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3-({[(4-{1-azabicyclo[3.2.1]octan-5-yloxy}phenyl)methyl]amino}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-amino-1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2,3-dimethylbutan-1-one
(2S,4S)-4-amino-N-methyl-1-{[5-(1,3-oxazol-5-yl)thiophen-2-yl]sulfonyl}pyrrolidine-2-carboxamide
N-[1-(3-phenylpropyl)piperidin-3-yl]cyclopropanesulfonamide
6-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-(4-methoxyphenyl)-N-[4-(4-{[3-(1H-pyrazol-1-yl)propyl]amino}piperidin-1-yl)phenyl]acetamide
1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-4-(1,3-thiazol-2-yl)piperazine
1-(6-ethyl-2-methylquinoline-4-carbonyl)-4-(2-methylpropyl)-1,4-diazepan-5-one
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({methyl[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)piperidin-2-one
N-cyclohexyl-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-(thiophen-3-ylmethyl)propanamide
1-[3-(furan-2-yl)phenyl]-3-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-3-methylurea
(5-{1-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1H-imidazol-2-yl}furan-2-yl)methanol
N-benzyl-2-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-sulfonamide
1-ethyl-N-[2-(2-methoxyphenyl)ethyl]-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[(2S)-2-amino-3-hydroxypropanoyl]-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
1-methyl-4-[(2-{[4-(trifluoromethyl)pyridin-2-yl]oxy}phenyl)methyl]piperazine
2-(2-{[5-(3-methoxyphenyl)-1,2,4-triazin-3-yl]amino}ethyl)-6-phenyl-2,3-dihydropyridazin-3-one
N-{2-[(5-methyl-4-{[1-(thiophen-2-yl)propyl]amino}thieno[2,3-d]pyrimidin-6-yl)formamido]ethyl}acetamide
1-{3-oxo-3-[3-(3-phenylpropanoyl)piperidin-1-yl]propyl}-1,2-dihydropyridin-2-one
(1R,3S,5S)-8-[3-(4-hydroxyphenyl)benzoyl]-8-azabicyclo[3.2.1]octan-3-ol
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
1-({5-[(5-fluoro-2-methoxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
8-methyl-N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
1-(carbamoylmethyl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}piperidine-4-carboxamide
1-(4-ethenylphenyl)-3-methyl-3-(1-methylpyrrolidin-3-yl)urea
2-{[(butylcarbamoyl)methyl](methyl)amino}-2-(2-methoxy-5-methylphenyl)acetic acid
2-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-5-(trifluoromethyl)pyridine
4,6-dimethyl-2-{[5-(morpholin-4-ylmethyl)quinolin-8-yl]oxy}pyridine-3-carbonitrile
2-{5-[(phenylsulfanyl)methyl]furan-2-carbonyl}-1,2,3,4-tetrahydroisoquinolin-4-ol
(2S,4S)-4-amino-N,N-diethyl-1-(3-phenyl-1,2-oxazole-5-carbonyl)pyrrolidine-2-carboxamide
1-ethyl-1-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-3-[1-(1-phenylethyl)-1H-pyrazol-5-yl]urea
2-methyl-1-(4-{[2-(morpholin-4-yl)butyl]amino}piperidin-1-yl)propan-1-one
4-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]phenol
5-(2-methoxyphenoxymethyl)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-1,2-oxazole-3-carboxamide
N-{[2-(3-methylphenyl)-6-oxo-1,6-dihydropyrimidin-4-yl]methyl}acetamide
1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(3-methoxybenzoyl)piperazine
3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-{4-[(3-methylphenyl)methyl]piperazin-1-yl}propan-1-one
2-(4-{[2-(oxolan-3-yl)-1H-imidazol-1-yl]methyl}cyclohexyl)-1H-1,3-benzodiazole
N-(2-hydroxyethyl)-1-[1-(4-methylpyrimidin-2-yl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
1-(1-methylpiperidin-4-yl)-4-[2-(methylsulfanyl)benzoyl]piperazine
4-(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidin-4-yl)thiomorpholine
methyl[(5-methyl-1H-indazol-3-yl)methyl][2-(1H-pyrazol-4-yl)ethyl]amine
1-(3-methylpyridin-4-yl)-4-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperazine
3-(3-fluorophenyl)-4-(1H-imidazol-2-yl)-1-(4-methoxyphenyl)-1H-pyrazole
N-(2,2-dimethyloxan-4-yl)-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carboxamide
2,7-dimethyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}imidazo[1,2-a]pyridine-3-carboxamide
2-({3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)-3-methyl-1H-indole
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
4-(3-chloro-4-methylbenzoyl)-1-(2-methylphenyl)piperazin-2-one
6-methyl-5-[5-(3-methyl-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]-2-(2-methylpyridin-4-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine