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2-cyclopentyl-9-[(2-fluoro-3-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(4-aminoazepan-1-yl)-2-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]ethan-1-one
1-(6-hydroxy-1,4-oxazepan-4-yl)-2-methyl-2-(1H-pyrrol-1-yl)propan-1-one
3-(2-tert-butyl-1H-imidazol-1-yl)-2-methoxypyridine
methyl 8-(2,1,3-benzothiadiazol-5-ylmethyl)-1-methoxy-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
1-[2-methoxy-1-(pyridin-2-yl)ethyl]-1-methyl-3-(2-propylphenyl)urea
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(2-methanesulfonylethyl)pyrrolidine-3-carboxylic acid
7-(5-chloropyridin-2-yl)-4-(1-methyl-1H-pyrazole-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N,1-dimethyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-N-(1,3-thiazol-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-1,2,3-benzotriazole
1-methyl-2-oxo-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-1,2-dihydroquinoline-3-carboxamide
2-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoacetamide
[(2S,6S)-4-(4,6-dimethylpyrimidin-2-yl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
N-(2-hydroxyethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-3-propyl-1H-pyrazole-5-carboxamide
1-ethyl-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-6-oxopiperidine-3-carboxamide
(1S,5R)-6-[2-(3,4-dimethylphenoxy)ethyl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonane-7-carbonyl]-6-methoxy-1,4-dihydroquinolin-4-one
N-{[1-(1H-indol-2-ylmethyl)piperidin-3-yl]methyl}-3-methylbut-2-enamide
4-(2,5-dimethylfuran-3-carbonyl)-1-(1H-indazol-6-yl)piperazin-2-one
5-[(2-fluoro-5-methoxyphenyl)methyl]-5-{3-[3-(methoxymethyl)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(pyridin-2-ylmethyl)acetamide
1-[2-({[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]piperidin-4-ol
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-2-(2-methoxyphenyl)-N-methylacetamide
3-chloro-N-cyclopentyl-4-{[1-(3-acetamidopropanoyl)piperidin-4-yl]oxy}benzamide
N-cyclopentyl-2-{4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}propanamide
3-(ethylsulfamoyl)-N-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}benzamide
dimethyl(2-{4-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]morpholin-2-yl}ethyl)amine
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzamide
4-[3-(5-methylfuran-2-yl)butyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-3,4-dihydro-2H-1,4-benzothiazin-3-one
N-(2-hydroxyethyl)-5-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-benzyl-4-oxo-N-(propan-2-yl)-5-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl}-1,4-dihydropyridine-3-carboxamide
4-benzoyl-1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)piperidine
2-(4-acetylphenoxy)-N-(2-methoxyethyl)-N-(thiophen-3-ylmethyl)acetamide
3-{2-oxo-4-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperazin-1-yl}benzonitrile
N-(2-{2-methyl-1-azatricyclo[6.3.1.04,12]dodeca-2,4,6,8(12)-tetraen-3-yl}ethyl)-1,9-dioxaspiro[5.5]undecan-4-amine
(4aS,8aR)-6-(5-fluoropyridine-2-carbonyl)-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
3-[(4-tert-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine
2-(7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-2-yl)propane-1,3-diol
1-{4-[(2S)-2-(morpholine-4-carbonyl)pyrrolidine-1-carbonyl]thiophen-2-yl}ethan-1-one
N-[(3-methyl-1H-pyrazol-5-yl)methyl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(ethyl)(2-methylprop-2-en-1-yl)amine
methyl 5-[(1-hydroxypropan-2-yl)amino]-3-(2-methylbutanamido)-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
ethyl 1-[(2-ethoxy-2-oxoethyl)carbamoyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
2-(2,3-difluorophenyl)-1-[1-(furan-2-yl)ethyl]-1H-imidazole
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-3,5,7-trimethyl-1H-indole-2-carboxamide
3-(3-methyl-1H-1,2,4-triazol-5-yl)-N-(2-methylquinolin-8-yl)piperidine-1-carboxamide
4-(4-chlorophenyl)-1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}butan-1-one
1-ethyl-5-[2-(ethylamino)-4-methyl-1,3-thiazole-5-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid