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3-[(3R,4S)-1-[2-(3-hydroxyphenyl)acetyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
4-({3-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]phenyl}methyl)morpholine
5-{[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]methyl}-N-propylpyrimidin-2-amine
1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)ethan-1-one
7-(5-propyl-1,2-oxazole-4-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindole-2-carbonyl]-9-hydroxy-4H-pyrido[1,2-a]pyrimidin-4-one
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl][(1-ethyl-1H-indazol-3-yl)methyl]amine
2-methyl-5-({3-[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]propyl}sulfanyl)-1,3,4-thiadiazole
2-(2,3-dimethylphenyl)-5-(1H-imidazol-1-ylmethyl)pyridine
2-{[4-(2-methyl-1-benzothiophen-3-yl)-1H-1,2,3-triazol-1-yl]methyl}pyridine
N1-phenyl-N2-[7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]ethane-1,2-diamine
1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
5-{[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]sulfanyl}-1H-1,2,3-triazole
2-amino-4-(2-cyclohexylpyrimidin-5-yl)-5H,7H,8H-pyrano[4,3-b]pyridine-3-carbonitrile
2-methoxy-5-{[3-oxo-4-(2-phenylethyl)piperazin-1-yl]methyl}benzoic acid
1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}-2-(piperidin-1-yl)ethan-1-one
N-(pyridin-2-ylmethyl)-4-(1H-1,2,4-triazol-3-yl)benzamide
N-methyl-5-[(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)methyl]furan-2-carboxamide
6-[3-(2-hydroxyethyl)-4-[(6-methylpyridin-2-yl)methyl]piperazin-1-yl]pyridine-2-carbonitrile
1-[7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}propan-1-one
4-(4-chlorophenyl)-N-[2-(3-fluorophenyl)-2-hydroxyethyl]butanamide
5-[1-(furan-3-carbonyl)piperidin-4-yl]-5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
(4aS,8aR)-6-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
2-{1-[(3-chlorophenyl)methyl]-1H-1,2,4-triazol-5-yl}ethan-1-ol
N-(2-cyclopropylphenyl)-2-[4-ethyl-5-oxo-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide
1-{4-[3-(2-fluorophenoxy)azetidine-1-carbonyl]phenyl}-3,5-dimethyl-1H-pyrazole
1-methyl-3-phenyl-8-[2-(pyridin-2-yl)acetyl]-1,8-diazaspiro[4.5]decan-2-one
2-[1-(1,4-dithiepan-6-yl)piperidin-3-yl]-1,2,3,4-tetrahydroisoquinoline
7-[(3,4-difluorophenyl)methyl]-2-(6-methylpyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-ethyl-1-methyl-3-[1-(2-methyl-1H-1,3-benzodiazole-4-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(1-ethyl-1H-indazol-3-yl)-2-[4-methyl-3-(1-methyl-1H-pyrazol-4-yl)-1H-pyrazol-1-yl]acetamide
(3S,4S)-4-methyl-1-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)piperidine-3,4-diol
N-methyl-4-oxo-4-phenyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}butanamide
N-[(2-fluorophenyl)methyl]-N-propyl-1H-pyrrole-2-carboxamide
N-[(3S,4R)-3-benzyl-1-methylpiperidin-4-yl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
N-{2-[(2R)-pyrrolidin-2-yl]ethyl}-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
4-(3,5-dimethylbenzoyl)-5-methyl-1-(2-methylphenyl)piperazin-2-one
4-(naphthalen-2-ylmethyl)-1-(pyridine-2-carbonyl)-1,4-diazepan-5-one
3-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-(propan-2-yl)propanamide
N-[(3S,4R)-1-(2-amino-6-methoxypyrimidin-4-yl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
(3aS,7aR)-5-methyl-2-[2-(pyrrolidin-1-yl)benzoyl]-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
4-[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
[1-(2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carbonyl)-3-methylpiperidin-3-yl]methanol
N'1-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}cyclopropane-1,1-dicarboxamide
N-[1-(4-methyl-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]thiophene-2-carboxamide
2-({3-[hydroxy(phenyl)methyl]-1-(2-hydroxyethyl)-1H-1,2,4-triazol-5-yl}methyl)-5,6-dimethyl-2,3-dihydropyridazin-3-one
1-(4-methylpiperazin-1-yl)-3-[1-(1H-pyrazole-4-carbonyl)piperidin-3-yl]propan-1-one
2-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-N,N-dimethylquinoline-4-carboxamide
(4aS,8aR)-1-[3-(methylsulfanyl)propyl]-6-(oxan-4-yl)-decahydro-1,6-naphthyridin-2-one
7-fluoro-3-(2-methoxyethyl)-3,4-dihydroquinazolin-4-one