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1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(3-fluorophenyl)ethan-1-one
N-ethyl-2-(2-methoxyphenyl)-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
2-{1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl}benzoic acid
(4aS,7aR)-1-[(6,8-dimethyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-ethyl-1-(4-methanesulfonylbenzoyl)piperidine-3-carboxylic acid
5-{[4-(1-methylpiperidin-4-yl)piperidin-1-yl]methyl}-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
N-{[2-(4-acetylpiperazin-1-yl)-6-methylquinolin-3-yl]methyl}-N-[2-(cyclohex-1-en-1-yl)ethyl]-2-(thiophen-3-yl)acetamide
2-[(2-chlorophenyl)methyl]-4-[4-(furan-3-ylmethyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
7-(3-methanesulfonylbenzoyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
5-[(2-methylpyrimidin-5-yl)methyl]-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(1R,5R)-6-(1-benzyl-1H-pyrazole-4-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
{3-[5-(1-ethyl-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]phenyl}methanol
4-(3-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}-3-oxopropyl)-N-methylbenzene-1-sulfonamide
N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}-1,3-benzothiazole-5-carboxamide
7-(1,3-benzothiazol-2-yl)-4-[(4-hydroxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-methyl-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide
5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]-2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}pyridine
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
1-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-5-oxopyrrolidine-3-carboxylic acid
6-{[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]sulfonyl}-1,3-dimethyl-1,2,3,4-tetrahydroquinazoline-2,4-dione
N-(2,3-dihydro-1H-inden-2-yl)-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}-N-propylacetamide
[(2,3-dimethoxyphenyl)methyl](methyl){[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}amine
2-{[methyl({[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl})amino]methyl}pyridine-3-carboxylic acid
N-methyl-5-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-carboxamide
N-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
1-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-phenylpyrrolidin-3-ol
1-{5-[5-(4-hydroxycyclohexyl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}butan-1-one
1-{4-[(3-phenylpropyl)amino]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
4-[(3-methoxyphenyl)methyl]-11-{[2-(propan-2-yloxy)ethyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-(3-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-3-oxopropyl)-4-methylbenzamide
1-methanesulfonyl-3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine
1-{4-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]phenyl}-1H-imidazole
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
methyl 3-benzamido-6-[(2-methylpiperidin-1-yl)methyl]thieno[2,3-b]pyridine-2-carboxylate
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-[(oxan-3-ylmethyl)amino]pyridine-3-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-8-[2-(propylsulfanyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[(3S,4R)-1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylimidazo[1,2-b]pyridazine-3-carboxamide
N-[4-(4-methoxyphenyl)butan-2-yl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-amino-4-(2-methoxypyrimidin-5-yl)-6-[4-(piperidin-1-yl)phenyl]pyridine-3-carbonitrile
2-({[(3R,4R)-1-[(2-fluoro-5-methoxyphenyl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-[2-(3-methyl-4H-1,2,4-triazol-4-yl)ethyl]-1,2-dihydroquinoxalin-2-one
(1S,5R)-6-(2-methoxyethyl)-3-(3-methyl-1-benzothiophene-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(3-methoxyphenyl)methyl]-2-{4-[2-(1H-1,2,4-triazol-1-yl)acetyl]morpholin-3-yl}acetamide
(1S,5R)-6-(cyclobutylmethyl)-3-(1-methyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methylbutanamide
4-(2,2-dimethyl-3-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}propyl)morpholine
N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrrolo[2,3-b]pyridin-6-amine