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2-(1H-imidazol-2-yl)-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]benzamide
ethyl 3-[(2E)-3-phenylprop-2-en-1-yl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxylate
6-({[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]amino}methyl)-1,4-oxazepan-6-ol
N-[(2-fluorophenyl)methyl]-2-{[2-methyl-1-(pyridin-2-yl)propyl]amino}acetamide
4-amino-1-[(3-fluorophenyl)methyl]pyrrolidin-2-one
2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]acetamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-5-yl]methyl}acetamide
N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
6,7-dimethoxy-2-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-1,2,3,4-tetrahydroisoquinoline
2-ethoxy-5-(2-{[2-(4-methyl-1,3-thiazol-2-yl)ethyl]amino}pyrimidin-4-yl)benzoic acid
N-(3-methoxyphenyl)-3-[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-4-yl]propanamide
2-(2-chlorophenyl)-5-(morpholin-2-ylmethyl)-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
1-(1-{1-[1-(2,3-dimethylphenyl)piperidin-4-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-2-ol
2-methyl-4-(4-{9-methyl-3,9-diazaspiro[5.6]dodecane-3-carbonyl}phenyl)but-3-yn-2-ol
N-ethyl-2-(3-methoxyphenoxymethyl)-N-(oxan-4-yl)-1,3-oxazole-4-carboxamide
(2S,4R)-4-(4-{[(3-methoxyphenyl)formamido]methyl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
(2S,4S)-N-[(2-chlorophenyl)methyl]-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
1-(2-methoxyethyl)-3,8-bis(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-N-{2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}thiophene-2-carboxamide
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-[3-(1H-pyrazol-1-yl)propyl]acetamide
1-[(4-fluorophenyl)methyl]-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(propan-2-yl)-1,4-diazepane
N4-methyl-N4-[(1-phenylpyrrolidin-3-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
4-{6-[1-(2-ethoxyethyl)piperidin-4-yl]-2-methylpyrimidin-4-yl}morpholine
1-[4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]hexan-1-one
N-cyclopropyl-N-[(2E)-3-phenylprop-2-en-1-yl]-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
1-[2-methoxy-4-({[2-(pyrazin-2-yl)ethyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
3-methyl-6-(3-{1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyridazine
2-[(2,4-dimethoxyphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-{3-[({[1-(ethoxymethyl)cyclobutyl]methyl}carbamoyl)amino]-4-fluorophenyl}acetamide
3-(1-benzyl-1H-imidazol-2-yl)-1-(2-methyl-1,3-thiazole-5-carbonyl)piperidine
2,5-dimethyl-3-(3-{1-[2-(pyrrolidin-1-yl)ethyl]-1H-pyrazol-3-yl}phenyl)pyrazine
6-methyl-2-({2-[5-(5-methylfuran-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}amino)-3,4-dihydropyrimidin-4-one
3-(1-benzofuran-2-yl)-2-methyl-6-(4H-1,2,4-triazol-4-yl)pyridine
3-{4-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]piperazin-1-yl}phenol
3-[(3R,4S)-1-(4-ethyl-5-methylthiophene-3-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(4-hydroxyphenyl)acetamide
4-{2-[3-(hydroxymethyl)-3-propylpiperidin-1-yl]-2-oxoethyl}-1λ6-thiane-1,1-dione
1-(adamantan-1-yl)-4-(5-cyclopropyl-1,3-oxazole-4-carbonyl)piperazine
2-(2-chloro-6-fluorophenyl)-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
1-(7-chloroquinolin-4-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-ethyl-2-(methylamino)-N-[(2E)-3-phenylprop-2-en-1-yl]pyrimidine-5-carboxamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazine
4-methyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-3,4-dihydro-2H-1,4-benzoxazine-2-carboxamide
(3S,4R)-3-methoxy-1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]piperidin-4-amine
methyl 1-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxylate
(3aS,6aR)-3-[2-(4-methoxyphenyl)ethyl]-5-(pyrrolidine-1-sulfonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
7-[3-(2-chlorophenyl)-5-methyl-1,2-oxazole-4-carbonyl]-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-6-methylpyridine-2-carboxamide
3-propyl-1-[2-(pyrrolidin-1-yl)acetyl]piperidine-3-carboxylic acid
N-[(1-methylpyrrolidin-3-yl)methyl]-5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole-3-carboxamide