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1-[4-(4-methoxybenzoyl)piperazin-1-yl]-3-(2-methyl-1H-imidazol-1-yl)butan-1-one
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-ethyl-1H-imidazol-2-yl)methyl]acetamide
1-(2-{[2-(cyclohex-1-en-1-yl)ethyl]amino}pyrimidin-4-yl)pyrrolidin-3-ol
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]-2,3-dihydro-1H-indene-2-carboxamide
4-(4-aminopyrimidin-2-yl)-9-(2-methoxyethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-hydroxy-N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
3-methyl-5-(4-{2-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}phenyl)-4H-1,2,4-triazole
1-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-yl}pent-4-en-1-one
1-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-(1H-imidazol-1-ylmethyl)piperidine
2-{5-[2-(benzenesulfonyl)ethyl]-3-cyclopentyl-1H-1,2,4-triazol-1-yl}acetic acid
N-[(3R,4R)-1-(4-cyclobutyl-6-methylpyrimidin-2-yl)-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
(3S,4S)-1-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetyl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
(3S,4S)-1-(furan-3-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
2-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]pyridine-3-carboxylic acid
1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-4-(pyrrolidin-1-yl)pentan-1-one
6-{1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]piperidin-3-yl}-2-methylpyrimidin-4-ol
1-{2-[3-(2-chlorophenoxy)azetidin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
4-(piperidin-1-ylmethyl)-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]benzamide
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]morpholine-2-carboxamide
1,3,6-trimethyl-N-[2-methyl-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[1-(cyclohexylmethyl)piperidin-3-yl]-6-methylpyridazin-3-amine
3-methyl-6-[3-(2-methylphenyl)piperidin-1-yl]pyridazine
2-amino-4-(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)-6-(4-methyl-1,3-thiazol-5-yl)pyridine-3-carbonitrile
2-butyl-8-[(3-methylquinoxalin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N,2-dimethyl-1H-1,3-benzodiazole-5-carboxamide
N2-benzyl-6-(pyridin-3-yl)-1,3,5-triazine-2,4-diamine
(4-{[1-(2,6-dimethoxybenzoyl)pyrrolidin-3-yl]methyl}phenyl)methanol
5-[4-(5-chloro-2-methylphenyl)piperazin-1-yl]-1-[(2,4-difluorophenyl)methyl]azepan-2-one
(1S,5R)-3-[2-hydroxy-6-(trifluoromethyl)pyridine-3-carbonyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
7-(cyclobutylmethyl)-2-[2-(pyrazin-2-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
6-[3-cyclopropyl-1-(3-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]-3,5-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
1-(4-methyl-1H-imidazole-5-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
1-benzoyl-4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperazine
3-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidine-1-carbonyl]benzonitrile
4-{[7-methoxy-2-(thiophen-2-yl)quinolin-3-yl]methyl}-1,3-dimethylpiperazin-2-one
2-(adamantan-1-ylsulfanyl)-1-(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
4-[3-(3-methylphenoxy)azetidine-1-carbonyl]benzene-1-sulfonamide
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl][(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]methylamine
(3aS,6aR)-5-cyclohexyl-3-[(3,4-dimethoxyphenyl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
4-(1,3-benzoxazol-2-yl)-N-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]piperidine-1-carboxamide
4-hydroxy-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(pyridin-2-yl)pyrimidine-5-carboxamide
(2S,4R)-N-(1,1-dioxo-1λ6-thian-4-yl)-N-methyl-4-(4-methylbenzamido)pyrrolidine-2-carboxamide
N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-2,3-dihydro-1,4-benzodioxine-5-carboxamide
3-{1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-4-yl)-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-cyclopropyl-5-({3-[3-(1-methyl-1H-imidazol-2-yl)phenyl]-1H-pyrazol-1-yl}methyl)-1,3,4-oxadiazole
4-hydroxy-1-[2-(morpholin-4-yl)-2-(pyridin-3-yl)acetyl]piperidine-4-carboxylic acid
1-[2-(2,3-difluoro-4-pentylphenyl)pyrimidin-4-yl]pyrrolidin-3-ol
5-(3-acetylphenoxymethyl)-N-(3-hydroxypropyl)-N-methyl-1,2-oxazole-3-carboxamide
(2-methoxyethyl)[(2E)-3-phenylprop-2-en-1-yl](1,3-thiazol-2-ylmethyl)amine