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N-{4-[2-(cyclopropylcarbamoyl)ethyl]phenyl}azocane-1-carboxamide
methyl({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}){[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}amine
2-{1-[(3-methoxyphenyl)methyl]-4-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-[(2-chloro-6-fluorophenyl)methyl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
ethyl 4-[(6-methoxyquinolin-8-yl)carbamoyl]piperazine-1-carboxylate
2-[1-(4-chlorophenyl)-3-(furan-2-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(2-hydroxypropyl)acetamide
1-amino-N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}cyclopropane-1-carboxamide
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-2-methyl-4-phenyl-1,3-thiazole-5-carboxamide
N-(5-chloro-2-methoxyphenyl)-4-[4-(2-hydroxyethyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
(2-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}quinolin-3-yl)methanol
1-(cyclopropylmethyl)-4-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-2-(propan-2-yl)-1,4-diazepane
(1S,5R)-3-[2-(benzenesulfonyl)ethyl]-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-({7-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-2-carboxamide
N-(2-methoxyethyl)-2,6-dimethyl-N-(1,3-thiazol-2-ylmethyl)quinoline-4-carboxamide
1-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-3-(trimethyl-1H-pyrazol-4-yl)urea
1-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-4-benzylpiperidin-4-ol
3-phenyl-1-[1-(2,4,5-trifluorobenzoyl)piperidin-3-yl]propan-1-one
(3S,5R)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
(1S,6R)-3-[5-(trifluoromethyl)pyridin-2-yl]-3,9-diazabicyclo[4.2.1]nonane
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
N-ethyl-2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(2-hydroxyethyl)acetamide
(2S,4S)-4-amino-1-(2,3-difluoro-4-methoxybenzoyl)-N-ethylpyrrolidine-2-carboxamide
1-[1-(6-methyl-2-phenylpyrimidin-4-yl)piperidin-4-yl]azepan-4-ol
N-(2-methoxyethyl)-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-amine
1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(dimethyl-1,2-oxazol-4-yl)propan-1-one
3-{2-[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-4-[(2-methoxyphenyl)methyl]piperazin-2-one
N-[(3-methyloxetan-3-yl)methyl]-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
6,6-dimethyl-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-5-oxothiomorpholine-3-carboxamide
2-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]-1-methyl-1H-indole
N,2-bis(cyclopropylmethyl)-7-(1H-imidazol-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N,N-dimethyl-4-{2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine-1-carboxamide
9-[3-(difluoromethoxy)benzoyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
N-[(2,3-dimethoxyphenyl)methyl]-N-ethyl-2-methylthieno[2,3-d]pyrimidin-4-amine
ethyl 1-cyclohexanecarbonyl-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylate
propan-2-yl 4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
4-(2-methoxyphenyl)-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidine
3-{1-[(3-chlorophenyl)methyl]piperidin-4-yl}-N-(2,3-dihydro-1,4-benzodioxin-6-yl)propanamide
2-{3-[3-(2-methylpyridin-4-yl)phenyl]-1H-pyrazol-1-yl}-1-(piperidin-1-yl)ethan-1-one
2-{5-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
(2S)-2-({5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazol-3-yl}formamido)propanamide
8-[(3-hydroxyphenyl)methyl]-1-(2-methoxyethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
9-(3-fluoropyridine-4-carbonyl)-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
N-[3-(4-fluorophenyl)phenyl]-3-(piperidin-1-yl)azetidine-1-carboxamide
4-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]-1-methylimidazolidin-2-one
2-chloro-4-({4-[(3,5-dimethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenol
1-(4-methyl-1,3-thiazol-2-yl)-4-(3-methylpyridin-4-yl)-1,4-diazepane
9-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecane
7-{[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
1,3-dimethyl-6-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione