl]-N-(3-phenylpropyl)-1,2-oxazole-3-carboxamide
N-(1-benzylpyrrolidin-3-yl)-3-{1-[(2-fluorophenyl)methyl]piperidin-4-yl}propanamide
N-[(3S,4R)-1-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
2-{3-[3-(3-chloropyridin-2-yl)phenyl]-1H-pyrazol-1-yl}acetamide
2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]-2-[3-(trifluoromethyl)phenyl]acetic acid
4-methoxy-N-(4-{4-[methyl(1,2-oxazol-3-ylmethyl)amino]piperidin-1-yl}phenyl)benzamide
4-chloro-N,N-dimethyl-5-({3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)-1,3-thiazol-2-amine
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-2-[(2-fluorophenyl)methyl]-1,3-benzoxazole-6-carboxamide
8-chloro-2-{[2-(pyridin-3-yl)morpholin-4-yl]methyl}quinoline
N,1-dimethyl-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-(1-methyl-4-phenyl-1H-pyrazol-5-yl)acetamide
2-[3-(methoxymethyl)piperidin-1-yl]-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridine
6-methoxy-N4-methyl-N4-[2-(morpholin-4-yl)ethyl]pyrimidine-2,4-diamine
N-({5-[(6-methoxynaphthalen-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
4-[3-({1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}oxy)benzoyl]morpholine
5-({[2-(dimethylamino)ethyl](thiophen-3-ylmethyl)amino}methyl)-2-hydroxybenzoic acid
5-acetyl-N-(2H-1,3-benzodioxol-5-ylmethyl)-N-(propan-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-3-(pyridin-2-yl)propanamide
1-[4-(1-benzyl-1H-1,2,4-triazol-5-yl)phenyl]pyrrolidin-2-one
N-(2-methyl-5-propanamidophenyl)-4-(pyrimidin-4-yl)piperidine-1-carboxamide
6-[(diethylamino)methyl]-N-(1H-indazol-6-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})amine
3-{[(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-4-yl)oxy]methyl}pyridine
6-{2-cyclopropyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-2,4-dimethylpyridine-3-carbonitrile
2,3-difluoro-6-methoxy-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]benzamide
N-(1-{7-[(5-methylthiophen-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxane-4-carboxamide
[(2S,4R,5R)-5-(4-chlorophenyl)-1-ethyl-2-methyl-4-({[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]amino}methyl)pyrrolidin-2-yl]methanol
(2S)-2-amino-3-phenyl-1-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propan-1-one
2,6-diamino-4-(5-chlorothiophen-2-yl)-5,6,7,8-tetrahydroquinoline-3-carbonitrile
(3S,4S)-4-(4-fluorophenyl)-1-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}piperidin-3-ol
N,N-dimethyl-5-({4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}methyl)pyrimidin-2-amine